Q8WTS6 SETD7_HUMAN
Gene name: SETD7
Protein name: Histone-lysine N-methyltransferase SETD7

List of molecules and drugs that interact with protein Q8WTS6

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 Q8WTS6_0N6 0N6 n/a 56851708 n/a (R)-(3-(3-cyanophenyl)-1-oxo-1-(pyrrolidin-1-yl)propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide n/a
2 Q8WTS6_1L4 1L4 n/a 71296073 n/a N-[(2R)-3-(3-cyanophenyl)-1-oxo-1-(pyrrolidin-1-yl)propan-2-yl]-8-fluoro-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide n/a
3 Q8WTS6_1L8 1L8 n/a 71300326 CHEMBL3414622 8-fluoro-N-{(2R)-1-oxo-1-(pyrrolidin-1-yl)-3-[3-(trifluoromethyl)phenyl]propan-2-yl}-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide n/a
4 Q8WTS6_BME BME DB03345 1567 CHEMBL254951 BETA-MERCAPTOETHANOL n/a
5 Q8WTS6_C7H C7H DB00434 2913 CHEMBL516 4-(dibenzo[1,2-a:2',1'-d][7]annulen-11-ylidene)-1-methyl-piperidine n/a Ki(nM) = 15000.0
IC50(nM) = 1000.0
6 Q8WTS6_C7N C7N n/a 85727193 n/a 2-(1-methylpiperidin-4-ylidene)tricyclo[9.4.0.0^{3,8}]pentadeca-1(11),3(8),4,6,9,12,14-heptaen-6-ol n/a
7 Q8WTS6_CO CO n/a 104729 n/a COBALT (II) ION n/a
8 Q8WTS6_EDO EDO n/a 174 CHEMBL457299 1,2-ETHANEDIOL n/a
9 Q8WTS6_GOL GOL DB09462 753 CHEMBL692 GLYCEROL n/a
10 Q8WTS6_K15 K15 n/a 52944960 CHEMBL1290526 5'-{[(3S)-3-amino-3-carboxypropyl](hexyl)amino}-5'-deoxyadenosine n/a
11 Q8WTS6_KH3 KH3 n/a 50915251 CHEMBL1290525 5'-{[(3S)-3-amino-3-carboxypropyl][2-(hexylamino)ethyl]amino}-5'-deoxyadenosine n/a
12 Q8WTS6_MG MG n/a 888 n/a MAGNESIUM ION n/a
13 Q8WTS6_NA NA n/a 923 n/a SODIUM ION n/a
14 Q8WTS6_SAH SAH DB01752 439155;25246222; CHEMBL418052 S-ADENOSYL-L-HOMOCYSTEINE n/a
15 Q8WTS6_SAM SAM DB00118 n/a CHEMBL1235831 S-ADENOSYLMETHIONINE n/a
16 Q8WTS6_SFG SFG DB01910 65482 CHEMBL1214186 SINEFUNGIN n/a
17 Q8WTS6_SO4 SO4 DB14546 1117 n/a SULFATE ION n/a
18 Q8WTS6_TRS TRS DB03754 3777159;88088752;152743085; n/a 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL n/a
19 Q8WTS6_UNL UNL n/a
20 Q8WTS6_UNX UNX n/a