P21918 DRD5_HUMAN
Gene name: DRD5
Protein name: D(1B) dopamine receptor

List of molecules and drugs that interact with protein P21918

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 P21918_DB00246 n/a DB00246 n/a n/a Ziprasidone antagonist
2 P21918_DB00248 n/a DB00248 n/a n/a Cabergoline agonist
3 P21918_DB00334 n/a DB00334 n/a n/a Olanzapine antagonist
4 P21918_DB00408 n/a DB00408 n/a n/a Loxapine binder
5 P21918_Z80 Z80 DB00477 2726 CHEMBL71 Chlorpromazine inhibitor Ki(nM) = 133.0
6 P21918_H8G H8G DB00589 28864 CHEMBL157138 Lisuride antagonist Ki(nM) = 77.0
7 P21918_OR9 OR9 DB00714 6005 CHEMBL53 Apomorphine agonist Ki(nM) = 14.79
8 P21918_DB00800 n/a DB00800 n/a n/a Fenoldopam agonist Ki(nM) = 15.0
9 P21918_LDP LDP DB00988 681 CHEMBL59 Dopamine agonist Ki(nM) = 228.0
EC50(nM) = 2.0
10 P21918_DB01038 n/a DB01038 n/a n/a Carphenazine antagonist
11 P21918_DB01186 n/a DB01186 n/a n/a Pergolide agonist Ki(nM) = 33.11
12 P21918_08Y 08Y DB01200 31101 CHEMBL493 Bromocriptine agonist Ki(nM) = 454.0
13 P21918_DB01224 n/a DB01224 n/a n/a Quetiapine ligand Ki(nM) = 1513.0
14 P21918_DAH DAH DB01235 6047;6971033; CHEMBL1009 Levodopa agonist
15 P21918_9SC 9SC DB01238 60795 CHEMBL1112 Aripiprazole antagonist Ki(nM) = 1051.0
16 P21918_DB01403 n/a DB01403 n/a n/a Methotrimeprazine antagonist
17 P21918_DB01624 n/a DB01624 n/a n/a Zuclopenthixol antagonist
18 P21918_DB05271 n/a DB05271 n/a n/a Rotigotine agonist Ki(nM) = 986.0
19 P21918_DB14185 n/a DB14185 n/a n/a Aripiprazole lauroxil n/a