Gene name: HTR7
Protein name: 5-hydroxytryptamine receptor 7
List of molecules and drugs that interact with protein P34969
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | P34969_DB00246 | n/a | DB00246 | n/a | n/a | Ziprasidone | antagonist | Ki(nM) = 5.0 |
2 | P34969_DB00247 | n/a | DB00247 | n/a | n/a | Methysergide | antagonist | |
3 | P34969_DB00248 | n/a | DB00248 | n/a | n/a | Cabergoline | antagonist | |
4 | P34969_DB00315 | n/a | DB00315 | n/a | n/a | Zolmitriptan | agonist | |
5 | P34969_TP0 | TP0 | DB00321 | 2160 | CHEMBL629 | Amitriptyline | antagonist | |
6 | P34969_DB00363 | n/a | DB00363 | n/a | n/a | Clozapine | antagonist | Ki(nM) = 9.0 |
7 | P34969_DB00408 | n/a | DB00408 | n/a | n/a | Loxapine | binder | Ki(nM) = 87.2 |
8 | P34969_C7H | C7H | DB00434 | 2913 | CHEMBL516 | Cyproheptadine | antagonist | Ki(nM) = 50.0 |
9 | P34969_IXX | IXX | DB00458 | 3696 | CHEMBL11 | Imipramine | antagonist | Ki(nM) = 1000.0 |
10 | P34969_Z80 | Z80 | DB00477 | 2726 | CHEMBL71 | Chlorpromazine | binder | Ki(nM) = 11.0 |
11 | P34969_GMJ | GMJ | DB00502 | 3559 | CHEMBL54 | Haloperidol | n/a | Ki(nM) = 316.0 |
12 | P34969_DB00543 | n/a | DB00543 | n/a | n/a | Amoxapine | antagonist | Ki(nM) = 500.0 |
13 | P34969_H8G | H8G | DB00589 | 28864 | CHEMBL157138 | Lisuride | n/a | Ki(nM) = 6.8 |
14 | P34969_DB00734 | n/a | DB00734 | n/a | n/a | Risperidone | antagonist | Ki(nM) = 0.4 |
15 | P34969_DB00751 | n/a | DB00751 | n/a | n/a | Epinastine | antagonist | |
16 | P34969_DB00924 | n/a | DB00924 | n/a | n/a | Cyclobenzaprine | antagonist | |
17 | P34969_DB00934 | n/a | DB00934 | n/a | n/a | Maprotiline | antagonist | |
18 | P34969_LDP | LDP | DB00988 | 681 | CHEMBL59 | Dopamine | binder | Ki(nM) = 10000.0 |
19 | P34969_08Y | 08Y | DB01200 | 31101 | CHEMBL493 | Bromocriptine | antagonist | |
20 | P34969_DB01224 | n/a | DB01224 | n/a | n/a | Quetiapine | ligand | Ki(nM) = 63.0 |
21 | P34969_9SC | 9SC | DB01238 | 60795 | CHEMBL1112 | Aripiprazole | antagonist | Ki(nM) = 9.6 |
22 | P34969_DB01267 | n/a | DB01267 | n/a | n/a | Paliperidone | n/a | |
23 | P34969_DB04946 | n/a | DB04946 | n/a | n/a | Iloperidone | antagonist | Ki(nM) = 112.0 |
24 | P34969_DB04948 | n/a | DB04948 | n/a | n/a | Lofexidine | agonist | |
25 | P34969_DB06148 | n/a | DB06148 | n/a | n/a | Mianserin | antagonist | |
26 | P34969_DB06216 | n/a | DB06216 | n/a | n/a | Asenapine | antagonist | |
27 | P34969_DB06288 | n/a | DB06288 | n/a | n/a | Amisulpride | antagonist | Ki(nM) = 11.5 |
28 | P34969_DB08815 | n/a | DB08815 | n/a | n/a | Lurasidone | antagonist | Ki(nM) = 0.5 IC50(nM) = 16.0 |
29 | P34969_DB09068 | n/a | DB09068 | n/a | n/a | Vortioxetine | antagonist | |
30 | P34969_ZOT | ZOT | DB09225 | 5736 | CHEMBL285802 | Zotepine | antagonist | |
31 | P34969_DB13988 | n/a | DB13988 | n/a | n/a | SB-269970 | antagonist | |
32 | P34969_DB14185 | n/a | DB14185 | n/a | n/a | Aripiprazole lauroxil | n/a |