O15075 DCLK1_HUMAN
Gene name: DCLK1
Protein name: Serine/threonine-protein kinase DCLK1

List of molecules and drugs that interact with protein O15075

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 O15075_AN2 AN2 n/a 448170;53813146; CHEMBL574810 AMP PHOSPHORAMIDATE n/a
2 O15075_GUI GUI n/a 16038120 CHEMBL509032 5-CHLORO-N-[2-METHOXY-4-[4-(4-METHYLPIPERAZIN-1-YL)PIPERIDIN-1-YL]PHENYL]-N'-(2-PROPAN-2-YLSULFONYLPHENYL)PYRIMIDINE-2,4-DIAMINE n/a
3 O15075_MG MG n/a 888 n/a MAGNESIUM ION n/a
4 O15075_PEG PEG n/a 8117 CHEMBL1235226 DI(HYDROXYETHYL)ETHER n/a
5 O15075_PG4 PG4 n/a 8200 CHEMBL1235254 TETRAETHYLENE GLYCOL n/a
6 O15075_RXT RXT DB08877 25126798 CHEMBL1789941 (3R)-3-cyclopentyl-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]propanenitrile n/a Kd(nM) = 68.0
7 O15075_X7Y X7Y n/a 46844147 CHEMBL1673039 2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6H-pyrimido[4,5-b][1,4]benzodiazepin-6-one n/a
8 O15075_X8J X8J n/a 134457974 CHEMBL4634326 5-ethyl-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-11-methyl-5,11-dihydro-6H-pyrimido[4,5-b][1,4]benzodiazepin-6-one n/a
9 O15075_XBD XBD n/a 134457640 CHEMBL4639395 2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-11-methyl-5-(2,2,2-trifluoroethyl)-5,11-dihydro-6H-pyrimido[4,5-b][1,4]benzodiazepin-6-one n/a
10 O15075_SO4 SO4 DB14546 1117 n/a SULFATE ION n/a
11 O15075_2RC 2RC DB12010 11671467 CHEMBL2103830 Fostamatinib inhibitor