Gene name: HTR1D
Protein name: 5-hydroxytryptamine receptor 1D
List of molecules and drugs that interact with protein P28221
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | P28221_DB00216 | n/a | DB00216 | n/a | n/a | Eletriptan | agonist | |
2 | P28221_DB00246 | n/a | DB00246 | n/a | n/a | Ziprasidone | antagonist | Ki(nM) = 2.4 |
3 | P28221_DB00248 | n/a | DB00248 | n/a | n/a | Cabergoline | agonist | |
4 | P28221_DB00315 | n/a | DB00315 | n/a | n/a | Zolmitriptan | agonist | Ki(nM) = 0.4 IC50(nM) = 2.8 Kd(nM) = 1.5 |
5 | P28221_2GM | 2GM | DB00320 | 10531 | CHEMBL1732 | Dihydroergotamine | agonist | |
6 | P28221_TP0 | TP0 | DB00321 | 2160 | CHEMBL629 | Amitriptyline | binder | |
7 | P28221_DB00363 | n/a | DB00363 | n/a | n/a | Clozapine | antagonist | |
8 | P28221_DB00408 | n/a | DB00408 | n/a | n/a | Loxapine | binder | |
9 | P28221_DB00574 | n/a | DB00574 | n/a | n/a | Fenfluramine | agonist | |
10 | P28221_H8G | H8G | DB00589 | 28864 | CHEMBL157138 | Lisuride | agonist | Ki(nM) = 10000.0 |
11 | P28221_DB00669 | n/a | DB00669 | n/a | n/a | Sumatriptan | agonist | Ki(nM) = 0.5 IC50(nM) = 3.0 EC50(nM) = 4.3 |
12 | P28221_ERM | ERM | DB00696 | 8223 | CHEMBL442 | Ergotamine | agonist | Ki(nM) = 0.8 |
13 | P28221_OR9 | OR9 | DB00714 | 6005 | CHEMBL53 | Apomorphine | agonist | Ki(nM) = 1230.27 |
14 | P28221_DB00726 | n/a | DB00726 | n/a | n/a | Trimipramine | binder | |
15 | P28221_DB00734 | n/a | DB00734 | n/a | n/a | Risperidone | antagonist | Ki(nM) = 3.9 |
16 | P28221_DB00918 | n/a | DB00918 | n/a | n/a | Almotriptan | agonist | |
17 | P28221_J5C | J5C | DB00935 | 4636 | CHEMBL762 | Oxymetazoline | agonist | Ki(nM) = 0.4 EC50(nM) = 137.0 |
18 | P28221_DB00952 | n/a | DB00952 | n/a | n/a | Naratriptan | agonist | Ki(nM) = 1.5 EC50(nM) = 1.6 |
19 | P28221_DB00953 | n/a | DB00953 | n/a | n/a | Rizatriptan | agonist | Ki(nM) = 3.0 IC50(nM) = 11.0 EC50(nM) = 3.0 |
20 | P28221_DB00998 | n/a | DB00998 | n/a | n/a | Frovatriptan | agonist | Ki(nM) = 4.4 |
21 | P28221_DB01186 | n/a | DB01186 | n/a | n/a | Pergolide | agonist | Ki(nM) = 13.18 |
22 | P28221_08Y | 08Y | DB01200 | 31101 | CHEMBL493 | Bromocriptine | agonist | Ki(nM) = 10.72 |
23 | P28221_DB01224 | n/a | DB01224 | n/a | n/a | Quetiapine | ligand | Ki(nM) = 560.0 |
24 | P28221_9SC | 9SC | DB01238 | 60795 | CHEMBL1112 | Aripiprazole | antagonist | Ki(nM) = 68.0 |
25 | P28221_DB01267 | n/a | DB01267 | n/a | n/a | Paliperidone | antagonist | Ki(nM) = 19.0 |
26 | P28221_DB01392 | n/a | DB01392 | n/a | n/a | Yohimbine | partial agonist | Ki(nM) = 15.84 |
27 | P28221_DB04948 | n/a | DB04948 | n/a | n/a | Lofexidine | agonist | |
28 | P28221_DB14185 | n/a | DB14185 | n/a | n/a | Aripiprazole lauroxil | n/a |