Gene name: CACNA2D1
Protein name: Voltage-dependent calcium channel
List of molecules and drugs that interact with protein P54289
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | P54289_DB00230 | n/a | DB00230 | n/a | n/a | Pregabalin | modulator | Ki(nM) = 19.0 |
2 | P54289_DB00270 | n/a | DB00270 | n/a | n/a | Isradipine | inhibitor | |
3 | P54289_DB00308 | n/a | DB00308 | n/a | n/a | Ibutilide | activator | |
4 | P54289_DB00401 | n/a | DB00401 | n/a | n/a | Nisoldipine | inhibitor | |
5 | P54289_DB00622 | n/a | DB00622 | n/a | n/a | Nicardipine | inhibitor | |
6 | P54289_GBN | GBN | DB00996 | 3446;6919078; | CHEMBL940 | Gabapentin | inhibitor | IC50(nM) = 27.0 |
7 | P54289_DB01023 | n/a | DB01023 | n/a | n/a | Felodipine | inhibitor | |
8 | P54289_DB01054 | n/a | DB01054 | n/a | n/a | Nitrendipine | inhibitor | |
9 | P54289_DB04838 | n/a | DB04838 | n/a | n/a | Cyclandelate | inhibitor | |
10 | P54289_DB06712 | n/a | DB06712 | n/a | n/a | Nilvadipine | inhibitor | |
11 | P54289_DB08872 | n/a | DB08872 | n/a | n/a | Gabapentin enacarbil | n/a |