Gene name: ADRA1D
Protein name: Alpha-1D adrenergic receptor
List of molecules and drugs that interact with protein P25100
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data | |
---|---|---|---|---|---|---|---|---|---|
1 | P25100_DB00211 | n/a | DB00211 | n/a | n/a | Midodrine | agonist | ||
2 | P25100_DB00248 | n/a | DB00248 | n/a | n/a | Cabergoline | binder | ||
3 | P25100_DB00298 | n/a | DB00298 | n/a | n/a | Dapiprazole | antagonist | ||
4 | P25100_TP0 | TP0 | DB00321 | 2160 | CHEMBL629 | Amitriptyline | antagonist | ||
5 | P25100_DB00346 | n/a | DB00346 | n/a | n/a | Alfuzosin | antagonist | Ki(nM) = 3.6 | |
6 | P25100_LNR | LNR | DB00368 | 439260 | CHEMBL1437 | Norepinephrine | agonist | ||
7 | P25100_DB00388 | n/a | DB00388 | n/a | n/a | Phenylephrine | agonist | ||
8 | P25100_XRA | XRA | DB00457 | 4893 | CHEMBL2 | Prazosin | n/a | antagonist | Ki(nM) = 0.06 |
9 | P25100_IXX | IXX | DB00458 | 3696 | CHEMBL11 | Imipramine | antagonist | ||
10 | P25100_21B | 21B | DB00540 | 4543 | CHEMBL445 | Nortriptyline | antagonist | ||
11 | P25100_CLU | CLU | DB00575 | 2803 | CHEMBL134 | Clonidine | agonist | ||
12 | P25100_DB00590 | n/a | DB00590 | n/a | n/a | Doxazosin | antagonist | Ki(nM) = 0.323594 | |
13 | P25100_DB00622 | n/a | DB00622 | n/a | n/a | Nicardipine | antagonist | ||
14 | P25100_DB00661 | n/a | DB00661 | n/a | n/a | Verapamil | antagonist | ||
15 | P25100_ALE | ALE | DB00668 | 5816;139148732; | CHEMBL679 | Epinephrine | antagonist | ||
16 | P25100_DB00692 | n/a | DB00692 | n/a | n/a | Phentolamine | antagonist | Ki(nM) = 7.6 IC50(nM) = 13.0 | |
17 | P25100_ERM | ERM | DB00696 | 8223 | CHEMBL442 | Ergotamine | partial agonist | ||
18 | P25100_DB00706 | n/a | DB00706 | n/a | n/a | Tamsulosin | antagonist | Ki(nM) = 0.056 IC50(nM) = 0.15 | |
19 | P25100_DB00723 | n/a | DB00723 | n/a | n/a | Methoxamine | binder | ||
20 | P25100_DB00800 | n/a | DB00800 | n/a | n/a | Fenoldopam | inhibitor | ||
21 | P25100_QDN | QDN | DB00908 | 441074 | CHEMBL1294 | Quinidine | antagonist | ||
22 | P25100_DB00925 | n/a | DB00925 | n/a | n/a | Phenoxybenzamine | antagonist | ||
23 | P25100_J5C | J5C | DB00935 | 4636 | CHEMBL762 | Oxymetazoline | agonist | Ki(nM) = 1349.0 EC50(nM) = 5012.0 | |
24 | P25100_DB01136 | n/a | DB01136 | n/a | n/a | Carvedilol | antagonist | ||
25 | P25100_DB01142 | no_lig_id | DB01142 | n/a | n/a | Doxepin | antagonist | ||
26 | P25100_DB01162 | n/a | DB01162 | n/a | n/a | Terazosin | antagonist | Ki(nM) = 0.66 | |
27 | P25100_DB01186 | n/a | DB01186 | n/a | n/a | Pergolide | agonist | Ki(nM) = 295.12 | |
28 | P25100_08Y | 08Y | DB01200 | 31101 | CHEMBL493 | Bromocriptine | agonist | Ki(nM) = 1.12 | |
29 | P25100_DB01403 | n/a | DB01403 | n/a | n/a | Methotrimeprazine | antagonist | ||
30 | P25100_DB04855 | n/a | DB04855 | n/a | n/a | Dronedarone | antagonist | ||
31 | P25100_NP1 | NP1 | DB05492 | 5276854 | CHEMBL609728 | Epicept NP-1 | n/a | ||
32 | P25100_DB06144 | n/a | DB06144 | n/a | n/a | Sertindole | n/a | ||
33 | P25100_DB06153 | n/a | DB06153 | n/a | n/a | Pizotifen | antagonist | ||
34 | P25100_DB06207 | n/a | DB06207 | n/a | n/a | Silodosin | antagonist | IC50(nM) = 6.3 | |
35 | P25100_DB06229 | n/a | DB06229 | n/a | n/a | Ocaperidone | n/a | ||
36 | P25100_DB06262 | n/a | DB06262 | n/a | n/a | Droxidopa | agonist | ||
37 | P25100_DB06694 | n/a | DB06694 | n/a | n/a | Xylometazoline | agonist | ||
38 | P25100_DB09202 | n/a | DB09202 | n/a | n/a | Cirazoline | partial agonist | EC50(nM) = 126.0 |