Gene name: HCAR2
Protein name: Hydroxycarboxylic acid receptor
List of molecules and drugs that interact with protein Q8TDS4
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | Q8TDS4_AW9 | AW9 | n/a | 61799 | CHEMBL4577612 | (2Z)-4-methoxy-4-oxobut-2-enoic acid | n/a | |
2 | Q8TDS4_CLR | CLR | DB04540 | 5997 | CHEMBL112570 | CHOLESTEROL | n/a | |
3 | Q8TDS4_FI7 | FI7 | n/a | 135416394 | CHEMBL1086657 | 2-[[2,2-dimethyl-3-[3-(5-oxidanylpyridin-2-yl)-1,2,4-oxadiazol-5-yl]propanoyl]amino]cyclohexene-1-carboxylic acid | n/a | |
4 | Q8TDS4_IX8 | IX8 | n/a | 25101223 | CHEMBL490599 | 7-methyl-N-[(2R)-1-phenoxypropan-2-yl]-3-(4-propan-2-ylphenyl)pyrazolo[1,5-a]pyrimidine-6-carboxamide | n/a | |
5 | Q8TDS4_NIO | NIO | DB00627 | 938;117629482; | CHEMBL573 | NICOTINIC ACID | agonist | Ki(nM) = 50.0 IC50(nM) = 130.0 EC50(nM) = 8.7 |
6 | Q8TDS4_OJX | OJX | n/a | 59806020 | n/a | 5-methyl-4-oxidanyl-pyrazin-4-ium-2-carboxylic acid | n/a | |
7 | Q8TDS4_OKL | OKL | n/a | 46215799 | CHEMBL3730241 | 8-chloranyl-3-pentyl-7H-purine-2,6-dione | n/a | |
8 | Q8TDS4_OLA | OLA | n/a | 445639 | CHEMBL8659 | OLEIC ACID | n/a | |
9 | Q8TDS4_OLC | OLC | n/a | 11451146 | n/a | (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate | n/a | |
10 | Q8TDS4_CL6 | CL6 | DB00257 | 2812 | CHEMBL104 | Clotrimazole | partial agonist | |
11 | Q8TDS4_DB08949 | n/a | DB08949 | n/a | n/a | Inositol nicotinate | agonist |