P34969 5HT7R_HUMAN
Gene name: HTR7
Protein name: 5-hydroxytryptamine receptor 7

List of molecules and drugs that interact with protein P34969

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 P34969_DB00246 n/a DB00246 n/a n/a Ziprasidone antagonist Ki(nM) = 5.0
2 P34969_DB00247 n/a DB00247 n/a n/a Methysergide antagonist
3 P34969_DB00248 n/a DB00248 n/a n/a Cabergoline antagonist
4 P34969_DB00315 n/a DB00315 n/a n/a Zolmitriptan agonist
5 P34969_TP0 TP0 DB00321 2160 CHEMBL629 Amitriptyline antagonist
6 P34969_DB00363 n/a DB00363 n/a n/a Clozapine antagonist Ki(nM) = 9.0
7 P34969_DB00408 n/a DB00408 n/a n/a Loxapine binder Ki(nM) = 87.2
8 P34969_C7H C7H DB00434 2913 CHEMBL516 Cyproheptadine antagonist Ki(nM) = 50.0
9 P34969_IXX IXX DB00458 3696 CHEMBL11 Imipramine antagonist Ki(nM) = 1000.0
10 P34969_Z80 Z80 DB00477 2726 CHEMBL71 Chlorpromazine binder Ki(nM) = 11.0
11 P34969_GMJ GMJ DB00502 3559 CHEMBL54 Haloperidol n/a Ki(nM) = 316.0
12 P34969_DB00543 n/a DB00543 n/a n/a Amoxapine antagonist Ki(nM) = 500.0
13 P34969_H8G H8G DB00589 28864 CHEMBL157138 Lisuride n/a Ki(nM) = 6.8
14 P34969_DB00734 n/a DB00734 n/a n/a Risperidone antagonist Ki(nM) = 0.4
15 P34969_DB00751 n/a DB00751 n/a n/a Epinastine antagonist
16 P34969_DB00924 n/a DB00924 n/a n/a Cyclobenzaprine antagonist
17 P34969_DB00934 n/a DB00934 n/a n/a Maprotiline antagonist
18 P34969_LDP LDP DB00988 681 CHEMBL59 Dopamine binder Ki(nM) = 10000.0
19 P34969_08Y 08Y DB01200 31101 CHEMBL493 Bromocriptine antagonist
20 P34969_DB01224 n/a DB01224 n/a n/a Quetiapine ligand Ki(nM) = 63.0
21 P34969_9SC 9SC DB01238 60795 CHEMBL1112 Aripiprazole antagonist Ki(nM) = 9.6
22 P34969_DB01267 n/a DB01267 n/a n/a Paliperidone n/a
23 P34969_DB04946 n/a DB04946 n/a n/a Iloperidone antagonist Ki(nM) = 112.0
24 P34969_DB04948 n/a DB04948 n/a n/a Lofexidine agonist
25 P34969_DB06148 n/a DB06148 n/a n/a Mianserin antagonist
26 P34969_DB06216 n/a DB06216 n/a n/a Asenapine antagonist
27 P34969_DB06288 n/a DB06288 n/a n/a Amisulpride antagonist Ki(nM) = 11.5
28 P34969_DB08815 n/a DB08815 n/a n/a Lurasidone antagonist Ki(nM) = 0.5
IC50(nM) = 16.0
29 P34969_DB09068 n/a DB09068 n/a n/a Vortioxetine antagonist
30 P34969_ZOT ZOT DB09225 5736 CHEMBL285802 Zotepine antagonist
31 P34969_DB13988 n/a DB13988 n/a n/a SB-269970 antagonist
32 P34969_DB14185 n/a DB14185 n/a n/a Aripiprazole lauroxil n/a