Gene name: SCN9A
Protein name: Sodium channel protein
List of molecules and drugs that interact with protein Q15858
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | Q15858_9SL | 9SL | n/a | 37165;56947150; | CHEMBL501134 | [(3aS,4R,10aS)-2,6-diamino-10,10-dihydroxy-3a,4,9,10-tetrahydro-3H,8H-pyrrolo[1,2-c]purin-4-yl]methyl carbamate | n/a | |
2 | Q15858_9SR | 9SR | n/a | 11174599 | CHEMBL507974 | (1R,5R,6R,7R,9S,11S,12S,13S,14S)-3-amino-14-(hydroxymethyl)-8,10-dioxa-2,4-diazatetracyclo[7.3.1.1~7,11~.0~1,6~]tetradec-3-ene-5,9,12,13,14-pentol (non-preferred name) | n/a | |
3 | Q15858_G2W | G2W | n/a | 53348208 | CHEMBL3944666 | 3-[[4-[3-(4-fluoranyl-2-methyl-phenoxy)azetidin-1-yl]pyrimidin-2-yl]amino]-~{N}-methyl-benzamide | n/a | |
4 | Q15858_G4I | G4I | n/a | 53361524 | CHEMBL1813048 | (1~{Z})-~{N}-[2-methyl-3-[(~{E})-[6-[4-[[4-(trifluoromethyloxy)phenyl]methoxy]piperidin-1-yl]-1~{H}-1,3,5-triazin-2-ylidene]amino]phenyl]ethanimidic acid | n/a | |
5 | Q15858_NAG | NAG | DB00141 | 24139 | CHEMBL447878 | 2-acetamido-2-deoxy-beta-D-glucopyranose | n/a | |
6 | Q15858_LQZ | LQZ | DB00281 | 3676 | CHEMBL79 | Lidocaine | inhibitor | IC50(nM) = 16000.0 |
7 | Q15858_ZON | ZON | DB00909 | 5734;11967800; | CHEMBL750 | Zonisamide | inhibitor | |
8 | Q15858_DB06201 | n/a | DB06201 | n/a | n/a | Rufinamide | modulator | |
9 | Q15858_DB06218 | n/a | DB06218 | n/a | n/a | Lacosamide | blocker | IC50(nM) = 182.0 |