Gene name: GABRA2
Protein name: Gamma-aminobutyric acid receptor
List of molecules and drugs that interact with protein P47869
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | P47869_DB00241 | n/a | DB00241 | n/a | n/a | Butalbital | positive allosteric modulator | |
2 | P47869_DB00306 | n/a | DB00306 | n/a | n/a | Talbutal | potentiator | |
3 | P47869_DB00312 | n/a | DB00312 | n/a | n/a | Pentobarbital | positive allosteric modulator | EC50(nM) = 50000.0 |
4 | P47869_DB00371 | n/a | DB00371 | n/a | n/a | Meprobamate | positive allosteric modulator | |
5 | P47869_DB00402 | n/a | DB00402 | n/a | n/a | Eszopiclone | positive allosteric modulator | |
6 | P47869_DB00418 | n/a | DB00418 | n/a | n/a | Secobarbital | potentiator | |
7 | P47869_R5R | R5R | DB00425 | 5732 | CHEMBL911 | Zolpidem | agonist | Ki(nM) = 103.0 EC50(nM) = 737.0 |
8 | P47869_VOK | VOK | DB00463 | 4099 | CHEMBL450 | Metharbital | positive allosteric modulator | |
9 | P47869_DB00599 | n/a | DB00599 | n/a | n/a | Thiopental | potentiator | |
10 | P47869_DB00794 | n/a | DB00794 | n/a | n/a | Primidone | potentiator | |
11 | P47869_DB00849 | n/a | DB00849 | n/a | n/a | Methylphenobarbital | potentiator | |
12 | P47869_EOH | EOH | DB00898 | 702 | CHEMBL545 | Ethanol | n/a | |
13 | P47869_DB01198 | n/a | DB01198 | n/a | n/a | Zopiclone | potentiator | |
14 | P47869_DB01346 | n/a | DB01346 | n/a | n/a | Quinidine barbiturate | potentiator | |
15 | P47869_DB01351 | n/a | DB01351 | n/a | n/a | Amobarbital | potentiator | |
16 | P47869_DB01352 | n/a | DB01352 | n/a | n/a | Aprobarbital | potentiator | |
17 | P47869_DB01353 | n/a | DB01353 | n/a | n/a | Butobarbital | potentiator | |
18 | P47869_DB01354 | n/a | DB01354 | n/a | n/a | Heptabarbital | potentiator | |
19 | P47869_DB01355 | n/a | DB01355 | n/a | n/a | Hexobarbital | potentiator | |
20 | P47869_DB01483 | n/a | DB01483 | n/a | n/a | Barbital | potentiator | |
21 | P47869_DB01496 | n/a | DB01496 | n/a | n/a | Dihydro-2-thioxo-5-((5-(2-(trifluoromethyl)phenyl)-2-furanyl)methyl)-4,6(1H,5H)-pyrimidinedione | potentiator | |
22 | P47869_DB01567 | n/a | DB01567 | n/a | n/a | Fludiazepam | potentiator | |
23 | P47869_DB04903 | n/a | DB04903 | n/a | n/a | Pagoclone | n/a | |
24 | P47869_DB13994 | n/a | DB13994 | n/a | n/a | AZD-7325 | positive allosteric modulator |