Q15858 SCN9A_HUMAN
Gene name: SCN9A
Protein name: Sodium channel protein

List of molecules and drugs that interact with protein Q15858

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 Q15858_9SL 9SL n/a 37165;56947150; CHEMBL501134 [(3aS,4R,10aS)-2,6-diamino-10,10-dihydroxy-3a,4,9,10-tetrahydro-3H,8H-pyrrolo[1,2-c]purin-4-yl]methyl carbamate n/a
2 Q15858_9SR 9SR n/a 11174599 CHEMBL507974 (1R,5R,6R,7R,9S,11S,12S,13S,14S)-3-amino-14-(hydroxymethyl)-8,10-dioxa-2,4-diazatetracyclo[7.3.1.1~7,11~.0~1,6~]tetradec-3-ene-5,9,12,13,14-pentol (non-preferred name) n/a
3 Q15858_G2W G2W n/a 53348208 CHEMBL3944666 3-[[4-[3-(4-fluoranyl-2-methyl-phenoxy)azetidin-1-yl]pyrimidin-2-yl]amino]-~{N}-methyl-benzamide n/a
4 Q15858_G4I G4I n/a 53361524 CHEMBL1813048 (1~{Z})-~{N}-[2-methyl-3-[(~{E})-[6-[4-[[4-(trifluoromethyloxy)phenyl]methoxy]piperidin-1-yl]-1~{H}-1,3,5-triazin-2-ylidene]amino]phenyl]ethanimidic acid n/a
5 Q15858_NAG NAG DB00141 24139 CHEMBL447878 2-acetamido-2-deoxy-beta-D-glucopyranose n/a
6 Q15858_LQZ LQZ DB00281 3676 CHEMBL79 Lidocaine inhibitor IC50(nM) = 16000.0
7 Q15858_ZON ZON DB00909 5734;11967800; CHEMBL750 Zonisamide inhibitor
8 Q15858_DB06201 n/a DB06201 n/a n/a Rufinamide modulator
9 Q15858_DB06218 n/a DB06218 n/a n/a Lacosamide blocker IC50(nM) = 182.0