Q12852 M3K12_HUMAN
Gene name: MAP3K12
Protein name: Mitogen-activated protein kinase

List of molecules and drugs that interact with protein Q12852

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 Q12852_50D 50D n/a 72547959 CHEMBL3393333 2-[[6-[3,3-bis(fluoranyl)pyrrolidin-1-yl]-4-[1-(oxetan-3-yl)piperidin-4-yl]pyridin-2-yl]amino]pyridine-4-carbonitrile n/a
2 Q12852_50E 50E n/a 91936969 CHEMBL3629009 N-(5-piperidin-4-yl-1-propan-2-yl-pyrazol-3-yl)-4-(trifluoromethyl)pyridin-2-amine n/a
3 Q12852_50F 50F n/a 91936970 CHEMBL3629013 2-[[1-cyclopentyl-5-[1-(oxetan-3-yl)piperidin-4-yl]pyrazol-3-yl]amino]pyridine-4-carbonitrile n/a
4 Q12852_9FS 9FS n/a n/a CHEMBL3717481 5-{5-[(1R,5S,6r)-3-(oxetan-3-yl)-3-azabicyclo[3.1.0]hexan-6-yl]-1-(propan-2-yl)-1H-pyrazol-3-yl}-3-(trifluoromethyl)pyridin-2-amine n/a
5 Q12852_SIQ SIQ n/a n/a n/a methyl (1S,4S)-5-{(4P)-4-[5-amino-6-(difluoromethoxy)pyrazin-2-yl]-6-[(1R,4R)-2-azabicyclo[2.1.1]hexan-2-yl]pyridin-2-yl}-2,5-diazabicyclo[2.2.1]heptane-2-carboxylate n/a
6 Q12852_W38 W38 n/a n/a n/a 5-[1-(3-morpholin-4-yl-1-bicyclo[1.1.1]pentanyl)-2-propan-2-yl-imidazol-4-yl]-3-(trifluoromethyloxy)pyridin-2-amine n/a
7 Q12852_W3C W3C n/a n/a n/a (1R)-1-[4-[6-azanyl-5-(trifluoromethyloxy)pyridin-3-yl]-1-(3-fluoranyl-1-bicyclo[1.1.1]pentanyl)imidazol-2-yl]-2,2,2-tris(fluoranyl)ethanol n/a
8 Q12852_2RC 2RC DB12010 11671467 CHEMBL2103830 Fostamatinib inhibitor