P06213 INSR_HUMAN
Gene name: INSR
Protein name: Insulin receptor (IR)

List of molecules and drugs that interact with protein P06213

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 P06213_112 112 n/a 5287416 n/a THIOPHOSPHORIC ACID O-((ADENOSYL-PHOSPHO)PHOSPHO)-S-ACETAMIDYL-DIESTER n/a
2 P06213_351 351 n/a 25920884 CHEMBL563292 1-(3-{5-[4-(aminomethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-3-yl}phenyl)-3-(2-phenoxyphenyl)urea n/a
3 P06213_5JA 5JA n/a 91936978 CHEMBL5308290 (5R)-N-(1-{2-[4-(2-methoxyethyl)piperazin-1-yl]ethyl}-1H-pyrazol-3-yl)-5,8-dimethyl-9-phenyl-6,8-dihydro-5H-pyrazolo[3,4-h]quinazolin-2-amine n/a
4 P06213_60O 60O n/a n/a CHEMBL3786383 7-[3-(azetidin-1-ylmethyl)cyclobutyl]-5-[3-[[(2~{R})-oxan-2-yl]methoxy]phenyl]pyrrolo[2,3-d]pyrimidin-4-amine n/a
5 P06213_ACP ACP DB03909 91532 CHEMBL133463 PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTER inhibitor
6 P06213_ANP ANP n/a 33113 CHEMBL1230989 PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER n/a
7 P06213_ATP ATP DB00171 5957 CHEMBL14249 ADENOSINE-5'-TRIPHOSPHATE n/a
8 P06213_CA CA n/a 271 n/a CALCIUM ION n/a
9 P06213_EDO EDO n/a 174 CHEMBL457299 1,2-ETHANEDIOL n/a
10 P06213_EMC EMC n/a 5442 n/a ETHYL MERCURY ION n/a
11 P06213_GOL GOL DB09462 753 CHEMBL692 GLYCEROL n/a
12 P06213_GS2 GS2 n/a 25113169 n/a 2-[(2-{[1-(N,N-dimethylglycyl)-5-methoxy-1H-indol-6-yl]amino}-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-6-fluoro-N-methylbenzamide n/a
13 P06213_GS3 GS3 n/a 25113170 CHEMBL507625 2-fluoro-6-{[2-({2-methoxy-4-[4-(1-methylethyl)piperazin-1-yl]phenyl}amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide n/a
14 P06213_IR1 IR1 n/a 71660641 n/a 5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-3H-pyrazolo[3,4-c]pyridazin-3-one n/a
15 P06213_MG MG n/a 888 n/a MAGNESIUM ION n/a
16 P06213_MN MN n/a 27854 n/a MANGANESE (II) ION n/a
17 P06213_NAG NAG DB00141 24139 CHEMBL447878 2-acetamido-2-deoxy-beta-D-glucopyranose n/a
18 P06213_P33 P33 DB03394 79718 n/a 3,6,9,12,15,18-HEXAOXAICOSANE-1,20-DIOL n/a
19 P06213_S91 S91 DB08513 24871491 n/a [4-({5-(AMINOCARBONYL)-4-[(3-METHYLPHENYL)AMINO]PYRIMIDIN-2-YL}AMINO)PHENYL]ACETIC ACID n/a
20 P06213_SO4 SO4 DB14546 1117 n/a SULFATE ION n/a
21 P06213_DB06075 n/a DB06075 n/a n/a Linsitinib inhibitor
22 P06213_DB09129 n/a DB09129 n/a n/a Chromic chloride activator
23 P06213_2RC 2RC DB12010 11671467 CHEMBL2103830 Fostamatinib inhibitor
24 P06213_6GY 6GY DB12267 68165256 CHEMBL3545311 Brigatinib binding
25 P06213_EBI EBI DB15399 24785538 CHEMBL575448 BMS-754807 inhibitor
26 P06213_DB16637 n/a DB16637 n/a n/a KW-2450 free base inhibitor