Gene name: ABCB1
Protein name: ATP-dependent translocase ABCB1
List of molecules and drugs that interact with protein P08183
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | P08183_3PE | 3PE | n/a | 447078;15061530; | n/a | 1,2-Distearoyl-sn-glycerophosphoethanolamine | n/a | |
2 | P08183_ATP | ATP | DB00171 | 5957 | CHEMBL14249 | ADENOSINE-5'-TRIPHOSPHATE | n/a | |
3 | P08183_CLR | CLR | DB04540 | 5997 | CHEMBL112570 | CHOLESTEROL | n/a | |
4 | P08183_MG | MG | n/a | 888 | n/a | MAGNESIUM ION | n/a | |
5 | P08183_NAG | NAG | DB00141 | 24139 | CHEMBL447878 | 2-acetamido-2-deoxy-beta-D-glucopyranose | n/a | |
6 | P08183_R0Z | R0Z | DB04881 | 119373 | CHEMBL396298 | elacridar | inhibitor | Ki(nM) = 40.0 IC50(nM) = 4.9 EC50(nM) = 2000.0 |
7 | P08183_R1H | R1H | DB06240 | 148201 | CHEMBL348475 | tariquidar | modulator | |
8 | P08183_R1Q | R1Q | DB00541 | 5388993 | CHEMBL499458 | vincristine | n/a | Ki(nM) = 213000.0 |
9 | P08183_V5Q | V5Q | n/a | n/a | n/a | ~{N}-[2-[2-[4-[2-(6,7-dimethoxy-3,4-dihydro-1~{H}-isoquinolin-2-yl)ethyl]phenyl]-1,2,3,4-tetrazol-5-yl]-4,5-dimethoxy-phenyl]-4-oxidanylidene-2,3-dihydrochromene-2-carboxamide | n/a | |
10 | P08183_ZQU | ZQU | DB06191 | n/a | CHEMBL444172 | Zosuquidar | inhibitor | |
11 | P08183_TA1 | TA1 | DB01229 | 36314 | CHEMBL428647 | TAXOL | n/a | IC50(nM) = 2596.0 |
12 | P08183_DB00603 | n/a | DB00603 | n/a | n/a | Medroxyprogesterone acetate | inhibitor | |
13 | P08183_DB00661 | n/a | DB00661 | n/a | n/a | Verapamil | inhibitor | Ki(nM) = 880.0 IC50(nM) = 3.0 EC50(nM) = 120.0 |
14 | P08183_ROX | ROX | DB00778 | 6915744 | CHEMBL1214185 | Roxithromycin | n/a | |
15 | P08183_7V7 | 7V7 | DB00813 | 3345 | CHEMBL596 | Fentanyl | n/a | IC50(nM) = 6500.0 |
16 | P08183_DB04877 | n/a | DB04877 | n/a | n/a | Voacamine | inhibitor | |
17 | P08183_DB04905 | n/a | DB04905 | n/a | n/a | Tesmilifene | inducer | |
18 | P08183_DB09031 | n/a | DB09031 | n/a | n/a | Miltefosine | n/a | |
19 | P08183_QHM | QHM | DB14061 | 3634 | CHEMBL22077 | Hycanthone | inhibitor | |
20 | P08183_DB14062 | n/a | DB14062 | n/a | n/a | Concanamycin A | inhibitor | |
21 | P08183_I6H | I6H | DB14063 | 65808 | CHEMBL197 | Dexverapamil | inhibitor | |
22 | P08183_DB14064 | n/a | DB14064 | n/a | n/a | Emopamil | inhibitor | |
23 | P08183_DB14065 | n/a | DB14065 | n/a | n/a | Lomerizine | inhibitor | |
24 | P08183_DB14066 | n/a | DB14066 | n/a | n/a | Tetrandrine | inhibitor | |
25 | P08183_DB14067 | n/a | DB14067 | n/a | n/a | Dofequidar | inhibitor | |
26 | P08183_DB14068 | n/a | DB14068 | n/a | n/a | Dexniguldipine | inhibitor | |
27 | P08183_DB14069 | n/a | DB14069 | n/a | n/a | ONT-093 | inhibitor | |
28 | P08183_DB14070 | n/a | DB14070 | n/a | n/a | HM-30181 | inhibitor | |
29 | P08183_DB14071 | n/a | DB14071 | n/a | n/a | Desmethylsertraline | inhibitor | |
30 | P08183_DB14072 | n/a | DB14072 | n/a | n/a | Reversin 121 | inhibitor | |
31 | P08183_DB16407 | n/a | DB16407 | n/a | n/a | Azvudine | activator |