P47869 GBRA2_HUMAN
Gene name: GABRA2
Protein name: Gamma-aminobutyric acid receptor

List of molecules and drugs that interact with protein P47869

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 P47869_DB00241 n/a DB00241 n/a n/a Butalbital positive allosteric modulator
2 P47869_DB00306 n/a DB00306 n/a n/a Talbutal potentiator
3 P47869_DB00312 n/a DB00312 n/a n/a Pentobarbital positive allosteric modulator EC50(nM) = 50000.0
4 P47869_DB00371 n/a DB00371 n/a n/a Meprobamate positive allosteric modulator
5 P47869_DB00402 n/a DB00402 n/a n/a Eszopiclone positive allosteric modulator
6 P47869_DB00418 n/a DB00418 n/a n/a Secobarbital potentiator
7 P47869_R5R R5R DB00425 5732 CHEMBL911 Zolpidem agonist Ki(nM) = 103.0
EC50(nM) = 737.0
8 P47869_VOK VOK DB00463 4099 CHEMBL450 Metharbital positive allosteric modulator
9 P47869_DB00599 n/a DB00599 n/a n/a Thiopental potentiator
10 P47869_DB00794 n/a DB00794 n/a n/a Primidone potentiator
11 P47869_DB00849 n/a DB00849 n/a n/a Methylphenobarbital potentiator
12 P47869_EOH EOH DB00898 702 CHEMBL545 Ethanol n/a
13 P47869_DB01198 n/a DB01198 n/a n/a Zopiclone potentiator
14 P47869_DB01346 n/a DB01346 n/a n/a Quinidine barbiturate potentiator
15 P47869_DB01351 n/a DB01351 n/a n/a Amobarbital potentiator
16 P47869_DB01352 n/a DB01352 n/a n/a Aprobarbital potentiator
17 P47869_DB01353 n/a DB01353 n/a n/a Butobarbital potentiator
18 P47869_DB01354 n/a DB01354 n/a n/a Heptabarbital potentiator
19 P47869_DB01355 n/a DB01355 n/a n/a Hexobarbital potentiator
20 P47869_DB01483 n/a DB01483 n/a n/a Barbital potentiator
21 P47869_DB01496 n/a DB01496 n/a n/a Dihydro-2-thioxo-5-((5-(2-(trifluoromethyl)phenyl)-2-furanyl)methyl)-4,6(1H,5H)-pyrimidinedione potentiator
22 P47869_DB01567 n/a DB01567 n/a n/a Fludiazepam potentiator
23 P47869_DB04903 n/a DB04903 n/a n/a Pagoclone n/a
24 P47869_DB13994 n/a DB13994 n/a n/a AZD-7325 positive allosteric modulator