P25100 ADA1D_HUMAN
Gene name: ADRA1D
Protein name: Alpha-1D adrenergic receptor

List of molecules and drugs that interact with protein P25100

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 P25100_DB00211 n/a DB00211 n/a n/a Midodrine agonist
2 P25100_DB00248 n/a DB00248 n/a n/a Cabergoline binder
3 P25100_DB00298 n/a DB00298 n/a n/a Dapiprazole antagonist
4 P25100_TP0 TP0 DB00321 2160 CHEMBL629 Amitriptyline antagonist
5 P25100_DB00346 n/a DB00346 n/a n/a Alfuzosin antagonist Ki(nM) = 3.6
6 P25100_LNR LNR DB00368 439260 CHEMBL1437 Norepinephrine agonist
7 P25100_DB00388 n/a DB00388 n/a n/a Phenylephrine agonist
8 P25100_XRA XRA DB00457 4893 CHEMBL2 Prazosin n/a antagonist Ki(nM) = 0.06
9 P25100_IXX IXX DB00458 3696 CHEMBL11 Imipramine antagonist
10 P25100_21B 21B DB00540 4543 CHEMBL445 Nortriptyline antagonist
11 P25100_CLU CLU DB00575 2803 CHEMBL134 Clonidine agonist
12 P25100_DB00590 n/a DB00590 n/a n/a Doxazosin antagonist Ki(nM) = 0.323594
13 P25100_DB00622 n/a DB00622 n/a n/a Nicardipine antagonist
14 P25100_DB00661 n/a DB00661 n/a n/a Verapamil antagonist
15 P25100_ALE ALE DB00668 5816;139148732; CHEMBL679 Epinephrine antagonist
16 P25100_DB00692 n/a DB00692 n/a n/a Phentolamine antagonist Ki(nM) = 7.6
IC50(nM) = 13.0
17 P25100_ERM ERM DB00696 8223 CHEMBL442 Ergotamine partial agonist
18 P25100_DB00706 n/a DB00706 n/a n/a Tamsulosin antagonist Ki(nM) = 0.056
IC50(nM) = 0.15
19 P25100_DB00723 n/a DB00723 n/a n/a Methoxamine binder
20 P25100_DB00800 n/a DB00800 n/a n/a Fenoldopam inhibitor
21 P25100_QDN QDN DB00908 441074 CHEMBL1294 Quinidine antagonist
22 P25100_DB00925 n/a DB00925 n/a n/a Phenoxybenzamine antagonist
23 P25100_J5C J5C DB00935 4636 CHEMBL762 Oxymetazoline agonist Ki(nM) = 1349.0
EC50(nM) = 5012.0
24 P25100_DB01136 n/a DB01136 n/a n/a Carvedilol antagonist
25 P25100_DB01142 no_lig_id DB01142 n/a n/a Doxepin antagonist
26 P25100_DB01162 n/a DB01162 n/a n/a Terazosin antagonist Ki(nM) = 0.66
27 P25100_DB01186 n/a DB01186 n/a n/a Pergolide agonist Ki(nM) = 295.12
28 P25100_08Y 08Y DB01200 31101 CHEMBL493 Bromocriptine agonist Ki(nM) = 1.12
29 P25100_DB01403 n/a DB01403 n/a n/a Methotrimeprazine antagonist
30 P25100_DB04855 n/a DB04855 n/a n/a Dronedarone antagonist
31 P25100_NP1 NP1 DB05492 5276854 CHEMBL609728 Epicept NP-1 n/a
32 P25100_DB06144 n/a DB06144 n/a n/a Sertindole n/a
33 P25100_DB06153 n/a DB06153 n/a n/a Pizotifen antagonist
34 P25100_DB06207 n/a DB06207 n/a n/a Silodosin antagonist IC50(nM) = 6.3
35 P25100_DB06229 n/a DB06229 n/a n/a Ocaperidone n/a
36 P25100_DB06262 n/a DB06262 n/a n/a Droxidopa agonist
37 P25100_DB06694 n/a DB06694 n/a n/a Xylometazoline agonist
38 P25100_DB09202 n/a DB09202 n/a n/a Cirazoline partial agonist EC50(nM) = 126.0