Gene name: TEK
Protein name: Angiopoietin-1 receptor (EC
List of molecules and drugs that interact with protein Q02763
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | Q02763_0CE | 0CE | n/a | 46907784 | n/a | 2-methyl-11-(1-methylethyl)-8-[(2S)-tetrahydro-2H-pyran-2-yl]-2,11,12,13-tetrahydro-4H-indazolo[5,4-a]pyrrolo[3,4-c]carbazol-4-one | n/a | |
2 | Q02763_3WR | 3WR | n/a | 11213277 | n/a | 1-[4-(4-amino-5-oxopyrido[2,3-d]pyrimidin-8(5H)-yl)phenyl]-3-[2-fluoro-5-(trifluoromethyl)phenyl]urea | n/a | |
3 | Q02763_919 | 919 | DB13005 | 25066467 | CHEMBL1738757 | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1H-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-N-methylpyridine-2-carboxamide | inhibitor | |
4 | Q02763_EDO | EDO | n/a | 174 | CHEMBL457299 | 1,2-ETHANEDIOL | n/a | |
5 | Q02763_MR9 | MR9 | n/a | 16040290 | CHEMBL219158 | 4-METHYL-3-({3-[2-(METHYLAMINO)PYRIMIDIN-4-YL]PYRIDIN-2-YL}OXY)-N-[2-MORPHOLIN-4-YL-5-(TRIFLUOROMETHYL)PHENYL]BENZAMIDE | n/a | |
6 | Q02763_MUH | MUH | DB08221 | 16040281 | CHEMBL245549 | N-{4-METHYL-3-[(3-PYRIMIDIN-4-YLPYRIDIN-2-YL)AMINO]PHENYL}-3-(TRIFLUOROMETHYL)BENZAMIDE | n/a | IC50(nM) = 17.0 |
7 | Q02763_NAG | NAG | DB00141 | 24139 | CHEMBL447878 | 2-acetamido-2-deoxy-beta-D-glucopyranose | n/a | |
8 | Q02763_QQ1 | QQ1 | n/a | 10362983 | CHEMBL1079589 | 2-[3-(CYCLOHEXYLMETHYL)-5-PHENYL-IMIDAZOL-4-YL]-[1,3]THIAZOLO[4,5-E]PYRIMIDIN-7-AMINE | n/a | |
9 | Q02763_RAJ | RAJ | n/a | 11497471 | CHEMBL221484 | N-{3-[3-(DIMETHYLAMINO)PROPYL]-5-(TRIFLUOROMETHYL)PHENYL}-4-METHYL-3-[(3-PYRIMIDIN-4-YLPYRIDIN-2-YL)AMINO]BENZAMIDE | n/a | |
10 | Q02763_SO4 | SO4 | DB14546 | 1117 | n/a | SULFATE ION | n/a | |
11 | Q02763_AIC | AIC | DB00415 | 6249;7048611; | CHEMBL174 | Ampicillin | n/a | Kd(nM) = 82000.0 |
12 | Q02763_ZD6 | ZD6 | DB05294 | 3081361 | CHEMBL24828 | Vandetanib | inhibitor | |
13 | Q02763_DB08896 | n/a | DB08896 | n/a | n/a | Regorafenib | inhibitor | IC50(nM) = 1.5 |
14 | Q02763_0LI | 0LI | DB08901 | 24826799 | CHEMBL1171837 | Ponatinib | inhibitor | |
15 | Q02763_AV9 | AV9 | DB11800 | 9911830 | CHEMBL1289494 | Tivozanib | n/a | |
16 | Q02763_2RC | 2RC | DB12010 | 11671467 | CHEMBL2103830 | Fostamatinib | inhibitor | |
17 | Q02763_DB14840 | n/a | DB14840 | n/a | n/a | Ripretinib | inhibitor |