P29275 AA2BR_HUMAN
Gene name: ADORA2B
Protein name: Adenosine receptor A2b

List of molecules and drugs that interact with protein P29275

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 P29275_ADN ADN DB00640 60961 CHEMBL477 ADENOSINE agonist EC50(nM) = 52.0
2 P29275_CLR CLR DB04540 5997 CHEMBL112570 CHOLESTEROL n/a
3 P29275_I5D I5D n/a 11717831 CHEMBL4202825 2-[6-azanyl-3,5-dicyano-4-[4-(cyclopropylmethoxy)phenyl]pyridin-2-yl]sulfanylethanamide n/a
4 P29275_CFF CFF DB00201 2519 CHEMBL113 Caffeine antagonist Ki(nM) = 10000.0
IC50(nM) = 10400.0
5 P29275_TEP TEP DB00277 2153 CHEMBL190 Theophylline antagonist Ki(nM) = 2700.0
6 P29275_DB00824 n/a DB00824 n/a n/a Enprofylline antagonist Ki(nM) = 4700.0
7 P29275_DB05936 n/a DB05936 n/a n/a CVT-6883 modulator