P32297 ACHA3_HUMAN
Gene name: CHRNA3
Protein name: Neuronal acetylcholine receptor

List of molecules and drugs that interact with protein P32297

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 P32297_DD9 DD9 n/a 8141 CHEMBL335900 nonane n/a
2 P32297_NA NA n/a 923 n/a SODIUM ION n/a
3 P32297_NAG NAG DB00141 24139 CHEMBL447878 2-acetamido-2-deoxy-beta-D-glucopyranose n/a
4 P32297_NCT NCT DB00184 89594 CHEMBL3 (S)-3-(1-METHYLPYRROLIDIN-2-YL)PYRIDINE agonist Ki(nM) = 5.0
5 P32297_P1M P1M n/a n/a n/a (3-endo)-N-(2-bromophenyl)-9-methyl-9-azabicyclo[3.3.1]nonan-3-amine n/a
6 P32297_Y01 Y01 n/a 65082 n/a CHOLESTEROL HEMISUCCINATE n/a
7 P32297_DB00333 n/a DB00333 n/a n/a Methadone antagonist
8 P32297_DB00472 n/a DB00472 n/a n/a Fluoxetine antagonist
9 P32297_DB00514 n/a DB00514 n/a n/a Dextromethorphan antagonist
10 P32297_DB00848 n/a DB00848 n/a n/a Levamisole agonist
11 P32297_EOH EOH DB00898 702 CHEMBL545 Ethanol n/a
12 P32297_DB00915 n/a DB00915 n/a n/a Amantadine antagonist
13 P32297_DB01090 n/a DB01090 n/a n/a Pentolinium antagonist
14 P32297_DB01156 n/a DB01156 n/a n/a Bupropion antagonist IC50(nM) = 1800.0
15 P32297_DB01227 n/a DB01227 n/a n/a Levacetylmethadol antagonist
16 P32297_QMR QMR DB01273 5310966 CHEMBL1076903 Varenicline partial agonist Ki(nM) = 40.0
17 P32297_DB05710 n/a DB05710 n/a n/a Gantacurium antagonist
18 P32297_EPJ EPJ DB07720 854023 CHEMBL298826 Epibatidine agonist Ki(nM) = 0.15
Kd(nM) = 0.3
19 P32297_C5E C5E DB09028 10235 CHEMBL497939 Cytisine agonist EC50(nM) = 26000.0