Gene name: GRIA1
Protein name: Glutamate receptor 1
List of molecules and drugs that interact with protein P42261
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | P42261_GGL | GGL | DB00142 | 33032;44272391;88747398; | CHEMBL575060 | Glutamic acid | n/a | Ki(nM) = 1360.0 EC50(nM) = 2260.0 |
2 | P42261_DB00237 | n/a | DB00237 | n/a | n/a | Butabarbital | antagonist | |
3 | P42261_DB00555 | n/a | DB00555 | n/a | n/a | Lamotrigine | inhibitor | |
4 | P42261_DB00753 | n/a | DB00753 | n/a | n/a | Isoflurane | antagonist | |
5 | P42261_EOH | EOH | DB00898 | 702 | CHEMBL545 | Ethanol | n/a | |
6 | P42261_DB01028 | n/a | DB01028 | n/a | n/a | Methoxyflurane | antagonist | |
7 | P42261_DB01189 | n/a | DB01189 | n/a | n/a | Desflurane | antagonist | |
8 | P42261_DB01236 | n/a | DB01236 | n/a | n/a | Sevoflurane | antagonist | |
9 | P42261_DB04982 | n/a | DB04982 | n/a | n/a | Talampanel | n/a | |
10 | P42261_DB05047 | n/a | DB05047 | n/a | n/a | CX-717 | n/a | |
11 | P42261_CX5 | CX5 | DB06247 | 148184 | CHEMBL136800 | CX516 | n/a | |
12 | P42261_6ZP | 6ZP | DB08883 | 9924495 | CHEMBL1214124 | Perampanel | antagonist | |
13 | P42261_DB09289 | n/a | DB09289 | n/a | n/a | Tianeptine | modulator | |
14 | P42261_DB13146 | n/a | DB13146 | n/a | n/a | Fluciclovine (18F) | inhibitor |