Gene name: GABRA4
Protein name: Gamma-aminobutyric acid receptor
List of molecules and drugs that interact with protein P48169
| # | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
|---|---|---|---|---|---|---|---|---|
| 1 | P48169_ABU | ABU | DB02530 | 119;6992099; | CHEMBL96 | GAMMA-AMINO-BUTANOIC ACID | n/a | EC50(nM) = 3700.0 |
| 2 | P48169_D10 | D10 | n/a | 15600 | CHEMBL134537 | DECANE | n/a | |
| 3 | P48169_EI7 | EI7 | DB06554 | 3448;28360827; | CHEMBL312443 | 4,5,6,7-tetrahydro-[1,2]oxazolo[5,4-c]pyridin-3-one | n/a | |
| 4 | P48169_HSM | HSM | DB05381 | 774 | CHEMBL90 | HISTAMINE | n/a | |
| 5 | P48169_NAG | NAG | DB00141 | 24139 | CHEMBL447878 | 2-acetamido-2-deoxy-beta-D-glucopyranose | n/a | |
| 6 | P48169_OCT | OCT | n/a | 356 | CHEMBL134886 | N-OCTANE | n/a | |
| 7 | P48169_PX6 | PX6 | n/a | 49867543 | n/a | 1,2-DIPALMITOYL-SN-GLYCERO-3-PHOSPHATE | n/a | |
| 8 | P48169_DB00241 | n/a | DB00241 | n/a | n/a | Butalbital | potentiator | |
| 9 | P48169_DB00306 | n/a | DB00306 | n/a | n/a | Talbutal | potentiator | |
| 10 | P48169_DB00312 | n/a | DB00312 | n/a | n/a | Pentobarbital | positive allosteric modulator | |
| 11 | P48169_DB00371 | n/a | DB00371 | n/a | n/a | Meprobamate | agonist | |
| 12 | P48169_DB00418 | n/a | DB00418 | n/a | n/a | Secobarbital | potentiator | |
| 13 | P48169_VOK | VOK | DB00463 | 4099 | CHEMBL450 | Metharbital | potentiator | |
| 14 | P48169_DB00599 | n/a | DB00599 | n/a | n/a | Thiopental | potentiator | |
| 15 | P48169_DB00794 | n/a | DB00794 | n/a | n/a | Primidone | potentiator | |
| 16 | P48169_DB00849 | n/a | DB00849 | n/a | n/a | Methylphenobarbital | potentiator | |
| 17 | P48169_EOH | EOH | DB00898 | 702 | CHEMBL545 | Ethanol | n/a | |
| 18 | P48169_DB01351 | n/a | DB01351 | n/a | n/a | Amobarbital | potentiator | |
| 19 | P48169_DB01352 | n/a | DB01352 | n/a | n/a | Aprobarbital | potentiator | |
| 20 | P48169_DB01353 | n/a | DB01353 | n/a | n/a | Butobarbital | potentiator | |
| 21 | P48169_DB01354 | n/a | DB01354 | n/a | n/a | Heptabarbital | potentiator | |
| 22 | P48169_DB01355 | n/a | DB01355 | n/a | n/a | Hexobarbital | potentiator | |
| 23 | P48169_DB01483 | n/a | DB01483 | n/a | n/a | Barbital | potentiator | |
| 24 | P48169_DB01496 | n/a | DB01496 | n/a | n/a | Dihydro-2-thioxo-5-((5-(2-(trifluoromethyl)phenyl)-2-furanyl)methyl)-4,6(1H,5H)-pyrimidinedione | potentiator |