Gene name: TNK2
Protein name: Activated CDC42 kinase
List of molecules and drugs that interact with protein Q07912
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | Q07912_1G0 | 1G0 | n/a | n/a | CHEMBL3651314 | cis-3-[8-amino-1-(4-phenoxyphenyl)imidazo[1,5-a]pyrazin-3-yl]cyclobutanol | n/a | |
2 | Q07912_9KO | 9KO | n/a | 137348835 | CHEMBL4214342 | N-{3-[7-{[6-(4-acetylpiperazin-1-yl)pyridin-3-yl]amino}-1-methyl-2-oxo-1,4-dihydropyrimido[4,5-d]pyrimidin-3(2H)-yl]-4-methylphenyl}-3-(trifluoromethyl)benzamide | n/a | |
3 | Q07912_ACP | ACP | DB03909 | 91532 | CHEMBL133463 | PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTER | n/a | |
4 | Q07912_CL | CL | n/a | 312 | n/a | CHLORIDE ION | n/a | |
5 | Q07912_DBQ | DBQ | DB04367 | 5288032;135451156; | CHEMBL255465 | DEBROMOHYMENIALDISINE | n/a | |
6 | Q07912_EDO | EDO | n/a | 174 | CHEMBL457299 | 1,2-ETHANEDIOL | n/a | |
7 | Q07912_MG | MG | n/a | 888 | n/a | MAGNESIUM ION | n/a | |
8 | Q07912_R7P | R7P | n/a | 155804523 | CHEMBL4792672 | 2-({4-[(3R,5S)-3,5-dimethylpiperazin-1-yl]-2-methoxyphenyl}amino)-9-methyl-5,7-dihydro-6H-pyrimido[5,4-d][1,3]benzodiazepin-6-one | n/a | |
9 | Q07912_SO4 | SO4 | DB14546 | 1117 | n/a | SULFATE ION | n/a | |
10 | Q07912_WTP | WTP | n/a | 90479825 | CHEMBL3426891 | 5-chloro-N~2~-[4-(4-methylpiperazin-1-yl)phenyl]-N~4~-{[(2R)-oxolan-2-yl]methyl}pyrimidine-2,4-diamine | n/a | |
11 | Q07912_T74 | T74 | n/a | 15965424 | CHEMBL472392 | N~3~-(2,6-dimethylphenyl)-1-(3-methoxy-3-methylbutyl)-N~6~-(4-piperazin-1-ylphenyl)-1H-pyrazolo[3,4-d]pyrimidine-3,6-diamine | n/a | |
12 | Q07912_T77 | T77 | n/a | 11576813 | CHEMBL2087873 | 6-{4-[2-(dimethylamino)ethoxy]phenyl}-N-(1,3-dithiolan-2-ylmethyl)-5-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine | n/a | |
13 | Q07912_T95 | T95 | n/a | 25113175 | n/a | N-(2,6-dimethylphenyl)-4-(2-ethoxyphenoxy)-2-({4-[4-(2-hydroxyethyl)piperazin-1-yl]phenyl}amino)pyrimidine-5-carboxamide | n/a | |
14 | Q07912_ATP | ATP | DB00171 | 5957 | CHEMBL14249 | ATP | n/a | |
15 | Q07912_YMX | YMX | DB11986 | 25141092 | CHEMBL1983268 | Entrectinib | n/a | |
16 | Q07912_2RC | 2RC | DB12010 | 11671467 | CHEMBL2103830 | Fostamatinib | inhibitor |