P0DMS8 AA3R_HUMAN
Gene name: ADORA3
Protein name: Adenosine receptor A3

List of molecules and drugs that interact with protein P0DMS8

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 P0DMS8_CFF CFF DB00201 2519 CHEMBL113 Caffeine antagonist Ki(nM) = 13300.0
IC50(nM) = 13300.0
2 P0DMS8_ADN ADN DB00640 60961 CHEMBL477 Adenosine agonist Ki(nM) = 290.0
IC50(nM) = 1.1
Kd(nM) = 740.0
EC50(nM) = 13.0
3 P0DMS8_DB00824 n/a DB00824 n/a n/a Enprofylline inhibitor Ki(nM) = 10000.0
4 P0DMS8_DB01223 n/a DB01223 n/a n/a Aminophylline antagonist
5 P0DMS8_DB05511 n/a DB05511 n/a n/a Piclidenoson agonist Ki(nM) = 0.215
IC50(nM) = 0.022909
EC50(nM) = 0.251189
6 P0DMS8_2RC 2RC DB12010 11671467 CHEMBL2103830 Fostamatinib antagonist