Gene name: EIF2AK4
Protein name: eIF-2-alpha kinase GCN2
List of molecules and drugs that interact with protein Q9P2K8
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | Q9P2K8_38O | 38O | DB05928 | 135398510 | CHEMBL522892 | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1H-benzimidazol-2-yl]quinolin-2(1H)-one | n/a | |
2 | Q9P2K8_DMS | DMS | DB01093 | 679 | CHEMBL504 | DIMETHYL SULFOXIDE | n/a | |
3 | Q9P2K8_G41 | G41 | n/a | 163201229 | n/a | (2~{S})-~{N}-[(1~{S})-1-[4-[(6-pyridin-4-ylquinazolin-2-yl)amino]phenyl]ethyl]piperidine-2-carboxamide | n/a | |
4 | Q9P2K8_KA4 | KA4 | n/a | 137347437 | n/a | N-{3-[(2-aminopyrimidin-5-yl)ethynyl]-2,4-difluorophenyl}-2,5-dichloro-3-(hydroxymethyl)benzene-1-sulfonamide | n/a | |
5 | Q9P2K8_KA7 | KA7 | n/a | 134814489 | n/a | N-{3-[(2-aminopyrimidin-5-yl)ethynyl]-2,4-difluorophenyl}-5-chloro-2-methoxypyridine-3-sulfonamide | n/a | |
6 | Q9P2K8_KAV | KAV | n/a | 139208930 | n/a | N-{6-[(1-methyl-2-{[4-(trifluoromethyl)phenyl]amino}-1H-benzimidazol-5-yl)oxy]pyrimidin-4-yl}cyclopropanecarboxamide | n/a | |
7 | Q9P2K8_2RC | 2RC | DB12010 | 11671467 | CHEMBL2103830 | Fostamatinib | inhibitor |