Gene name: CCKAR
Protein name: Cholecystokinin receptor type
List of molecules and drugs that interact with protein P32238
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | P32238_1OE | 1OE | DB04867 | 122077 | CHEMBL249973 | 2-[2-[[4-(2-chlorophenyl)-1,3-thiazol-2-yl]carbamoyl]indol-1-yl]ethanoic acid | antagonist | IC50(nM) = 0.56 |
2 | P32238_1OZ | 1OZ | n/a | 443375 | CHEMBL9506 | N-[(3S)-1-methyl-2-oxidanylidene-5-phenyl-3H-1,4-benzodiazepin-3-yl]-1H-indole-2-carboxamide | n/a | |
3 | P32238_IA1 | IA1 | n/a | 9852833 | CHEMBL3302616 | 2-[2-[[4-(4-chloranyl-2,5-dimethoxy-phenyl)-5-(2-cyclohexylethyl)-1,3-thiazol-2-yl]carbamoyl]-5,7-dimethyl-indol-1-yl]ethanoic acid | n/a | |
4 | P32238_Y01 | Y01 | n/a | 65082 | n/a | CHOLESTEROL HEMISUCCINATE | n/a | |
5 | P32238_DB00403 | n/a | DB00403 | n/a | n/a | Ceruletide | inducer | |
6 | P32238_DB04856 | n/a | DB04856 | n/a | n/a | Dexloxiglumide | inhibitor |