Gene name: CDK7
Protein name: Cyclin-dependent kinase 7
List of molecules and drugs that interact with protein P50613
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | P50613_1PE | 1PE | n/a | 62551 | CHEMBL1229766 | PENTAETHYLENE GLYCOL | n/a | |
2 | P50613_AGS | AGS | DB02930 | 440317;444377; | CHEMBL131890 | PHOSPHOTHIOPHOSPHORIC ACID-ADENYLATE ESTER | n/a | |
3 | P50613_ATP | ATP | DB00171 | 5957 | CHEMBL14249 | ADENOSINE-5'-TRIPHOSPHATE | n/a | |
4 | P50613_GOL | GOL | DB09462 | 753 | CHEMBL692 | GLYCEROL | n/a | |
5 | P50613_I74 | I74 | DB16061 | 91844733 | CHEMBL4297488 | (3R,4R)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | inhibitor | |
6 | P50613_MG | MG | n/a | 888 | n/a | MAGNESIUM ION | n/a | |
7 | P50613_PGE | PGE | DB02327 | 8172 | CHEMBL1235259 | TRIETHYLENE GLYCOL | n/a | |
8 | P50613_V0G | V0G | n/a | 119081415 | CHEMBL4303279 | N-(3-{[5-chloro-4-(1H-indol-3-yl)pyrimidin-2-yl]amino}phenyl)-4-{[4-(dimethylamino)butanoyl]amino}benzamide | n/a | |
9 | P50613_WZ8 | WZ8 | n/a | 71730493 | n/a | 2-[(3R)-piperidin-3-yl]oxy-8-propan-2-yl-N-[(2-pyrazol-1-ylphenyl)methyl]pyrazolo[1,5-a][1,3,5]triazin-4-amine | n/a | |
10 | P50613_D11 | D11 | DB02482 | n/a | n/a | Phosphonothreonine | inhibitor | |
11 | P50613_CPB | CPB | DB03496 | 5287969 | CHEMBL428690 | Alvocidib | n/a | IC50(nM) = 10.0 Kd(nM) = 23.0 |
12 | P50613_56H | 56H | DB05969 | 3025986 | CHEMBL296468 | SNS-032 | inhibitor | |
13 | P50613_RRC | RRC | DB06195 | 160355 | CHEMBL14762 | Seliciclib | inhibitor | |
14 | P50613_DB15442 | n/a | DB15442 | n/a | n/a | Trilaciclib | inhibitor |