P09619 PGFRB_HUMAN
Gene name: PDGFRB
Protein name: Platelet-derived growth factor

List of molecules and drugs that interact with protein P09619

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 P09619_NAG NAG DB00141 24139 CHEMBL447878 2-acetamido-2-deoxy-beta-D-glucopyranose n/a
2 P09619_NDG NDG DB03740 82313 CHEMBL1234669 2-acetamido-2-deoxy-alpha-D-glucopyranose n/a
3 P09619_BAX BAX DB00398 216239 CHEMBL1336 Sorafenib inhibitor IC50(nM) = 0.26
Kd(nM) = 37.0
4 P09619_STI STI DB00619 5291 CHEMBL941 Imatinib antagonist Ki(nM) = 3.0
IC50(nM) = 50.0
Kd(nM) = 14.0
5 P09619_1N1 1N1 DB01254 3062316 CHEMBL1421 Dasatinib antagonist IC50(nM) = 28.0
Kd(nM) = 0.63
6 P09619_B49 B49 DB01268 5329102 CHEMBL535 Sunitinib inhibitor Ki(nM) = 8.0
IC50(nM) = 2.0
Kd(nM) = 0.075
7 P09619_DB06589 n/a DB06589 n/a n/a Pazopanib inhibitor IC50(nM) = 83.0
Kd(nM) = 2.0
8 P09619_2K2 2K2 DB06595 9829523 CHEMBL608533 Midostaurin antagonist
9 P09619_DB08896 n/a DB08896 n/a n/a Regorafenib inhibitor IC50(nM) = 1.5
10 P09619_XIN XIN DB09079 9809715 CHEMBL502835 Nintedanib inhibitor
11 P09619_DB09221 n/a DB09221 n/a n/a Polaprezinc agonist
12 P09619_K1S K1S DB09283 5531 CHEMBL132767 Trapidil antagonist
13 P09619_AV9 AV9 DB11800 9911830 CHEMBL1289494 Tivozanib inhibitor
14 P09619_2RC 2RC DB12010 11671467 CHEMBL2103830 Fostamatinib inhibitor
15 P09619_5SF 5SF DB12147 67462786 CHEMBL3545376 Erdafitinib substrate
16 P09619_P31 P31 DB12978 25151352 CHEMBL3813873 Pexidartinib inhibitor
17 P09619_DB14840 n/a DB14840 n/a n/a Ripretinib inhibitor
18 P09619_Q4J Q4J DB15822 n/a CHEMBL4297597 Pralsetinib inhibitor