Gene name: SCN5A
Protein name: Sodium channel protein
List of molecules and drugs that interact with protein Q14524
| # | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
|---|---|---|---|---|---|---|---|---|
| 1 | Q14524_NAG | NAG | DB00141 | 24139 | CHEMBL447878 | 2-acetamido-2-deoxy-beta-D-glucopyranose | n/a | |
| 2 | Q14524_QDN | QDN | DB00908 | 441074 | CHEMBL1294 | Quinidine | inhibitor | |
| 3 | Q14524_SO4 | SO4 | DB14546 | 1117 | n/a | SULFATE ION | n/a | |
| 4 | Q14524_DB00192 | n/a | DB00192 | n/a | n/a | Indecainide | inhibitor | |
| 5 | Q14524_DB00252 | n/a | DB00252 | n/a | n/a | Phenytoin | inhibitor | IC50(nM) = 49000.0 |
| 6 | Q14524_DB00280 | n/a | DB00280 | n/a | n/a | Disopyramide | inhibitor | |
| 7 | Q14524_LQZ | LQZ | DB00281 | 3676 | CHEMBL79 | Lidocaine | inhibitor | IC50(nM) = 50000.0 |
| 8 | Q14524_DB00379 | n/a | DB00379 | n/a | n/a | Mexiletine | inhibitor | IC50(nM) = 3000.0 |
| 9 | Q14524_DB00473 | n/a | DB00473 | n/a | n/a | Hexylcaine | inhibitor | |
| 10 | Q14524_DB00527 | n/a | DB00527 | n/a | n/a | Cinchocaine | inhibitor | |
| 11 | Q14524_DB00532 | n/a | DB00532 | n/a | n/a | Mephenytoin | inhibitor | |
| 12 | Q14524_DB00680 | n/a | DB00680 | n/a | n/a | Moricizine | inhibitor | |
| 13 | Q14524_657 | 657 | DB00740 | 5070 | CHEMBL744 | Riluzole | inhibitor | |
| 14 | Q14524_DB00750 | n/a | DB00750 | n/a | n/a | Prilocaine | inhibitor | |
| 15 | Q14524_DB00754 | n/a | DB00754 | n/a | n/a | Ethotoin | inhibitor | |
| 16 | Q14524_DB00868 | n/a | DB00868 | n/a | n/a | Benzonatate | antagonist | |
| 17 | Q14524_ZON | ZON | DB00909 | 5734;11967800; | CHEMBL750 | Zonisamide | inhibitor | |
| 18 | Q14524_DB01035 | n/a | DB01035 | n/a | n/a | Procainamide | inhibitor | |
| 19 | Q14524_DB01056 | n/a | DB01056 | n/a | n/a | Tocainide | inhibitor | |
| 20 | Q14524_DB01182 | n/a | DB01182 | n/a | n/a | Propafenone | inhibitor | IC50(nM) = 1190.0 |
| 21 | Q14524_DB01195 | n/a | DB01195 | n/a | n/a | Flecainide | inhibitor | IC50(nM) = 6500.0 |
| 22 | Q14524_DB01228 | n/a | DB01228 | n/a | n/a | Encainide | inhibitor | |
| 23 | Q14524_DB01320 | n/a | DB01320 | n/a | n/a | Fosphenytoin | inhibitor | |
| 24 | Q14524_DB01346 | n/a | DB01346 | n/a | n/a | Quinidine barbiturate | inhibitor | |
| 25 | Q14524_DB01426 | n/a | DB01426 | n/a | n/a | Ajmaline | inhibitor | |
| 26 | Q14524_DB01429 | n/a | DB01429 | n/a | n/a | Aprindine | inhibitor | |
| 27 | Q14524_DB04855 | n/a | DB04855 | n/a | n/a | Dronedarone | inhibitor | |
| 28 | Q14524_DB06217 | n/a | DB06217 | n/a | n/a | Vernakalant | blocker | |
| 29 | Q14524_QKM | QKM | DB11633 | 6918485 | CHEMBL409153 | Isavuconazole | inhibitor |