Gene name: AVPR2
Protein name: Vasopressin V2 receptor
List of molecules and drugs that interact with protein P30518
| # | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
|---|---|---|---|---|---|---|---|---|
| 1 | P30518_CLR | CLR | DB04540 | 5997 | CHEMBL112570 | CHOLESTEROL | n/a | |
| 2 | P30518_DB00035 | n/a | DB00035 | n/a | n/a | Desmopressin | agonist | |
| 3 | P30518_DB00067 | n/a | DB00067 | n/a | n/a | Vasopressin | agonist | |
| 4 | P30518_DB00618 | n/a | DB00618 | n/a | n/a | Demeclocycline | inhibitor | |
| 5 | P30518_DB00872 | n/a | DB00872 | n/a | n/a | Conivaptan | antagonist | Ki(nM) = 0.36 IC50(nM) = 11.0 |
| 6 | P30518_DB05838 | n/a | DB05838 | n/a | n/a | OPC-51803 | agonist | Ki(nM) = 92.0 IC50(nM) = 330.0 EC50(nM) = 189.0 |
| 7 | P30518_DB06212 | n/a | DB06212 | n/a | n/a | Tolvaptan | antagonist | |
| 8 | P30518_DB09059 | n/a | DB09059 | n/a | n/a | Atosiban | antagonist | |
| 9 | P30518_DB14642 | n/a | DB14642 | n/a | n/a | Lypressin | n/a | |
| 10 | P30518_DB16279 | n/a | DB16279 | n/a | n/a | Pecavaptan | antagonist |