Q9UBS5 GABR1_HUMAN
Gene name: GABBR1
Protein name: Gamma-aminobutyric acid type

List of molecules and drugs that interact with protein Q9UBS5

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 Q9UBS5_2BQ 2BQ n/a 6603711;7005136; CHEMBL1556176 2-hydroxysaclofen n/a
2 Q9UBS5_2BV 2BV n/a 197584 CHEMBL1213187 (R)-(cyclohexylmethyl)[(2S)-3-{[(1S)-1-(3,4-dichlorophenyl)ethyl]amino}-2-hydroxypropyl]phosphinic acid n/a
3 Q9UBS5_2BW 2BW n/a 107699 CHEMBL40157 (S)-(3-aminopropyl)(diethoxymethyl)phosphinic acid n/a
4 Q9UBS5_2BX 2BX n/a 5311429;86294992; CHEMBL1895916 [(2S)-5,5-dimethylmorpholin-2-yl]acetic acid n/a
5 Q9UBS5_2BY 2BY n/a 6603957 CHEMBL1435984 phaclofen n/a
6 Q9UBS5_2C0 2C0 DB08891 44602;6918881; CHEMBL301742 baclofen agonist
7 Q9UBS5_381 381 n/a 130022 CHEMBL112362 (S)-(3-aminopropyl)(cyclohexylmethyl)phosphinic acid n/a
8 Q9UBS5_ABU ABU DB02530 119;6992099; CHEMBL96 GAMMA-AMINO-BUTANOIC ACID inhibitor IC50(nM) = 25.0
EC50(nM) = 530.0
9 Q9UBS5_CA CA n/a 271 n/a CALCIUM ION n/a
10 Q9UBS5_CLR CLR DB04540 5997 CHEMBL112570 CHOLESTEROL n/a
11 Q9UBS5_FN0 FN0 n/a 7023848 CHEMBL3600959 (3S)-5,7-ditert-butyl-3-oxidanyl-3-(trifluoromethyl)-1-benzofuran-2-one n/a
12 Q9UBS5_L9Q L9Q n/a 23727970 n/a (1S)-2-{[(S)-(2-aminoethoxy)(hydroxy)phosphoryl]oxy}-1-[(octadecanoyloxy)methyl]ethyl (9Z)-octadec-9-enoate n/a
13 Q9UBS5_MG MG n/a 888 n/a MAGNESIUM ION n/a
14 Q9UBS5_NAG NAG DB00141 24139 CHEMBL447878 2-acetamido-2-deoxy-beta-D-glucopyranose n/a
15 Q9UBS5_QD7 QD7 n/a 5230;28559746; CHEMBL112710 (R)-(3-aminopropyl)methylphosphinic acid n/a
16 Q9UBS5_QDA QDA n/a 6604928 CHEMBL392394 N~4~,N~6~-dicyclopentyl-2-(methylsulfanyl)-5-nitropyrimidine-4,6-diamine n/a
17 Q9UBS5_SGG SGG n/a 5311042 CHEMBL455185 [(2~{S})-3-[[(1~{S})-1-(3,4-dichlorophenyl)ethyl]amino]-2-oxidanyl-propyl]-(phenylmethyl)phosphinic acid n/a
18 Q9UBS5_U3G U3G n/a 52924645 n/a (2R)-3-{[(S)-(2-aminoethoxy)(hydroxy)phosphoryl]oxy}-2-{[(9Z)-octadec-9-enoyl]oxy}propyl (5Z,8Z,11Z,14Z)-icosa-5,8,11,14-tetraenoate n/a
19 Q9UBS5_UNL UNL n/a
20 Q9UBS5_DB00181 n/a DB00181 n/a n/a Baclofen agonist Ki(nM) = 6000.0
IC50(nM) = 35.0
EC50(nM) = 1700.0
21 Q9UBS5_DB00659 n/a DB00659 n/a n/a Acamprosate inhibitor
22 Q9UBS5_DB00837 n/a DB00837 n/a n/a Progabide agonist
23 Q9UBS5_TAU TAU DB01956 1123;4068592; CHEMBL239243 Taurine agonist
24 Q9UBS5_DB05010 n/a DB05010 n/a n/a SGS-742 modulator
25 Q9UBS5_DB06354 n/a DB06354 n/a n/a Tezampanel n/a
26 Q9UBS5_DB08892 n/a DB08892 n/a n/a Arbaclofen Placarbil agonist
27 Q9UBS5_DB12098 n/a DB12098 n/a n/a L-Baclofen agonist