Gene name: HTR3A
Protein name: 5-hydroxytryptamine receptor 3A
List of molecules and drugs that interact with protein P46098
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | P46098_DB00333 | n/a | DB00333 | n/a | n/a | Methadone | antagonist | |
2 | P46098_DB00334 | n/a | DB00334 | n/a | n/a | Olanzapine | antagonist | |
3 | P46098_DB00363 | n/a | DB00363 | n/a | n/a | Clozapine | antagonist | Ki(nM) = 186.0 |
4 | P46098_O7B | O7B | DB00377 | 6337614 | CHEMBL1189679 | Palonosetron | antagonist | |
5 | P46098_DB00408 | n/a | DB00408 | n/a | n/a | Loxapine | binder | |
6 | P46098_DB00543 | n/a | DB00543 | n/a | n/a | Amoxapine | antagonist | |
7 | P46098_DB00555 | n/a | DB00555 | n/a | n/a | Lamotrigine | inhibitor | |
8 | P46098_DB00604 | n/a | DB00604 | n/a | n/a | Cisapride | agonist | |
9 | P46098_DB00721 | n/a | DB00721 | n/a | n/a | Procaine | antagonist | |
10 | P46098_DB00726 | n/a | DB00726 | n/a | n/a | Trimipramine | binder | |
11 | P46098_DB00728 | n/a | DB00728 | n/a | n/a | Rocuronium | antagonist | |
12 | P46098_DB00757 | n/a | DB00757 | n/a | n/a | Dolasetron | antagonist | |
13 | P46098_CWB | CWB | DB00889 | n/a | CHEMBL1290003 | Granisetron | antagonist | Ki(nM) = 1.45 |
14 | P46098_EOH | EOH | DB00898 | 702 | CHEMBL545 | Ethanol | n/a | |
15 | P46098_S87 | S87 | DB00904 | 4595 | CHEMBL46 | Ondansetron | antagonist | Ki(nM) = 2.8 IC50(nM) = 0.09 |
16 | P46098_S7Y | S7Y | DB00969 | 2099 | CHEMBL1110 | Alosetron | antagonist | Ki(nM) = 0.5 |
17 | P46098_LDP | LDP | DB00988 | 681 | CHEMBL59 | Dopamine | n/a | |
18 | P46098_DB01043 | n/a | DB01043 | n/a | n/a | Memantine | antagonist | |
19 | P46098_DB01156 | n/a | DB01156 | n/a | n/a | Bupropion | negative modulator | |
20 | P46098_DB01199 | n/a | DB01199 | n/a | n/a | Tubocurarine | antagonist | |
21 | P46098_DB01221 | n/a | DB01221 | n/a | n/a | Ketamine | potentiator | |
22 | P46098_DB01224 | n/a | DB01224 | n/a | n/a | Quetiapine | ligand | |
23 | P46098_DB01233 | n/a | DB01233 | n/a | n/a | Metoclopramide | antagonist | |
24 | P46098_9SC | 9SC | DB01238 | 60795 | CHEMBL1112 | Aripiprazole | antagonist | |
25 | P46098_DB04885 | n/a | DB04885 | n/a | n/a | Cilansetron | modulator | |
26 | P46098_DB04917 | n/a | DB04917 | n/a | n/a | Renzapride | n/a | |
27 | P46098_DB05642 | n/a | DB05642 | n/a | n/a | DDP-225 | n/a | |
28 | P46098_DB06204 | n/a | DB06204 | n/a | n/a | Tapentadol | n/a | |
29 | P46098_DB06422 | n/a | DB06422 | n/a | n/a | Ticalopride | n/a | |
30 | P46098_SRO | SRO | DB08839 | 5202 | CHEMBL39 | Serotonin | inhibitor | |
31 | P46098_P0T | P0T | DB09061 | 644019 | CHEMBL190461 | Cannabidiol | antagonist | |
32 | P46098_DB09068 | n/a | DB09068 | n/a | n/a | Vortioxetine | antagonist | |
33 | P46098_DB09290 | n/a | DB09290 | n/a | n/a | Ramosetron | antagonist | |
34 | P46098_TKT | TKT | DB11699 | n/a | CHEMBL56564 | Tropisetron | antagonist | |
35 | P46098_DB14185 | n/a | DB14185 | n/a | n/a | Aripiprazole lauroxil | n/a |