P28221 5HT1D_HUMAN
Gene name: HTR1D
Protein name: 5-hydroxytryptamine receptor 1D

List of molecules and drugs that interact with protein P28221

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 P28221_DB00216 n/a DB00216 n/a n/a Eletriptan agonist
2 P28221_DB00246 n/a DB00246 n/a n/a Ziprasidone antagonist Ki(nM) = 2.4
3 P28221_DB00248 n/a DB00248 n/a n/a Cabergoline agonist
4 P28221_DB00315 n/a DB00315 n/a n/a Zolmitriptan agonist Ki(nM) = 0.4
IC50(nM) = 2.8
Kd(nM) = 1.5
5 P28221_2GM 2GM DB00320 10531 CHEMBL1732 Dihydroergotamine agonist
6 P28221_TP0 TP0 DB00321 2160 CHEMBL629 Amitriptyline binder
7 P28221_DB00363 n/a DB00363 n/a n/a Clozapine antagonist
8 P28221_DB00408 n/a DB00408 n/a n/a Loxapine binder
9 P28221_DB00574 n/a DB00574 n/a n/a Fenfluramine agonist
10 P28221_H8G H8G DB00589 28864 CHEMBL157138 Lisuride agonist Ki(nM) = 10000.0
11 P28221_DB00669 n/a DB00669 n/a n/a Sumatriptan agonist Ki(nM) = 0.5
IC50(nM) = 3.0
EC50(nM) = 4.3
12 P28221_ERM ERM DB00696 8223 CHEMBL442 Ergotamine agonist Ki(nM) = 0.8
13 P28221_OR9 OR9 DB00714 6005 CHEMBL53 Apomorphine agonist Ki(nM) = 1230.27
14 P28221_DB00726 n/a DB00726 n/a n/a Trimipramine binder
15 P28221_DB00734 n/a DB00734 n/a n/a Risperidone antagonist Ki(nM) = 3.9
16 P28221_DB00918 n/a DB00918 n/a n/a Almotriptan agonist
17 P28221_J5C J5C DB00935 4636 CHEMBL762 Oxymetazoline agonist Ki(nM) = 0.4
EC50(nM) = 137.0
18 P28221_DB00952 n/a DB00952 n/a n/a Naratriptan agonist Ki(nM) = 1.5
EC50(nM) = 1.6
19 P28221_DB00953 n/a DB00953 n/a n/a Rizatriptan agonist Ki(nM) = 3.0
IC50(nM) = 11.0
EC50(nM) = 3.0
20 P28221_DB00998 n/a DB00998 n/a n/a Frovatriptan agonist Ki(nM) = 4.4
21 P28221_DB01186 n/a DB01186 n/a n/a Pergolide agonist Ki(nM) = 13.18
22 P28221_08Y 08Y DB01200 31101 CHEMBL493 Bromocriptine agonist Ki(nM) = 10.72
23 P28221_DB01224 n/a DB01224 n/a n/a Quetiapine ligand Ki(nM) = 560.0
24 P28221_9SC 9SC DB01238 60795 CHEMBL1112 Aripiprazole antagonist Ki(nM) = 68.0
25 P28221_DB01267 n/a DB01267 n/a n/a Paliperidone antagonist Ki(nM) = 19.0
26 P28221_DB01392 n/a DB01392 n/a n/a Yohimbine partial agonist Ki(nM) = 15.84
27 P28221_DB04948 n/a DB04948 n/a n/a Lofexidine agonist
28 P28221_DB14185 n/a DB14185 n/a n/a Aripiprazole lauroxil n/a