Gene name: DRD4
Protein name: D(4) dopamine receptor
List of molecules and drugs that interact with protein P21917
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | P21917_AQD | AQD | DB19314 | 156333 | n/a | Nemonapride | n/a | |
2 | P21917_GOL | GOL | DB09462 | 753 | CHEMBL692 | GLYCEROL | n/a | |
3 | P21917_NA | NA | n/a | 923 | n/a | SODIUM ION | n/a | |
4 | P21917_OLA | OLA | n/a | 445639 | CHEMBL8659 | OLEIC ACID | n/a | |
5 | P21917_PEG | PEG | n/a | 8117 | CHEMBL1235226 | DI(HYDROXYETHYL)ETHER | n/a | |
6 | P21917_PO4 | PO4 | DB14523 | 1061 | n/a | PHOSPHATE ION | n/a | |
7 | P21917_DB00246 | n/a | DB00246 | n/a | n/a | Ziprasidone | antagonist | Ki(nM) = 0.8 |
8 | P21917_DB00248 | n/a | DB00248 | n/a | n/a | Cabergoline | agonist | |
9 | P21917_DB00268 | n/a | DB00268 | n/a | n/a | Ropinirole | agonist | Ki(nM) = 851.14 |
10 | P21917_2GM | 2GM | DB00320 | 10531 | CHEMBL1732 | Dihydroergotamine | agonist | |
11 | P21917_DB00334 | n/a | DB00334 | n/a | n/a | Olanzapine | antagonist | Ki(nM) = 20.0 IC50(nM) = 173.0 |
12 | P21917_DB00363 | n/a | DB00363 | n/a | n/a | Clozapine | antagonist | Ki(nM) = 7.27 IC50(nM) = 17.0 |
13 | P21917_DB00391 | n/a | DB00391 | n/a | n/a | Sulpiride | antagonist | Ki(nM) = 20.0 |
14 | P21917_DB00408 | n/a | DB00408 | n/a | n/a | Loxapine | binder | Ki(nM) = 4.3 IC50(nM) = 14.0 |
15 | P21917_DB00409 | n/a | DB00409 | n/a | n/a | Remoxipride | antagonist | Ki(nM) = 1000.0 IC50(nM) = 3872.0 |
16 | P21917_G6L | G6L | DB00413 | 119570 | CHEMBL301265 | Pramipexole | agonist | Ki(nM) = 1.3 EC50(nM) = 15.0 |
17 | P21917_Z80 | Z80 | DB00477 | 2726 | CHEMBL71 | Chlorpromazine | binder | Ki(nM) = 1.15 |
18 | P21917_DB00490 | n/a | DB00490 | n/a | n/a | Buspirone | antagonist | Ki(nM) = 78.0 |
19 | P21917_DB00543 | n/a | DB00543 | n/a | n/a | Amoxapine | antagonist | Ki(nM) = 2.0 |
20 | P21917_H8G | H8G | DB00589 | 28864 | CHEMBL157138 | Lisuride | agonist | Ki(nM) = 3.8 EC50(nM) = 89.0 |
21 | P21917_OR9 | OR9 | DB00714 | 6005 | CHEMBL53 | Apomorphine | agonist | Ki(nM) = 3.47 EC50(nM) = 1.5 |
22 | P21917_DB00875 | n/a | DB00875 | n/a | n/a | Flupentixol | antagonist | |
23 | P21917_LDP | LDP | DB00988 | 681 | CHEMBL59 | Dopamine | agonist | Ki(nM) = 1.2 IC50(nM) = 114.0 EC50(nM) = 1.8 |
24 | P21917_DB01186 | n/a | DB01186 | n/a | n/a | Pergolide | agonist | Ki(nM) = 53.2 |
25 | P21917_08Y | 08Y | DB01200 | 31101 | CHEMBL493 | Bromocriptine | antagonist | Ki(nM) = 285.0 |
26 | P21917_DB01224 | n/a | DB01224 | n/a | n/a | Quetiapine | ligand | Ki(nM) = 500.0 |
27 | P21917_DAH | DAH | DB01235 | 6047;6971033; | CHEMBL1009 | Levodopa | agonist | |
28 | P21917_9SC | 9SC | DB01238 | 60795 | CHEMBL1112 | Aripiprazole | antagonist | Ki(nM) = 44.0 |
29 | P21917_DB01267 | n/a | DB01267 | n/a | n/a | Paliperidone | antagonist | Ki(nM) = 30.0 |
30 | P21917_DB01403 | n/a | DB01403 | n/a | n/a | Methotrimeprazine | antagonist | |
31 | P21917_DB04908 | n/a | DB04908 | n/a | n/a | Flibanserin | antagonist | |
32 | P21917_DB04946 | n/a | DB04946 | n/a | n/a | Iloperidone | antagonist | Ki(nM) = 2.5 |
33 | P21917_DB05271 | n/a | DB05271 | n/a | n/a | Rotigotine | agonist | |
34 | P21917_DB06216 | n/a | DB06216 | n/a | n/a | Asenapine | antagonist | Ki(nM) = 3.8 |
35 | P21917_DB06477 | n/a | DB06477 | n/a | n/a | Sumanirole | n/a | |
36 | P21917_DB08922 | n/a | DB08922 | n/a | n/a | Perospirone | antagonist | |
37 | P21917_DB09286 | n/a | DB09286 | n/a | n/a | Pipamperone | antagonist | Ki(nM) = 5.1 |
38 | P21917_DB12061 | n/a | DB12061 | n/a | n/a | Pardoprunox | n/a | |
39 | P21917_DB14185 | n/a | DB14185 | n/a | n/a | Aripiprazole lauroxil | n/a |