Gene name: ADRB3
Protein name: Beta-3 adrenergic receptor
List of molecules and drugs that interact with protein P13945
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | P13945_2GM | 2GM | DB00320 | 10531 | CHEMBL1732 | Dihydroergotamine | agonist | |
2 | P13945_LNR | LNR | DB00368 | 439260 | CHEMBL1437 | Norepinephrine | agonist | EC50(nM) = 5.5 |
3 | P13945_DB00571 | n/a | DB00571 | n/a | n/a | Propranolol | antagonist | Ki(nM) = 186.0 Kd(nM) = 117.0 |
4 | P13945_DB00866 | n/a | DB00866 | n/a | n/a | Alprenolol | antagonist | Ki(nM) = 35.0 Kd(nM) = 76.0 |
5 | P13945_DB00871 | n/a | DB00871 | n/a | n/a | Terbutaline | agonist | Ki(nM) = 10000.0 Kd(nM) = 125893.0 |
6 | P13945_DB00938 | n/a | DB00938 | n/a | n/a | Salmeterol | inverse agonist | Ki(nM) = 7180.0 Kd(nM) = 1862.0 EC50(nM) = 1000.0 |
7 | P13945_DB00960 | n/a | DB00960 | n/a | n/a | Pindolol | agonist | Ki(nM) = 44.1 Kd(nM) = 166.0 |
8 | P13945_DB00983 | n/a | DB00983 | n/a | n/a | Formoterol | agonist | Ki(nM) = 8090.0 EC50(nM) = 25.0 |
9 | P13945_DB01001 | n/a | DB01001 | n/a | n/a | Salbutamol | n/a | Ki(nM) = 10000.0 Kd(nM) = 46774.0 |
10 | P13945_DB01064 | n/a | DB01064 | n/a | n/a | Isoprenaline | agonist | Ki(nM) = 1570.0 EC50(nM) = 0.97 |
11 | P13945_DB01102 | n/a | DB01102 | n/a | n/a | Arbutamine | agonist | |
12 | P13945_DB01288 | n/a | DB01288 | n/a | n/a | Fenoterol | agonist | Ki(nM) = 10000.0 |
13 | P13945_DB01407 | n/a | DB01407 | n/a | n/a | Clenbuterol | agonist | |
14 | P13945_DB01580 | n/a | DB01580 | n/a | n/a | Oxprenolol | n/a | |
15 | P13945_DB04846 | n/a | DB04846 | n/a | n/a | Celiprolol | agonist | |
16 | P13945_DB04861 | n/a | DB04861 | n/a | n/a | Nebivolol | agonist | |
17 | P13945_DB05395 | n/a | DB05395 | n/a | n/a | Amibegron | agonist | |
18 | P13945_DB06190 | n/a | DB06190 | n/a | n/a | Solabegron | agonist | |
19 | P13945_DB06262 | n/a | DB06262 | n/a | n/a | Droxidopa | agonist | |
20 | P13945_DB08807 | n/a | DB08807 | n/a | n/a | Bopindolol | modulator | |
21 | P13945_DB08808 | n/a | DB08808 | n/a | n/a | Bupranolol | antagonist | Kd(nM) = 91.0 |
22 | P13945_H6U | H6U | DB08893 | 9865528 | CHEMBL2095212 | Mirabegron | agonist | |
23 | P13945_DB14895 | n/a | DB14895 | n/a | n/a | Vibegron | agonist |