Q07912 ACK1_HUMAN
Gene name: TNK2
Protein name: Activated CDC42 kinase

List of molecules and drugs that interact with protein Q07912

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 Q07912_1G0 1G0 n/a n/a CHEMBL3651314 cis-3-[8-amino-1-(4-phenoxyphenyl)imidazo[1,5-a]pyrazin-3-yl]cyclobutanol n/a
2 Q07912_9KO 9KO n/a 137348835 CHEMBL4214342 N-{3-[7-{[6-(4-acetylpiperazin-1-yl)pyridin-3-yl]amino}-1-methyl-2-oxo-1,4-dihydropyrimido[4,5-d]pyrimidin-3(2H)-yl]-4-methylphenyl}-3-(trifluoromethyl)benzamide n/a
3 Q07912_ACP ACP DB03909 91532 CHEMBL133463 PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTER n/a
4 Q07912_CL CL n/a 312 n/a CHLORIDE ION n/a
5 Q07912_DBQ DBQ DB04367 5288032;135451156; CHEMBL255465 DEBROMOHYMENIALDISINE n/a
6 Q07912_EDO EDO n/a 174 CHEMBL457299 1,2-ETHANEDIOL n/a
7 Q07912_MG MG n/a 888 n/a MAGNESIUM ION n/a
8 Q07912_R7P R7P n/a 155804523 CHEMBL4792672 2-({4-[(3R,5S)-3,5-dimethylpiperazin-1-yl]-2-methoxyphenyl}amino)-9-methyl-5,7-dihydro-6H-pyrimido[5,4-d][1,3]benzodiazepin-6-one n/a
9 Q07912_SO4 SO4 DB14546 1117 n/a SULFATE ION n/a
10 Q07912_WTP WTP n/a 90479825 CHEMBL3426891 5-chloro-N~2~-[4-(4-methylpiperazin-1-yl)phenyl]-N~4~-{[(2R)-oxolan-2-yl]methyl}pyrimidine-2,4-diamine n/a
11 Q07912_T74 T74 n/a 15965424 CHEMBL472392 N~3~-(2,6-dimethylphenyl)-1-(3-methoxy-3-methylbutyl)-N~6~-(4-piperazin-1-ylphenyl)-1H-pyrazolo[3,4-d]pyrimidine-3,6-diamine n/a
12 Q07912_T77 T77 n/a 11576813 CHEMBL2087873 6-{4-[2-(dimethylamino)ethoxy]phenyl}-N-(1,3-dithiolan-2-ylmethyl)-5-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine n/a
13 Q07912_T95 T95 n/a 25113175 n/a N-(2,6-dimethylphenyl)-4-(2-ethoxyphenoxy)-2-({4-[4-(2-hydroxyethyl)piperazin-1-yl]phenyl}amino)pyrimidine-5-carboxamide n/a
14 Q07912_ATP ATP DB00171 5957 CHEMBL14249 ATP n/a
15 Q07912_YMX YMX DB11986 25141092 CHEMBL1983268 Entrectinib n/a
16 Q07912_2RC 2RC DB12010 11671467 CHEMBL2103830 Fostamatinib inhibitor