Gene name: CFTR
Protein name: Cystic fibrosis transmembrane
List of molecules and drugs that interact with protein P13569
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | P13569_AJP | AJP | n/a | 6474107 | n/a | Digitonin | n/a | |
2 | P13569_ATP | ATP | DB00171 | 5957 | CHEMBL14249 | ADENOSINE-5'-TRIPHOSPHATE | cofactor | |
3 | P13569_B44 | B44 | n/a | 11505398 | n/a | N-(2-phenylethyl)adenosine 5'-(tetrahydrogen triphosphate) | n/a | |
4 | P13569_C14 | C14 | n/a | 12389 | CHEMBL135488 | TETRADECANE | n/a | |
5 | P13569_CLR | CLR | DB04540 | 5997 | CHEMBL112570 | CHOLESTEROL | n/a | |
6 | P13569_CTP | CTP | DB02431 | 6176 | CHEMBL223533 | CYTIDINE-5'-TRIPHOSPHATE | n/a | |
7 | P13569_CV6 | CV6 | DB11712 | 46199646 | CHEMBL3544914 | Tezacaftor | positive allosteric modulator | |
8 | P13569_D10 | D10 | n/a | 15600 | CHEMBL134537 | DECANE | n/a | |
9 | P13569_D12 | D12 | n/a | 8182 | CHEMBL30959 | DODECANE | n/a | |
10 | P13569_DCP | DCP | DB03258 | 65091 | CHEMBL560403 | 2'-DEOXYCYTIDINE-5'-TRIPHOSPHATE | n/a | |
11 | P13569_DD9 | DD9 | n/a | 8141 | CHEMBL335900 | nonane | n/a | |
12 | P13569_DGT | DGT | DB02181 | 65103;5280333;135398599; | CHEMBL477486 | 2'-DEOXYGUANOSINE-5'-TRIPHOSPHATE | n/a | |
13 | P13569_DTP | DTP | DB03222 | 15993 | CHEMBL335538 | 2'-DEOXYADENOSINE 5'-TRIPHOSPHATE | n/a | |
14 | P13569_DUT | DUT | DB02333 | 65070 | CHEMBL374361 | DEOXYURIDINE-5'-TRIPHOSPHATE | n/a | |
15 | P13569_GOL | GOL | DB09462 | 753 | CHEMBL692 | GLYCEROL | n/a | |
16 | P13569_GTP | GTP | DB04137 | 6830;5280317;135398633; | CHEMBL1233147 | GUANOSINE-5'-TRIPHOSPHATE | n/a | |
17 | P13569_LJP | LJP | DB16835 | 117857370 | CHEMBL4075348 | N-(3-carbamoyl-5,5,7,7-tetramethyl-4,7-dihydro-5H-thieno[2,3-c]pyran-2-yl)-1H-pyrazole-3-carboxamide | n/a | |
18 | P13569_M5T | M5T | n/a | 451388 | CHEMBL220940 | 5-Methyluridine triphosphate | n/a | |
19 | P13569_MG | MG | n/a | 888 | n/a | MAGNESIUM ION | n/a | |
20 | P13569_MGP | MGP | DB02716 | 444378;5288806;135419182; | CHEMBL1234303 | 7-METHYL-GUANOSINE-5'-TRIPHOSPHATE | n/a | |
21 | P13569_PJ8 | PJ8 | n/a | 12398 | CHEMBL3185332 | heptadecane | n/a | |
22 | P13569_POV | POV | n/a | 10908846 | n/a | (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate | n/a | |
23 | P13569_TTP | TTP | DB02452 | 64968 | CHEMBL363559 | THYMIDINE-5'-TRIPHOSPHATE | n/a | |
24 | P13569_UNX | UNX | n/a | |||||
25 | P13569_UTP | UTP | DB04005 | 6133 | CHEMBL336296 | URIDINE 5'-TRIPHOSPHATE | n/a | |
26 | P13569_VX7 | VX7 | DB08820 | 16220172 | CHEMBL2010601 | N-(2,4-di-tert-butyl-5-hydroxyphenyl)-4-oxo-1,4-dihydroquinoline-3-carboxamide | potentiator | EC50(nM) = 3.0 |
27 | P13569_VX8 | VX8 | DB09280 | n/a | CHEMBL2103870 | Lumacaftor | modulator | |
28 | P13569_WJX | WJX | DB15444 | 134587348 | CHEMBL4298128 | (6P)-N-(1,3-dimethyl-1H-pyrazole-4-sulfonyl)-6-[3-(3,3,3-trifluoro-2,2-dimethylpropoxy)-1H-pyrazol-1-yl]-2-[(4S)-2,2,4-trimethylpyrrolidin-1-yl]pyridine-3-carboxamide | positive allosteric modulator | |
29 | P13569_82U | 82U | DB00887 | 2471 | CHEMBL1072 | Bumetanide | antagonist | |
30 | P13569_GBM | GBM | DB01016 | 3488 | CHEMBL472 | Glyburide | antagonist | IC50(nM) = 15000.0 |
31 | P13569_DB01050 | n/a | DB01050 | n/a | n/a | Ibuprofen | inhibitor | |
32 | P13569_GEN | GEN | DB01645 | 5280961 | CHEMBL44 | Genistein | activator | EC50(nM) = 6170.0 |
33 | P13569_FOK | FOK | DB02587 | 47936 | CHEMBL52606 | Colforsin | inhibitor | |
34 | P13569_A0P | A0P | DB04395 | 44462678 | n/a | Phosphoaminophosphonic Acid-Adenylate Ester | n/a | |
35 | P13569_SEP | SEP | DB04522 | 68841;57689797; | CHEMBL284377 | Dexfosfoserine | n/a | |
36 | P13569_DB06266 | n/a | DB06266 | n/a | n/a | Lonidamine | n/a | |
37 | P13569_IBP | IBP | DB09213 | 39912 | CHEMBL175 | Dexibuprofen | inhibitor |