Gene name: HTR4
Protein name: 5-hydroxytryptamine receptor 4
List of molecules and drugs that interact with protein Q13639
| # | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
|---|---|---|---|---|---|---|---|---|
| 1 | Q13639_2GM | 2GM | DB00320 | 10531 | CHEMBL1732 | Dihydroergotamine | agonist | |
| 2 | Q13639_DB00604 | n/a | DB00604 | n/a | n/a | Cisapride | agonist | |
| 3 | Q13639_S87 | S87 | DB00904 | 4595 | CHEMBL46 | Ondansetron | agonist | |
| 4 | Q13639_DB01079 | n/a | DB01079 | n/a | n/a | Tegaserod | antagonist | |
| 5 | Q13639_DB01233 | n/a | DB01233 | n/a | n/a | Metoclopramide | agonist | EC50(nM) = 794.0 |
| 6 | Q13639_DB04873 | n/a | DB04873 | n/a | n/a | Piboserod | antagonist | Ki(nM) = 0.01 IC50(nM) = 0.63 |
| 7 | Q13639_DB04917 | n/a | DB04917 | n/a | n/a | Renzapride | modulator | |
| 8 | Q13639_DB05542 | n/a | DB05542 | n/a | n/a | Naronapride | agonist | |
| 9 | Q13639_DB05905 | n/a | DB05905 | n/a | n/a | TD-2749 | agonist | |
| 10 | Q13639_DB06422 | n/a | DB06422 | n/a | n/a | Ticalopride | n/a | |
| 11 | Q13639_DB06480 | n/a | DB06480 | n/a | n/a | Prucalopride | agonist | Ki(nM) = 2.5 Kd(nM) = 2.0 EC50(nM) = 5.2 |
| 12 | Q13639_DB08810 | n/a | DB08810 | n/a | n/a | Cinitapride | agonist | |
| 13 | Q13639_DB12702 | n/a | DB12702 | n/a | n/a | Velusetrag | agonist |