Gene name: HRH2
Protein name: Histamine H2 receptor
List of molecules and drugs that interact with protein P25021
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | P25021_FO9 | FO9 | n/a | n/a | n/a | famotidine | n/a | |
2 | P25021_DB00272 | n/a | DB00272 | n/a | n/a | Betazole | agonist | |
3 | P25021_TP0 | TP0 | DB00321 | 2160 | CHEMBL629 | Amitriptyline | blocker | |
4 | P25021_DB00408 | n/a | DB00408 | n/a | n/a | Loxapine | binder | |
5 | P25021_C7H | C7H | DB00434 | 2913 | CHEMBL516 | Cyproheptadine | antagonist | |
6 | P25021_DB00501 | n/a | DB00501 | n/a | n/a | Cimetidine | antagonist | |
7 | P25021_DB00585 | n/a | DB00585 | n/a | n/a | Nizatidine | antagonist | |
8 | P25021_DB00751 | n/a | DB00751 | n/a | n/a | Epinastine | antagonist | |
9 | P25021_DB00768 | n/a | DB00768 | n/a | n/a | Olopatadine | antagonist | |
10 | P25021_DB00797 | n/a | DB00797 | n/a | n/a | Tolazoline | agonist | |
11 | P25021_DB00863 | n/a | DB00863 | n/a | n/a | Ranitidine | antagonist | Ki(nM) = 89.0 |
12 | P25021_DB00927 | n/a | DB00927 | n/a | n/a | Famotidine | antagonist | |
13 | P25021_DB00940 | n/a | DB00940 | n/a | n/a | Methantheline | antagonist | |
14 | P25021_DB00972 | n/a | DB00972 | n/a | n/a | Azelastine | inhibitor | |
15 | P25021_DB01069 | n/a | DB01069 | n/a | n/a | Promethazine | antagonist | |
16 | P25021_DB01142 | no_lig_id | DB01142 | n/a | n/a | Doxepin | antagonist | |
17 | P25021_9SC | 9SC | DB01238 | 60795 | CHEMBL1112 | Aripiprazole | ligand | Ki(nM) = 10000.0 |
18 | P25021_HSM | HSM | DB05381 | 774 | CHEMBL90 | Histamine | agonist | |
19 | P25021_DB06216 | n/a | DB06216 | n/a | n/a | Asenapine | antagonist | |
20 | P25021_DB08805 | n/a | DB08805 | n/a | n/a | Metiamide | antagonist | |
21 | P25021_DB08806 | n/a | DB08806 | n/a | n/a | Roxatidine acetate | antagonist | |
22 | P25021_DB09185 | n/a | DB09185 | n/a | n/a | Viloxazine | antagonist | |
23 | P25021_DB13760 | n/a | DB13760 | n/a | n/a | Niperotidine | antagonist |