Gene name: SCN5A
Protein name: Sodium channel protein
List of molecules and drugs that interact with protein Q14524
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | Q14524_NAG | NAG | DB00141 | 24139 | CHEMBL447878 | 2-acetamido-2-deoxy-beta-D-glucopyranose | n/a | |
2 | Q14524_QDN | QDN | DB00908 | 441074 | CHEMBL1294 | Quinidine | inhibitor | |
3 | Q14524_SO4 | SO4 | DB14546 | 1117 | n/a | SULFATE ION | n/a | |
4 | Q14524_DB00192 | n/a | DB00192 | n/a | n/a | Indecainide | inhibitor | |
5 | Q14524_DB00252 | n/a | DB00252 | n/a | n/a | Phenytoin | inhibitor | IC50(nM) = 49000.0 |
6 | Q14524_DB00280 | n/a | DB00280 | n/a | n/a | Disopyramide | inhibitor | |
7 | Q14524_LQZ | LQZ | DB00281 | 3676 | CHEMBL79 | Lidocaine | inhibitor | IC50(nM) = 50000.0 |
8 | Q14524_DB00379 | n/a | DB00379 | n/a | n/a | Mexiletine | inhibitor | IC50(nM) = 3000.0 |
9 | Q14524_DB00473 | n/a | DB00473 | n/a | n/a | Hexylcaine | inhibitor | |
10 | Q14524_DB00527 | n/a | DB00527 | n/a | n/a | Cinchocaine | inhibitor | |
11 | Q14524_DB00532 | n/a | DB00532 | n/a | n/a | Mephenytoin | inhibitor | |
12 | Q14524_DB00680 | n/a | DB00680 | n/a | n/a | Moricizine | inhibitor | |
13 | Q14524_657 | 657 | DB00740 | 5070 | CHEMBL744 | Riluzole | inhibitor | |
14 | Q14524_DB00750 | n/a | DB00750 | n/a | n/a | Prilocaine | inhibitor | |
15 | Q14524_DB00754 | n/a | DB00754 | n/a | n/a | Ethotoin | inhibitor | |
16 | Q14524_DB00868 | n/a | DB00868 | n/a | n/a | Benzonatate | antagonist | |
17 | Q14524_ZON | ZON | DB00909 | 5734;11967800; | CHEMBL750 | Zonisamide | inhibitor | |
18 | Q14524_DB01035 | n/a | DB01035 | n/a | n/a | Procainamide | inhibitor | |
19 | Q14524_DB01056 | n/a | DB01056 | n/a | n/a | Tocainide | inhibitor | |
20 | Q14524_DB01182 | n/a | DB01182 | n/a | n/a | Propafenone | inhibitor | IC50(nM) = 1190.0 |
21 | Q14524_DB01195 | n/a | DB01195 | n/a | n/a | Flecainide | inhibitor | IC50(nM) = 6500.0 |
22 | Q14524_DB01228 | n/a | DB01228 | n/a | n/a | Encainide | inhibitor | |
23 | Q14524_DB01320 | n/a | DB01320 | n/a | n/a | Fosphenytoin | inhibitor | |
24 | Q14524_DB01346 | n/a | DB01346 | n/a | n/a | Quinidine barbiturate | inhibitor | |
25 | Q14524_DB01426 | n/a | DB01426 | n/a | n/a | Ajmaline | inhibitor | |
26 | Q14524_DB01429 | n/a | DB01429 | n/a | n/a | Aprindine | inhibitor | |
27 | Q14524_DB04855 | n/a | DB04855 | n/a | n/a | Dronedarone | inhibitor | |
28 | Q14524_DB06217 | n/a | DB06217 | n/a | n/a | Vernakalant | blocker | |
29 | Q14524_QKM | QKM | DB11633 | 6918485 | CHEMBL409153 | Isavuconazole | inhibitor |