P42261 GRIA1_HUMAN
Gene name: GRIA1
Protein name: Glutamate receptor 1

List of molecules and drugs that interact with protein P42261

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 P42261_GGL GGL DB00142 33032;44272391;88747398; CHEMBL575060 Glutamic acid n/a Ki(nM) = 1360.0
EC50(nM) = 2260.0
2 P42261_DB00237 n/a DB00237 n/a n/a Butabarbital antagonist
3 P42261_DB00555 n/a DB00555 n/a n/a Lamotrigine inhibitor
4 P42261_DB00753 n/a DB00753 n/a n/a Isoflurane antagonist
5 P42261_EOH EOH DB00898 702 CHEMBL545 Ethanol n/a
6 P42261_DB01028 n/a DB01028 n/a n/a Methoxyflurane antagonist
7 P42261_DB01189 n/a DB01189 n/a n/a Desflurane antagonist
8 P42261_DB01236 n/a DB01236 n/a n/a Sevoflurane antagonist
9 P42261_DB04982 n/a DB04982 n/a n/a Talampanel n/a
10 P42261_DB05047 n/a DB05047 n/a n/a CX-717 n/a
11 P42261_CX5 CX5 DB06247 148184 CHEMBL136800 CX516 n/a
12 P42261_6ZP 6ZP DB08883 9924495 CHEMBL1214124 Perampanel antagonist
13 P42261_DB09289 n/a DB09289 n/a n/a Tianeptine modulator
14 P42261_DB13146 n/a DB13146 n/a n/a Fluciclovine (18F) inhibitor