Gene name: GNRHR
Protein name: Gonadotropin-releasing hormone receptor
List of molecules and drugs that interact with protein P30968
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | P30968_1QW | 1QW | n/a | 71598538 | n/a | (2R)-2,3-dihydroxypropyl dodecanoate | n/a | |
2 | P30968_F5O | F5O | DB11979 | 11250647 | CHEMBL1208155 | 4-[[(1R)-2-[5-(2-fluoranyl-3-methoxy-phenyl)-3-[[2-fluoranyl-6-(trifluoromethyl)phenyl]methyl]-4-methyl-2,6-bis(oxidanylidene)pyrimidin-1-yl]-1-phenyl-ethyl]amino]butanoic acid | antagonist | |
3 | P30968_FMT | FMT | DB01942 | 284;18971002; | CHEMBL116736 | FORMIC ACID | n/a | |
4 | P30968_OLC | OLC | n/a | 11451146 | n/a | (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate | n/a | |
5 | P30968_PEG | PEG | n/a | 8117 | CHEMBL1235226 | DI(HYDROXYETHYL)ETHER | n/a | |
6 | P30968_DB00007 | n/a | DB00007 | n/a | n/a | Leuprolide | agonist | |
7 | P30968_DB00014 | n/a | DB00014 | n/a | n/a | Goserelin | agonist | |
8 | P30968_DB00050 | n/a | DB00050 | n/a | n/a | Cetrorelix | antagonist | |
9 | P30968_DB00106 | n/a | DB00106 | n/a | n/a | Abarelix | antagonist | |
10 | P30968_DB00644 | n/a | DB00644 | n/a | n/a | Gonadorelin | agonist | |
11 | P30968_DB00666 | n/a | DB00666 | n/a | n/a | Nafarelin | agonist | |
12 | P30968_QA1 | QA1 | DB01406 | 28417 | CHEMBL1479 | Danazol | negative modulator | |
13 | P30968_DB05624 | n/a | DB05624 | n/a | n/a | Teverelix | antagonist | |
14 | P30968_DB06494 | n/a | DB06494 | n/a | n/a | Sufugolix | inhibitor | |
15 | P30968_DB06699 | n/a | DB06699 | n/a | n/a | Degarelix | antagonist | |
16 | P30968_DB06719 | n/a | DB06719 | n/a | n/a | Buserelin | n/a | |
17 | P30968_DB06785 | n/a | DB06785 | n/a | n/a | Ganirelix | antagonist | |
18 | P30968_DB06788 | n/a | DB06788 | n/a | n/a | Histrelin | agonist | |
19 | P30968_DB06825 | n/a | DB06825 | n/a | n/a | Triptorelin | agonist | |
20 | P30968_DB11619 | n/a | DB11619 | n/a | n/a | Gestrinone | antagonist | |
21 | P30968_DB11853 | n/a | DB11853 | n/a | n/a | Relugolix | antagonist | |
22 | P30968_DB17083 | n/a | DB17083 | n/a | n/a | Linzagolix | antagonist |