Gene name: GPER1
Protein name: G-protein coupled estrogen
List of molecules and drugs that interact with protein Q99527
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | Q99527_EST | EST | DB00783 | 5757 | CHEMBL135 | Estradiol | binder | Ki(nM) = 5.7 EC50(nM) = 0.3 |
2 | Q99527_GEN | GEN | DB01645 | 5280961 | CHEMBL44 | Genistein | n/a | |
3 | Q99527_DB05939 | n/a | DB05939 | n/a | n/a | MK-0354 | n/a | |
4 | Q99527_DB13952 | n/a | DB13952 | n/a | n/a | Estradiol acetate | n/a | |
5 | Q99527_DB13953 | n/a | DB13953 | n/a | n/a | Estradiol benzoate | n/a | |
6 | Q99527_DB13954 | n/a | DB13954 | n/a | n/a | Estradiol cypionate | n/a | |
7 | Q99527_DB13955 | n/a | DB13955 | n/a | n/a | Estradiol dienanthate | n/a | |
8 | Q99527_DB13956 | n/a | DB13956 | n/a | n/a | Estradiol valerate | n/a |