P13569 CFTR_HUMAN
Gene name: CFTR
Protein name: Cystic fibrosis transmembrane

List of molecules and drugs that interact with protein P13569

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 P13569_AJP AJP n/a 6474107 n/a Digitonin n/a
2 P13569_ATP ATP DB00171 5957 CHEMBL14249 ADENOSINE-5'-TRIPHOSPHATE cofactor
3 P13569_B44 B44 n/a 11505398 n/a N-(2-phenylethyl)adenosine 5'-(tetrahydrogen triphosphate) n/a
4 P13569_C14 C14 n/a 12389 CHEMBL135488 TETRADECANE n/a
5 P13569_CLR CLR DB04540 5997 CHEMBL112570 CHOLESTEROL n/a
6 P13569_CTP CTP DB02431 6176 CHEMBL223533 CYTIDINE-5'-TRIPHOSPHATE n/a
7 P13569_CV6 CV6 DB11712 46199646 CHEMBL3544914 Tezacaftor positive allosteric modulator
8 P13569_D10 D10 n/a 15600 CHEMBL134537 DECANE n/a
9 P13569_D12 D12 n/a 8182 CHEMBL30959 DODECANE n/a
10 P13569_DCP DCP DB03258 65091 CHEMBL560403 2'-DEOXYCYTIDINE-5'-TRIPHOSPHATE n/a
11 P13569_DD9 DD9 n/a 8141 CHEMBL335900 nonane n/a
12 P13569_DGT DGT DB02181 65103;5280333;135398599; CHEMBL477486 2'-DEOXYGUANOSINE-5'-TRIPHOSPHATE n/a
13 P13569_DTP DTP DB03222 15993 CHEMBL335538 2'-DEOXYADENOSINE 5'-TRIPHOSPHATE n/a
14 P13569_DUT DUT DB02333 65070 CHEMBL374361 DEOXYURIDINE-5'-TRIPHOSPHATE n/a
15 P13569_GOL GOL DB09462 753 CHEMBL692 GLYCEROL n/a
16 P13569_GTP GTP DB04137 6830;5280317;135398633; CHEMBL1233147 GUANOSINE-5'-TRIPHOSPHATE n/a
17 P13569_LJP LJP DB16835 117857370 CHEMBL4075348 N-(3-carbamoyl-5,5,7,7-tetramethyl-4,7-dihydro-5H-thieno[2,3-c]pyran-2-yl)-1H-pyrazole-3-carboxamide n/a
18 P13569_M5T M5T n/a 451388 CHEMBL220940 5-Methyluridine triphosphate n/a
19 P13569_MG MG n/a 888 n/a MAGNESIUM ION n/a
20 P13569_MGP MGP DB02716 444378;5288806;135419182; CHEMBL1234303 7-METHYL-GUANOSINE-5'-TRIPHOSPHATE n/a
21 P13569_PJ8 PJ8 n/a 12398 CHEMBL3185332 heptadecane n/a
22 P13569_POV POV n/a 10908846 n/a (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate n/a
23 P13569_TTP TTP DB02452 64968 CHEMBL363559 THYMIDINE-5'-TRIPHOSPHATE n/a
24 P13569_UNX UNX n/a
25 P13569_UTP UTP DB04005 6133 CHEMBL336296 URIDINE 5'-TRIPHOSPHATE n/a
26 P13569_VX7 VX7 DB08820 16220172 CHEMBL2010601 N-(2,4-di-tert-butyl-5-hydroxyphenyl)-4-oxo-1,4-dihydroquinoline-3-carboxamide potentiator EC50(nM) = 3.0
27 P13569_VX8 VX8 DB09280 n/a CHEMBL2103870 Lumacaftor modulator
28 P13569_WJX WJX DB15444 134587348 CHEMBL4298128 (6P)-N-(1,3-dimethyl-1H-pyrazole-4-sulfonyl)-6-[3-(3,3,3-trifluoro-2,2-dimethylpropoxy)-1H-pyrazol-1-yl]-2-[(4S)-2,2,4-trimethylpyrrolidin-1-yl]pyridine-3-carboxamide positive allosteric modulator
29 P13569_82U 82U DB00887 2471 CHEMBL1072 Bumetanide antagonist
30 P13569_GBM GBM DB01016 3488 CHEMBL472 Glyburide antagonist IC50(nM) = 15000.0
31 P13569_DB01050 n/a DB01050 n/a n/a Ibuprofen inhibitor
32 P13569_GEN GEN DB01645 5280961 CHEMBL44 Genistein activator EC50(nM) = 6170.0
33 P13569_FOK FOK DB02587 47936 CHEMBL52606 Colforsin inhibitor
34 P13569_A0P A0P DB04395 44462678 n/a Phosphoaminophosphonic Acid-Adenylate Ester n/a
35 P13569_SEP SEP DB04522 68841;57689797; CHEMBL284377 Dexfosfoserine n/a
36 P13569_DB06266 n/a DB06266 n/a n/a Lonidamine n/a
37 P13569_IBP IBP DB09213 39912 CHEMBL175 Dexibuprofen inhibitor