Gene name: RXRG
Protein name: Retinoic acid receptor
List of molecules and drugs that interact with protein P48443
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | P48443_PLM | PLM | DB03796 | 985;135369651; | CHEMBL82293 | PALMITIC ACID | n/a | |
2 | P48443_DB00210 | n/a | DB00210 | n/a | n/a | Adapalene | agonist | |
3 | P48443_9RA | 9RA | DB00307 | 82146 | CHEMBL1023 | Bexarotene | agonist | Ki(nM) = 8.3 EC50(nM) = 20.0 |
4 | P48443_DB00412 | n/a | DB00412 | n/a | n/a | Rosiglitazone | n/a | |
5 | P48443_DB00459 | n/a | DB00459 | n/a | n/a | Acitretin | agonist | |
6 | P48443_9CR | 9CR | DB00523 | 449171 | CHEMBL705 | Alitretinoin | agonist | Ki(nM) = 11.0 IC50(nM) = 4.0 Kd(nM) = 14.0 EC50(nM) = 4.3 |
7 | P48443_REA | REA | DB00755 | 444795 | CHEMBL38 | Tretinoin | agonist | |
8 | P48443_DB00926 | n/a | DB00926 | n/a | n/a | Etretinate | agonist | |
9 | P48443_PEM | PEM | DB01393 | 39042 | CHEMBL264374 | Bezafibrate | agonist | |
10 | P48443_PHT | PHT | DB02746 | 1017;18183610; | CHEMBL1045 | Phthalic Acid | n/a | |
11 | P48443_HXA | HXA | DB03756 | 445580 | CHEMBL367149 | Doconexent | activator |