Gene name: ADORA3
Protein name: Adenosine receptor A3
List of molecules and drugs that interact with protein P0DMS8
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | P0DMS8_CFF | CFF | DB00201 | 2519 | CHEMBL113 | Caffeine | antagonist | Ki(nM) = 13300.0 IC50(nM) = 13300.0 |
2 | P0DMS8_ADN | ADN | DB00640 | 60961 | CHEMBL477 | Adenosine | agonist | Ki(nM) = 290.0 IC50(nM) = 1.1 Kd(nM) = 740.0 EC50(nM) = 13.0 |
3 | P0DMS8_DB00824 | n/a | DB00824 | n/a | n/a | Enprofylline | inhibitor | Ki(nM) = 10000.0 |
4 | P0DMS8_DB01223 | n/a | DB01223 | n/a | n/a | Aminophylline | antagonist | |
5 | P0DMS8_DB05511 | n/a | DB05511 | n/a | n/a | Piclidenoson | agonist | Ki(nM) = 0.215 IC50(nM) = 0.022909 EC50(nM) = 0.251189 |
6 | P0DMS8_2RC | 2RC | DB12010 | 11671467 | CHEMBL2103830 | Fostamatinib | antagonist |