Q02763 TIE2_HUMAN
Gene name: TEK
Protein name: Angiopoietin-1 receptor (EC

List of molecules and drugs that interact with protein Q02763

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 Q02763_0CE 0CE n/a 46907784 n/a 2-methyl-11-(1-methylethyl)-8-[(2S)-tetrahydro-2H-pyran-2-yl]-2,11,12,13-tetrahydro-4H-indazolo[5,4-a]pyrrolo[3,4-c]carbazol-4-one n/a
2 Q02763_3WR 3WR n/a 11213277 n/a 1-[4-(4-amino-5-oxopyrido[2,3-d]pyrimidin-8(5H)-yl)phenyl]-3-[2-fluoro-5-(trifluoromethyl)phenyl]urea n/a
3 Q02763_919 919 DB13005 25066467 CHEMBL1738757 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1H-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-N-methylpyridine-2-carboxamide inhibitor
4 Q02763_EDO EDO n/a 174 CHEMBL457299 1,2-ETHANEDIOL n/a
5 Q02763_MR9 MR9 n/a 16040290 CHEMBL219158 4-METHYL-3-({3-[2-(METHYLAMINO)PYRIMIDIN-4-YL]PYRIDIN-2-YL}OXY)-N-[2-MORPHOLIN-4-YL-5-(TRIFLUOROMETHYL)PHENYL]BENZAMIDE n/a
6 Q02763_MUH MUH DB08221 16040281 CHEMBL245549 N-{4-METHYL-3-[(3-PYRIMIDIN-4-YLPYRIDIN-2-YL)AMINO]PHENYL}-3-(TRIFLUOROMETHYL)BENZAMIDE n/a IC50(nM) = 17.0
7 Q02763_NAG NAG DB00141 24139 CHEMBL447878 2-acetamido-2-deoxy-beta-D-glucopyranose n/a
8 Q02763_QQ1 QQ1 n/a 10362983 CHEMBL1079589 2-[3-(CYCLOHEXYLMETHYL)-5-PHENYL-IMIDAZOL-4-YL]-[1,3]THIAZOLO[4,5-E]PYRIMIDIN-7-AMINE n/a
9 Q02763_RAJ RAJ n/a 11497471 CHEMBL221484 N-{3-[3-(DIMETHYLAMINO)PROPYL]-5-(TRIFLUOROMETHYL)PHENYL}-4-METHYL-3-[(3-PYRIMIDIN-4-YLPYRIDIN-2-YL)AMINO]BENZAMIDE n/a
10 Q02763_SO4 SO4 DB14546 1117 n/a SULFATE ION n/a
11 Q02763_AIC AIC DB00415 6249;7048611; CHEMBL174 Ampicillin n/a Kd(nM) = 82000.0
12 Q02763_ZD6 ZD6 DB05294 3081361 CHEMBL24828 Vandetanib inhibitor
13 Q02763_DB08896 n/a DB08896 n/a n/a Regorafenib inhibitor IC50(nM) = 1.5
14 Q02763_0LI 0LI DB08901 24826799 CHEMBL1171837 Ponatinib inhibitor
15 Q02763_AV9 AV9 DB11800 9911830 CHEMBL1289494 Tivozanib n/a
16 Q02763_2RC 2RC DB12010 11671467 CHEMBL2103830 Fostamatinib inhibitor
17 Q02763_DB14840 n/a DB14840 n/a n/a Ripretinib inhibitor