Q460N3 PAR15_HUMAN
Gene name: PARP15
Protein name: Protein mono-ADP-ribosyltransferase PARP15

List of molecules and drugs that interact with protein Q460N3

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 Q460N3_0Q6 0Q6 n/a 26051380 CHEMBL4293771 4-[(3-bromophenyl)methoxy]benzamide n/a
2 Q460N3_0RU 0RU n/a 9202458;135566723; CHEMBL5187963 8-methyl-2-[(pyrimidin-2-ylsulfanyl)methyl]quinazolin-4(1H)-one n/a
3 Q460N3_0SI 0SI n/a 162368286 CHEMBL5076823 8-phenylmethoxy-4~{H}-thieno[2,3-c]isoquinolin-5-one n/a
4 Q460N3_0UI 0UI n/a 161231673 CHEMBL5077731 8-oxidanyl-4~{H}-thieno[2,3-c]isoquinolin-5-one n/a
5 Q460N3_1H9 1H9 n/a 162368287 CHEMBL5078132 8-[(3-bromophenyl)methoxy]-4~{H}-thieno[2,3-c]isoquinolin-5-one n/a
6 Q460N3_1O7 1O7 n/a 162368296 CHEMBL5091585 8-ethoxy-4~{H}-thieno[2,3-c]isoquinolin-5-one n/a
7 Q460N3_1OI 1OI n/a 58024740 CHEMBL5084343 8-methoxy-4~{H}-thieno[2,3-c]isoquinolin-5-one n/a
8 Q460N3_33E 33E DB13877 9796068 CHEMBL1170047 4-iodo-3-nitrobenzamide n/a
9 Q460N3_3AB 3AB n/a 1645 CHEMBL81977 3-aminobenzamide n/a
10 Q460N3_3JD 3JD DB11793 24958200 CHEMBL1094636 2-{4-[(3S)-piperidin-3-yl]phenyl}-2H-indazole-7-carboxamide n/a
11 Q460N3_89H 89H n/a 163203938 n/a 6-(cyclopropylmethoxy)phthalazine-1,4-dione n/a
12 Q460N3_89Q 89Q n/a 69813446 CHEMBL5198692 4-(cyclopropylmethoxy)benzamide n/a
13 Q460N3_89Z 89Z n/a 163203936 n/a 6-(cyclopentylmethoxy)phthalazine-1,4-dione n/a
14 Q460N3_8A8 8A8 n/a 163203935 n/a 6-(cyclohexylmethoxy)phthalazine-1,4-dione n/a
15 Q460N3_8AE 8AE n/a 67115989 CHEMBL5186967 4-(cyclobutylmethoxy)benzamide n/a
16 Q460N3_8AQ 8AQ n/a 163203933 CHEMBL5185276 4-(cyclohexylmethoxy)-2-methoxy-benzamide n/a
17 Q460N3_8B5 8B5 n/a n/a n/a 6-[(3-bromophenyl)methoxy]phthalazine-1,4-dione n/a
18 Q460N3_8BE 8BE n/a 163203934 CHEMBL5198615 4-[(3-bromophenyl)methoxy]-2-methoxy-benzamide n/a
19 Q460N3_8BK 8BK n/a 142600514 CHEMBL5185078 4-(1,3-thiazol-5-ylmethoxy)benzamide n/a
20 Q460N3_8BW 8BW n/a 163203937 n/a 6-(cyclobutylmethoxy)phthalazine-1,4-dione n/a
21 Q460N3_8C7 8C7 n/a 8608139 CHEMBL5178227 4-(cyclohexylmethoxy)benzamide n/a
22 Q460N3_8CI 8CI n/a 163203931 CHEMBL5206305 4-(cyclopentylmethoxy)benzamide n/a
23 Q460N3_8D2 8D2 n/a 163203940 n/a 6-[(2-fluorophenyl)methoxy]phthalazine-1,4-dione n/a
24 Q460N3_8DB 8DB n/a 163203941 n/a 6-(thiophen-2-ylmethoxy)phthalazine-1,4-dione n/a
25 Q460N3_AR6 AR6 DB02059 447048 n/a [(2R,3S,4R,5R)-5-(6-AMINOPURIN-9-YL)-3,4-DIHYDROXY-OXOLAN-2-YL]METHYL[HYDROXY-[[(2R,3S,4R,5S)-3,4,5-TRIHYDROXYOXOLAN-2-YL]METHOXY]PHOSPHORYL] HYDROGEN PHOSPHATE n/a
26 Q460N3_CL CL n/a 312 n/a CHLORIDE ION n/a
27 Q460N3_DMS DMS DB01093 679 CHEMBL504 DIMETHYL SULFOXIDE n/a
28 Q460N3_G18 G18 n/a 9899130 CHEMBL3108871 4H-thieno[2,3-c]isoquinolin-5-one n/a
29 Q460N3_GOL GOL DB09462 753 CHEMBL692 GLYCEROL n/a
30 Q460N3_I1B I1B n/a 326031 CHEMBL5402584 6,8-dimethyl-[1,2,4]triazolo[3,4-b][1,3]benzothiazole n/a
31 Q460N3_I1Q I1Q n/a 326023 CHEMBL4296925 6-methyl-[1,2,4]triazolo[3,4-b][1,3]benzothiazole n/a
32 Q460N3_I4X I4X n/a 145705616 CHEMBL5439304 6-propan-2-yl-[1,2,4]triazolo[3,4-b][1,3]benzothiazole n/a
33 Q460N3_I5F I5F n/a 33702003 CHEMBL5406267 [1,2,4]triazolo[3,4-b][1,3]benzothiazol-6-ol n/a
34 Q460N3_I9L I9L n/a 86240079 CHEMBL5395721 6-chloranyl-[1,2,4]triazolo[3,4-b][1,3]benzothiazole n/a
35 Q460N3_I9R I9R n/a 129897812 CHEMBL5416085 5,8-dimethoxy-[1,2,4]triazolo[3,4-b][1,3]benzothiazole n/a
36 Q460N3_IAJ IAJ n/a 13473717 CHEMBL5433172 8-methoxy-[1,2,4]triazolo[3,4-b][1,3]benzothiazole n/a
37 Q460N3_IAO IAO n/a 2771058 CHEMBL5404785 5,8-dimethoxy-[1,2,4]triazolo[3,4-b][1,3]benzothiazol-1-amine n/a
38 Q460N3_IAW IAW n/a 13473720 CHEMBL5398837 6-methoxy-[1,2,4]triazolo[3,4-b][1,3]benzothiazole n/a
39 Q460N3_KMW KMW n/a 69845715 CHEMBL4126054 3-(4-aminocarbonylphenoxy)benzamide n/a
40 Q460N3_MPD MPD DB03564 5288834 n/a (4S)-2-METHYL-2,4-PENTANEDIOL n/a
41 Q460N3_NA NA n/a 923 n/a SODIUM ION n/a
42 Q460N3_OUL OUL n/a 236501 CHEMBL1438938 4-(4-aminocarbonylphenoxy)benzamide n/a
43 Q460N3_P34 P34 DB08348 4858;5289097; CHEMBL372303 N~2~,N~2~-DIMETHYL-N~1~-(6-OXO-5,6-DIHYDROPHENANTHRIDIN-2-YL)GLYCINAMIDE n/a IC50(nM) = 8913.0
44 Q460N3_VJN VJN n/a 162368334 CHEMBL5083566 8-propan-2-yloxy-4~{H}-thieno[2,3-c]isoquinolin-5-one n/a