Gene name: FGR
Protein name: Tyrosine-protein kinase Fgr
List of molecules and drugs that interact with protein P09769
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | P09769_CL | CL | n/a | 312 | n/a | CHLORIDE ION | n/a | |
2 | P09769_EDO | EDO | n/a | 174 | CHEMBL457299 | 1,2-ETHANEDIOL | n/a | |
3 | P09769_GOL | GOL | DB09462 | 753 | CHEMBL692 | GLYCEROL | n/a | |
4 | P09769_OJL | OJL | n/a | 71254350 | n/a | 3-[(6,7-dimethoxyquinazolin-4-yl)oxy]-N-{4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}-4-methylbenzamide | n/a | |
5 | P09769_PO4 | PO4 | DB14523 | 1061 | n/a | PHOSPHATE ION | n/a | |
6 | P09769_VSE | VSE | n/a | n/a | CHEMBL45177 | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine | n/a | |
7 | P09769_1N1 | 1N1 | DB01254 | 3062316 | CHEMBL1421 | Dasatinib | inhibitor | IC50(nM) = 10.0 Kd(nM) = 0.5 |
8 | P09769_2RC | 2RC | DB12010 | 11671467 | CHEMBL2103830 | Fostamatinib | inhibitor | |
9 | P09769_DB15035 | n/a | DB15035 | n/a | n/a | Zanubrutinib | inhibitor |