Gene name: GRK1
Protein name: Rhodopsin kinase GRK1
List of molecules and drugs that interact with protein P28327
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | P28327_8PR | 8PR | DB00715 | 43815 | CHEMBL490 | Paroxetine | n/a | IC50(nM) = 100000.0 |
2 | P28327_ADP | ADP | DB16833 | 6022 | CHEMBL14830 | ADENOSINE-5'-DIPHOSPHATE | n/a | |
3 | P28327_ANW | ANW | DB01025 | 2161 | CHEMBL1096 | 2-amino-7-(1-methylethyl)-5-oxo-5H-chromeno[2,3-b]pyridine-3-carboxylic acid | n/a | |
4 | P28327_ATP | ATP | DB00171 | 5957 | CHEMBL14249 | ADENOSINE-5'-TRIPHOSPHATE | n/a | |
5 | P28327_BR | BR | n/a | 259 | n/a | BROMIDE ION | n/a | |
6 | P28327_CL | CL | n/a | 312 | n/a | CHLORIDE ION | n/a | |
7 | P28327_GOL | GOL | DB09462 | 753 | CHEMBL692 | GLYCEROL | n/a | |
8 | P28327_KQQ | KQQ | n/a | 25210972 | CHEMBL463931 | 3-[(2-{[1-(N,N-dimethylglycyl)-6-methoxy-4,4-dimethyl-1,2,3,4-tetrahydroquinolin-7-yl]amino}-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]thiophene-2-carboxamide | n/a | |
9 | P28327_MES | MES | DB03814 | 78165;4478249; | CHEMBL1234276 | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID | n/a | |
10 | P28327_MG | MG | n/a | 888 | n/a | MAGNESIUM ION | n/a | |
11 | P28327_SGV | SGV | n/a | 14978 | CHEMBL101892 | SANGIVAMYCIN | n/a |