P46098 5HT3A_HUMAN
Gene name: HTR3A
Protein name: 5-hydroxytryptamine receptor 3A

List of molecules and drugs that interact with protein P46098

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 P46098_DB00333 n/a DB00333 n/a n/a Methadone antagonist
2 P46098_DB00334 n/a DB00334 n/a n/a Olanzapine antagonist
3 P46098_DB00363 n/a DB00363 n/a n/a Clozapine antagonist Ki(nM) = 186.0
4 P46098_O7B O7B DB00377 6337614 CHEMBL1189679 Palonosetron antagonist
5 P46098_DB00408 n/a DB00408 n/a n/a Loxapine binder
6 P46098_DB00543 n/a DB00543 n/a n/a Amoxapine antagonist
7 P46098_DB00555 n/a DB00555 n/a n/a Lamotrigine inhibitor
8 P46098_DB00604 n/a DB00604 n/a n/a Cisapride agonist
9 P46098_DB00721 n/a DB00721 n/a n/a Procaine antagonist
10 P46098_DB00726 n/a DB00726 n/a n/a Trimipramine binder
11 P46098_DB00728 n/a DB00728 n/a n/a Rocuronium antagonist
12 P46098_DB00757 n/a DB00757 n/a n/a Dolasetron antagonist
13 P46098_CWB CWB DB00889 n/a CHEMBL1290003 Granisetron antagonist Ki(nM) = 1.45
14 P46098_EOH EOH DB00898 702 CHEMBL545 Ethanol n/a
15 P46098_S87 S87 DB00904 4595 CHEMBL46 Ondansetron antagonist Ki(nM) = 2.8
IC50(nM) = 0.09
16 P46098_S7Y S7Y DB00969 2099 CHEMBL1110 Alosetron antagonist Ki(nM) = 0.5
17 P46098_LDP LDP DB00988 681 CHEMBL59 Dopamine n/a
18 P46098_DB01043 n/a DB01043 n/a n/a Memantine antagonist
19 P46098_DB01156 n/a DB01156 n/a n/a Bupropion negative modulator
20 P46098_DB01199 n/a DB01199 n/a n/a Tubocurarine antagonist
21 P46098_DB01221 n/a DB01221 n/a n/a Ketamine potentiator
22 P46098_DB01224 n/a DB01224 n/a n/a Quetiapine ligand
23 P46098_DB01233 n/a DB01233 n/a n/a Metoclopramide antagonist
24 P46098_9SC 9SC DB01238 60795 CHEMBL1112 Aripiprazole antagonist
25 P46098_DB04885 n/a DB04885 n/a n/a Cilansetron modulator
26 P46098_DB04917 n/a DB04917 n/a n/a Renzapride n/a
27 P46098_DB05642 n/a DB05642 n/a n/a DDP-225 n/a
28 P46098_DB06204 n/a DB06204 n/a n/a Tapentadol n/a
29 P46098_DB06422 n/a DB06422 n/a n/a Ticalopride n/a
30 P46098_SRO SRO DB08839 5202 CHEMBL39 Serotonin inhibitor
31 P46098_P0T P0T DB09061 644019 CHEMBL190461 Cannabidiol antagonist
32 P46098_DB09068 n/a DB09068 n/a n/a Vortioxetine antagonist
33 P46098_DB09290 n/a DB09290 n/a n/a Ramosetron antagonist
34 P46098_TKT TKT DB11699 n/a CHEMBL56564 Tropisetron antagonist
35 P46098_DB14185 n/a DB14185 n/a n/a Aripiprazole lauroxil n/a