Gene name: GRK2
Protein name: Beta-adrenergic receptor kinase
List of molecules and drugs that interact with protein P25098
| # | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
|---|---|---|---|---|---|---|---|---|
| 1 | P25098_1PE | 1PE | n/a | 62551 | CHEMBL1229766 | PENTAETHYLENE GLYCOL | n/a | |
| 2 | P25098_29X | 29X | n/a | 72706110 | n/a | 5-{[(3S,4R)-4-(4-fluorophenyl)piperidin-3-yl]methoxy}-1H-isoindol-1-one | n/a | |
| 3 | P25098_8DJ | 8DJ | n/a | 124160646 | CHEMBL4070885 | 5-[(3S,4R)-3-{[(2H-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluoro-N-[(pyridin-2-yl)methyl]benzamide | n/a | |
| 4 | P25098_8DS | 8DS | n/a | 156619967 | n/a | 4-chloranyl-N-[2-(4-chlorophenyl)ethyl]thieno[2,3-c]pyridine-2-carboxamide | n/a | |
| 5 | P25098_8PR | 8PR | DB00715 | 43815 | CHEMBL490 | Paroxetine | n/a | IC50(nM) = 1100.0 Kd(nM) = 2980.0 |
| 6 | P25098_8PV | 8PV | n/a | 11494718 | CHEMBL4082775 | N-benzyl-3-({[5-(pyridin-4-yl)-4H-1,2,4-triazol-3-yl]methyl}amino)benzamide | n/a | |
| 7 | P25098_AFM | AFM | n/a | 131953472 | n/a | 2-fluoro-5-[(3S,4R)-3-{[(1H-indazol-5-yl)oxy]methyl}piperidin-4-yl]-N-[(1H-pyrazol-3-yl)methyl]benzamide | n/a | |
| 8 | P25098_AFV | AFV | n/a | 131953473 | n/a | 2-fluoro-5-[(3S,4R)-3-{[(1H-indazol-5-yl)oxy]methyl}piperidin-4-yl]-N-[(pyridin-2-yl)methyl]benzamide | n/a | |
| 9 | P25098_BA1 | BA1 | DB04098 | 5287736;72200118; | CHEMBL60254 | BALANOL | n/a | |
| 10 | P25098_CL | CL | n/a | 312 | n/a | CHLORIDE ION | n/a | |
| 11 | P25098_EJS | EJS | n/a | 137349258 | n/a | (4R,5R,6S)-4-[4-fluoro-3-({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}carbamoyl)phenyl]-N-(2H-indazol-5-yl)-6-methyl-2-oxohexahydropyrimidine-5-carboxamide | n/a | |
| 12 | P25098_GOL | GOL | DB09462 | 753 | CHEMBL692 | GLYCEROL | n/a | |
| 13 | P25098_KZQ | KZQ | n/a | 117072130 | n/a | (4S)-4-(4-fluorophenyl)-N-(2H-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide | n/a | |
| 14 | P25098_MES | MES | DB03814 | 78165;4478249; | CHEMBL1234276 | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID | n/a | |
| 15 | P25098_MG | MG | n/a | 888 | n/a | MAGNESIUM ION | n/a | |
| 16 | P25098_Q1Y | Q1Y | n/a | 146019255 | CHEMBL5414047 | 5-[(3S,4R)-3-{[(2H-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluoro-N-[(2H-indazol-3-yl)methyl]benzamide | n/a | |
| 17 | P25098_QRW | QRW | n/a | 11677079 | CHEMBL1738877 | 3-({[4-methyl-5-(pyridin-4-yl)-4H-1,2,4-triazol-3-yl]methyl}amino)-N-[2-(trifluoromethyl)benzyl]benzamide | n/a | |
| 18 | P25098_SIX | SIX | n/a | 126456405 | CHEMBL4070290 | 2-{5-[(3S,4R)-3-{[(2H-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluorophenyl}-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide | n/a | |
| 19 | P25098_SO4 | SO4 | DB14546 | 1117 | n/a | SULFATE ION | n/a | |
| 20 | P25098_W4D | W4D | n/a | 154815729 | CHEMBL4740635 | 3-benzyl-6-(1H-pyrazol-4-yl)quinazolin-4(3H)-one | n/a | |
| 21 | P25098_W4G | W4G | n/a | 154815730 | CHEMBL4788026 | 3-benzyl-7-(1H-pyrazol-4-yl)quinazolin-4(3H)-one | n/a | |
| 22 | P25098_ZS2 | ZS2 | n/a | 118988618 | n/a | (4~{S})-4-[4-fluoranyl-3-(isoquinolin-1-ylmethylcarbamoyl)phenyl]-~{N}-(1~{H}-indazol-5-yl)-6-methyl-2-oxidanylidene-3,4-dihydro-1~{H}-pyrimidine-5-carboxamide | n/a | |
| 23 | P25098_ZSO | ZSO | n/a | 131953474 | n/a | 5-{[(3S,4R)-4-(4-fluorophenyl)piperidin-3-yl]methoxy}-2H-indazole | n/a | |
| 24 | P25098_ATP | ATP | DB00171 | 5957 | CHEMBL14249 | ATP | n/a |