P13945 ADRB3_HUMAN
Gene name: ADRB3
Protein name: Beta-3 adrenergic receptor

List of molecules and drugs that interact with protein P13945

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 P13945_2GM 2GM DB00320 10531 CHEMBL1732 Dihydroergotamine agonist
2 P13945_LNR LNR DB00368 439260 CHEMBL1437 Norepinephrine agonist EC50(nM) = 5.5
3 P13945_DB00571 n/a DB00571 n/a n/a Propranolol antagonist Ki(nM) = 186.0
Kd(nM) = 117.0
4 P13945_DB00866 n/a DB00866 n/a n/a Alprenolol antagonist Ki(nM) = 35.0
Kd(nM) = 76.0
5 P13945_DB00871 n/a DB00871 n/a n/a Terbutaline agonist Ki(nM) = 10000.0
Kd(nM) = 125893.0
6 P13945_DB00938 n/a DB00938 n/a n/a Salmeterol inverse agonist Ki(nM) = 7180.0
Kd(nM) = 1862.0
EC50(nM) = 1000.0
7 P13945_DB00960 n/a DB00960 n/a n/a Pindolol agonist Ki(nM) = 44.1
Kd(nM) = 166.0
8 P13945_DB00983 n/a DB00983 n/a n/a Formoterol agonist Ki(nM) = 8090.0
EC50(nM) = 25.0
9 P13945_DB01001 n/a DB01001 n/a n/a Salbutamol n/a Ki(nM) = 10000.0
Kd(nM) = 46774.0
10 P13945_DB01064 n/a DB01064 n/a n/a Isoprenaline agonist Ki(nM) = 1570.0
EC50(nM) = 0.97
11 P13945_DB01102 n/a DB01102 n/a n/a Arbutamine agonist
12 P13945_DB01288 n/a DB01288 n/a n/a Fenoterol agonist Ki(nM) = 10000.0
13 P13945_DB01407 n/a DB01407 n/a n/a Clenbuterol agonist
14 P13945_DB01580 n/a DB01580 n/a n/a Oxprenolol n/a
15 P13945_DB04846 n/a DB04846 n/a n/a Celiprolol agonist
16 P13945_DB04861 n/a DB04861 n/a n/a Nebivolol agonist
17 P13945_DB05395 n/a DB05395 n/a n/a Amibegron agonist
18 P13945_DB06190 n/a DB06190 n/a n/a Solabegron agonist
19 P13945_DB06262 n/a DB06262 n/a n/a Droxidopa agonist
20 P13945_DB08807 n/a DB08807 n/a n/a Bopindolol modulator
21 P13945_DB08808 n/a DB08808 n/a n/a Bupranolol antagonist Kd(nM) = 91.0
22 P13945_H6U H6U DB08893 9865528 CHEMBL2095212 Mirabegron agonist
23 P13945_DB14895 n/a DB14895 n/a n/a Vibegron agonist