Gene name: EP300
Protein name: Histone acetyltransferase p300
List of molecules and drugs that interact with protein Q09472
| # | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
|---|---|---|---|---|---|---|---|---|
| 1 | Q09472_01K | 01K | n/a | 23727984 | n/a | [(2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-4-hydroxy-3-(phosphonooxy)tetrahydrofuran-2-yl]methyl (3R,20R)-20-carbamoyl-3-hydroxy-2,2-dimethyl-4,8,14,22-tetraoxo-12-thia-5,9,15,21-tetraazatricos-1-yl dihydrogen diphosphate | n/a | |
| 2 | Q09472_1VU | 1VU | DB02912 | 92753 | n/a | propionyl Coenzyme A | n/a | |
| 3 | Q09472_2LO | 2LO | n/a | 72201027 | CHEMBL3622373 | 2-[2-(3-chloro-4-methoxyphenyl)ethyl]-5-(3,5-dimethyl-1,2-oxazol-4-yl)-1-[(2S)-2-(morpholin-4-yl)propyl]-1H-benzimidazole | n/a | |
| 4 | Q09472_6QI | 6QI | n/a | 163196907 | n/a | [(6R)-6-(1H-indazol-4-ylmethyl)-1,4-oxazepan-4-yl]-[1-(4-methoxyphenyl)cyclopentyl]methanone | n/a | |
| 5 | Q09472_6TF | 6TF | n/a | 118958122 | CHEMBL4282264 | N-[(4-fluorophenyl)methyl]-2-{(1R)-5-[(methylcarbamoyl)amino]-2',4'-dioxo-2,3-dihydro-3'H-spiro[indene-1,5'-[1,3]oxazolidin]-3'-yl}-N-[(2S)-1,1,1-trifluoropropan-2-yl]acetamide | n/a | |
| 6 | Q09472_6TI | 6TI | n/a | 142504112 | CHEMBL5178312 | (2R)-N-(2H-indazol-4-yl)-1-[1-(4-methoxyphenyl)cyclopentyl]carbonyl-pyrrolidine-2-carboxamide | n/a | |
| 7 | Q09472_6YI | 6YI | n/a | 163196908 | CHEMBL5193672 | (4S)-N-(3H-indazol-4-yl)-3-[1-(4-methoxyphenyl)cyclopentyl]carbonyl-1,1-bis(oxidanylidene)-1,3-thiazolidine-4-carboxamide | n/a | |
| 8 | Q09472_71Y | 71Y | n/a | 129318943 | n/a | ~{N}-[(1~{S},2~{S})-7-chloranyl-2-oxidanyl-1,2,3,4-tetrahydronaphthalen-1-yl]-4-ethanoyl-3-ethyl-5-methyl-1~{H}-pyrrole -2-carboxamide | n/a | |
| 9 | Q09472_99E | 99E | n/a | 129318956 | CHEMBL4741587 | ~{N}-[[2,8-bis(oxidanyl)naphthalen-1-yl]methyl]-4-ethanoyl-3-ethyl-5-methyl-1~{H}-pyrrole-2-carboxamide | n/a | |
| 10 | Q09472_ACN | ACN | n/a | 180 | CHEMBL14253 | ACETONE | n/a | |
| 11 | Q09472_ACO | ACO | n/a | 444493 | CHEMBL1230809 | ACETYL COENZYME *A | n/a | |
| 12 | Q09472_ACT | ACT | DB14511 | 175 | n/a | ACETATE ION | n/a | |
| 13 | Q09472_BCO | BCO | n/a | 122283 | n/a | Butyryl Coenzyme A | n/a | |
| 14 | Q09472_BR | BR | n/a | 259 | n/a | BROMIDE ION | n/a | |
| 15 | Q09472_C0C | C0C | n/a | 165416302 | CHEMBL5219712 | 1-[1-(4-chlorophenyl)cyclopentane-1-carbonyl]-N-{[3-(methylcarbamoyl)phenyl]methyl}-D-prolinamide | n/a | |
| 16 | Q09472_C3I | C3I | n/a | 4880035 | CHEMBL1700017 | N-[2-(4-methoxyanilino)-2-oxoethyl]-N-methyl-1-phenylcyclopentane-1-carboxamide | n/a | |
| 17 | Q09472_CL | CL | n/a | 312 | n/a | CHLORIDE ION | n/a | |
| 18 | Q09472_COA | COA | DB01992 | 87642 | CHEMBL1213327 | COENZYME A | n/a | |
| 19 | Q09472_COO | COO | n/a | 92856 | n/a | CROTONYL COENZYME A | n/a | |
| 20 | Q09472_DMS | DMS | DB01093 | 679 | CHEMBL504 | DIMETHYL SULFOXIDE | n/a | |
| 21 | Q09472_EDO | EDO | n/a | 174 | CHEMBL457299 | 1,2-ETHANEDIOL | n/a | |
| 22 | Q09472_ETL | ETL | n/a | 165416315 | n/a | 1-[1-(4-chlorophenyl)cyclopentane-1-carbonyl]-N-1H-pyrazolo[4,3-b]pyridin-5-yl-D-prolinamide | n/a | |
| 23 | Q09472_GOL | GOL | DB09462 | 753 | CHEMBL692 | GLYCEROL | n/a | |
| 24 | Q09472_IPA | IPA | DB02325 | 3776 | CHEMBL582 | ISOPROPYL ALCOHOL | n/a | |
| 25 | Q09472_KQO | KQO | n/a | 142504056 | CHEMBL5401710 | (2~{R},4~{R})-4-fluoranyl-1-[1-(4-methoxyphenyl)cyclohexyl]carbonyl-~{N}-(1~{H}-pyrazolo[4,3-b]pyridin-5-yl)pyrrolidine-2-carboxamide | n/a | |
| 26 | Q09472_N6I | N6I | n/a | 135440466 | CHEMBL401930 | (3M)-4-{[(2S)-2-(3-chlorophenyl)-2-hydroxyethyl]amino}-3-[4-methyl-6-(morpholin-4-yl)-1H-benzimidazol-2-yl]pyridin-2(1H)-one | n/a | |
| 27 | Q09472_NA | NA | n/a | 923 | n/a | SODIUM ION | n/a | |
| 28 | Q09472_OJ7 | OJ7 | n/a | 1483806 | n/a | 3-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-2-methyl-1H-indole | n/a | |
| 29 | Q09472_OK7 | OK7 | n/a | 83087 | n/a | N-(thiophen-2-yl)acetamide | n/a | |
| 30 | Q09472_PE5 | PE5 | DB03556 | 657096 | n/a | 3,6,9,12,15,18,21,24-OCTAOXAHEXACOSAN-1-OL | n/a | |
| 31 | Q09472_PEG | PEG | n/a | 8117 | CHEMBL1235226 | DI(HYDROXYETHYL)ETHER | n/a | |
| 32 | Q09472_PG4 | PG4 | n/a | 8200 | CHEMBL1235254 | TETRAETHYLENE GLYCOL | n/a | |
| 33 | Q09472_QRY | QRY | n/a | 30008286 | n/a | 4-(2-{[(1R)-2-(1H-indol-3-yl)-2-oxo-1-phenylethyl]amino}ethyl)benzene-1-sulfonamide | n/a | |
| 34 | Q09472_QS1 | QS1 | n/a | 146014965 | CHEMBL4641354 | (2R)-2-{[(2S)-2-(4-cyanophenyl)propyl]amino}-N-[5-(1-methyl-1H-pyrazol-4-yl)pyridin-2-yl]-2-phenylacetamide | n/a | |
| 35 | Q09472_QS4 | QS4 | n/a | 920121 | n/a | 1-(2-methyl-1H-indol-3-yl)-2-[(2R)-2-methylpiperidin-1-yl]ethan-1-one | n/a | |
| 36 | Q09472_QSD | QSD | n/a | 146014966 | CHEMBL4636118 | (2R)-2-{[2-(4-cyanophenyl)ethyl]amino}-N-[5-(1-methyl-1H-pyrazol-4-yl)pyridin-2-yl]-2-phenylacetamide | n/a | |
| 37 | Q09472_SO4 | SO4 | DB14546 | 1117 | n/a | SULFATE ION | n/a | |
| 38 | Q09472_TCE | TCE | n/a | 119411 | CHEMBL171512 | 3,3',3''-phosphanetriyltripropanoic acid | n/a | |
| 39 | Q09472_XDM | XDM | n/a | 75415563 | n/a | ~{N}-[(3-chlorophenyl)methyl]-4-ethanoyl-3-ethyl-5-methyl-1~{H}-pyrrole-2-carboxamide | n/a | |
| 40 | Q09472_Y2P | Y2P | n/a | 118956836 | CHEMBL4787599 | 2-[4-[(3'R,4S)-3'-fluoro-1-[2-[(4-fluorophenyl)methyl-[(1S)-2,2,2-trifluoro-1-methyl-ethyl]amino]-2-oxo-ethyl]-2,5-dioxo-spiro[imidazolidine-4,1'-indane]-5'-yl]pyrazol-1-yl]-N-methyl-acetamide | n/a | |
| 41 | Q09472_ZN | ZN | n/a | 32051 | CHEMBL1236970 | ZINC ION | n/a | |
| 42 | Q09472_SOP | SOP | n/a | 194658 | n/a | [(2R,3S,4R,5R)-5-(6-AMINO-9H-PURIN-9-YL)-4-HYDROXY-3-(PHOSPHONOOXY)TETRAHYDROFURAN-2-YL]METHYL (3R)-3-HYDROXY-2,2-DIMETHYL-4-OXO-4-{[3-OXO-3-({2-[(2-OXOPROPYL)THIO]ETHYL}AMINO)PROPYL]AMINO}BUTYL DIHYDROGEN DIPHOSPHATE | n/a | |
| 43 | Q09472_TAM | TAM | DB04237 | 448009 | n/a | TRIS(HYDROXYETHYL)AMINOMETHANE | n/a |