Gene name: AVPR1A
Protein name: Vasopressin V1a receptor
List of molecules and drugs that interact with protein P37288
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | P37288_DB00035 | n/a | DB00035 | n/a | n/a | Desmopressin | agonist | |
2 | P37288_DB00067 | n/a | DB00067 | n/a | n/a | Vasopressin | agonist | |
3 | P37288_DB00872 | n/a | DB00872 | n/a | n/a | Conivaptan | antagonist | Ki(nM) = 0.43 IC50(nM) = 3.0 |
4 | P37288_DB06212 | n/a | DB06212 | n/a | n/a | Tolvaptan | antagonist | |
5 | P37288_DB09059 | n/a | DB09059 | n/a | n/a | Atosiban | antagonist | |
6 | P37288_DB13929 | n/a | DB13929 | n/a | n/a | Relcovaptan | antagonist | |
7 | P37288_DB14642 | n/a | DB14642 | n/a | n/a | Lypressin | n/a | |
8 | P37288_DB16279 | n/a | DB16279 | n/a | n/a | Pecavaptan | antagonist |