P35916 VGFR3_HUMAN
Gene name: FLT4
Protein name: Vascular endothelial growth

List of molecules and drugs that interact with protein P35916

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 P35916_NAG NAG DB00141 24139 CHEMBL447878 2-acetamido-2-deoxy-beta-D-glucopyranose n/a
2 P35916_BAX BAX DB00398 216239 CHEMBL1336 Sorafenib inhibitor IC50(nM) = 3.0
Kd(nM) = 16.0
3 P35916_B49 B49 DB01268 5329102 CHEMBL535 Sunitinib inhibitor Ki(nM) = 17.0
IC50(nM) = 8.9
Kd(nM) = 35.0
4 P35916_DB04879 n/a DB04879 n/a n/a Vatalanib inhibitor IC50(nM) = 64.0
Kd(nM) = 190.0
5 P35916_DB05075 n/a DB05075 n/a n/a TG-100801 n/a
6 P35916_DB05932 n/a DB05932 n/a n/a Denibulin n/a
7 P35916_DB06080 n/a DB06080 n/a n/a Linifanib modulator
8 P35916_DB06589 n/a DB06589 n/a n/a Pazopanib inhibitor IC50(nM) = 46.0
Kd(nM) = 27.0
9 P35916_AXI AXI DB06626 6450551 CHEMBL1289926 Axitinib inhibitor
10 P35916_DB08896 n/a DB08896 n/a n/a Regorafenib inhibitor IC50(nM) = 10.0
11 P35916_LEV LEV DB09078 9823820 CHEMBL1289601 Lenvatinib inhibitor
12 P35916_XIN XIN DB09079 9809715 CHEMBL502835 Nintedanib inhibitor
13 P35916_AV9 AV9 DB11800 9911830 CHEMBL1289494 Tivozanib inhibitor
14 P35916_2RC 2RC DB12010 11671467 CHEMBL2103830 Fostamatinib inhibitor
15 P35916_DB15685 n/a DB15685 n/a n/a Selpercatinib inhibitor