Q15118 PDK1_HUMAN
Gene name: PDK1
Protein name: [Pyruvate dehydrogenase (acetyl-transferring)]

List of molecules and drugs that interact with protein Q15118

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 Q15118_AZX AZX DB07403 16741245 CHEMBL1231132 4-[(3-CHLORO-4-{[(2R)-3,3,3-TRIFLUORO-2-HYDROXY-2-METHYLPROPANOYL]AMINO}PHENYL)SULFONYL]-N,N-DIMETHYLBENZAMIDE n/a
2 Q15118_K K n/a 813 CHEMBL1233793 POTASSIUM ION n/a
3 Q15118_TF4 TF4 DB08809 6597 CHEMBL13960 DICHLORO-ACETIC ACID inhibitor IC50(nM) = 100000.0
EC50(nM) = 50000.0