Gene name: PTAFR
Protein name: Platelet-activating factor receptor
List of molecules and drugs that interact with protein P25105
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | P25105_9ER | 9ER | n/a | 119368 | CHEMBL1628662 | N1,N1-dimethyl-N2-[(pyridin-3-yl)methyl]-N2-{4-[2,4,6-tri(propan-2-yl)phenyl]-1,3-thiazol-2-yl}ethane-1,2-diamine | n/a | |
2 | P25105_9EU | 9EU | n/a | 154087 | CHEMBL369225 | 4-ethynyl-3-{3-fluoro-4-[(2-methyl-1H-imidazo[4,5-c]pyridin-1-yl)methyl]benzene-1-carbonyl}-N,N-dimethyl-1H-indole-1-carboxamide | n/a | |
3 | P25105_OLC | OLC | n/a | 11451146 | n/a | (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate | n/a | |
4 | P25105_ZN | ZN | n/a | 32051 | CHEMBL1236970 | ZINC ION | n/a | |
5 | P25105_SO4 | SO4 | DB14546 | 1117 | n/a | SULFATE ION | n/a | |
6 | P25105_PFS | PFS | DB02261 | 108156 | CHEMBL1235246 | Platelet Activating Factor | agonist | Ki(nM) = 0.15 IC50(nM) = 0.28 |
7 | P25105_DB09166 | n/a | DB09166 | n/a | n/a | Etizolam | antagonist | |
8 | P25105_DB11614 | n/a | DB11614 | n/a | n/a | Rupatadine | antagonist |