P21917 DRD4_HUMAN
Gene name: DRD4
Protein name: D(4) dopamine receptor

List of molecules and drugs that interact with protein P21917

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 P21917_AQD AQD DB19314 156333 n/a Nemonapride n/a
2 P21917_GOL GOL DB09462 753 CHEMBL692 GLYCEROL n/a
3 P21917_NA NA n/a 923 n/a SODIUM ION n/a
4 P21917_OLA OLA n/a 445639 CHEMBL8659 OLEIC ACID n/a
5 P21917_PEG PEG n/a 8117 CHEMBL1235226 DI(HYDROXYETHYL)ETHER n/a
6 P21917_PO4 PO4 DB14523 1061 n/a PHOSPHATE ION n/a
7 P21917_DB00246 n/a DB00246 n/a n/a Ziprasidone antagonist Ki(nM) = 0.8
8 P21917_DB00248 n/a DB00248 n/a n/a Cabergoline agonist
9 P21917_DB00268 n/a DB00268 n/a n/a Ropinirole agonist Ki(nM) = 851.14
10 P21917_2GM 2GM DB00320 10531 CHEMBL1732 Dihydroergotamine agonist
11 P21917_DB00334 n/a DB00334 n/a n/a Olanzapine antagonist Ki(nM) = 20.0
IC50(nM) = 173.0
12 P21917_DB00363 n/a DB00363 n/a n/a Clozapine antagonist Ki(nM) = 7.27
IC50(nM) = 17.0
13 P21917_DB00391 n/a DB00391 n/a n/a Sulpiride antagonist Ki(nM) = 20.0
14 P21917_DB00408 n/a DB00408 n/a n/a Loxapine binder Ki(nM) = 4.3
IC50(nM) = 14.0
15 P21917_DB00409 n/a DB00409 n/a n/a Remoxipride antagonist Ki(nM) = 1000.0
IC50(nM) = 3872.0
16 P21917_G6L G6L DB00413 119570 CHEMBL301265 Pramipexole agonist Ki(nM) = 1.3
EC50(nM) = 15.0
17 P21917_Z80 Z80 DB00477 2726 CHEMBL71 Chlorpromazine binder Ki(nM) = 1.15
18 P21917_DB00490 n/a DB00490 n/a n/a Buspirone antagonist Ki(nM) = 78.0
19 P21917_DB00543 n/a DB00543 n/a n/a Amoxapine antagonist Ki(nM) = 2.0
20 P21917_H8G H8G DB00589 28864 CHEMBL157138 Lisuride agonist Ki(nM) = 3.8
EC50(nM) = 89.0
21 P21917_OR9 OR9 DB00714 6005 CHEMBL53 Apomorphine agonist Ki(nM) = 3.47
EC50(nM) = 1.5
22 P21917_DB00875 n/a DB00875 n/a n/a Flupentixol antagonist
23 P21917_LDP LDP DB00988 681 CHEMBL59 Dopamine agonist Ki(nM) = 1.2
IC50(nM) = 114.0
EC50(nM) = 1.8
24 P21917_DB01186 n/a DB01186 n/a n/a Pergolide agonist Ki(nM) = 53.2
25 P21917_08Y 08Y DB01200 31101 CHEMBL493 Bromocriptine antagonist Ki(nM) = 285.0
26 P21917_DB01224 n/a DB01224 n/a n/a Quetiapine ligand Ki(nM) = 500.0
27 P21917_DAH DAH DB01235 6047;6971033; CHEMBL1009 Levodopa agonist
28 P21917_9SC 9SC DB01238 60795 CHEMBL1112 Aripiprazole antagonist Ki(nM) = 44.0
29 P21917_DB01267 n/a DB01267 n/a n/a Paliperidone antagonist Ki(nM) = 30.0
30 P21917_DB01403 n/a DB01403 n/a n/a Methotrimeprazine antagonist
31 P21917_DB04908 n/a DB04908 n/a n/a Flibanserin antagonist
32 P21917_DB04946 n/a DB04946 n/a n/a Iloperidone antagonist Ki(nM) = 2.5
33 P21917_DB05271 n/a DB05271 n/a n/a Rotigotine agonist
34 P21917_DB06216 n/a DB06216 n/a n/a Asenapine antagonist Ki(nM) = 3.8
35 P21917_DB06477 n/a DB06477 n/a n/a Sumanirole n/a
36 P21917_DB08922 n/a DB08922 n/a n/a Perospirone antagonist
37 P21917_DB09286 n/a DB09286 n/a n/a Pipamperone antagonist Ki(nM) = 5.1
38 P21917_DB12061 n/a DB12061 n/a n/a Pardoprunox n/a
39 P21917_DB14185 n/a DB14185 n/a n/a Aripiprazole lauroxil n/a