Gene name: GABBR1
Protein name: Gamma-aminobutyric acid type
List of molecules and drugs that interact with protein Q9UBS5
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | Q9UBS5_2BQ | 2BQ | n/a | 6603711;7005136; | CHEMBL1556176 | 2-hydroxysaclofen | n/a | |
2 | Q9UBS5_2BV | 2BV | n/a | 197584 | CHEMBL1213187 | (R)-(cyclohexylmethyl)[(2S)-3-{[(1S)-1-(3,4-dichlorophenyl)ethyl]amino}-2-hydroxypropyl]phosphinic acid | n/a | |
3 | Q9UBS5_2BW | 2BW | n/a | 107699 | CHEMBL40157 | (S)-(3-aminopropyl)(diethoxymethyl)phosphinic acid | n/a | |
4 | Q9UBS5_2BX | 2BX | n/a | 5311429;86294992; | CHEMBL1895916 | [(2S)-5,5-dimethylmorpholin-2-yl]acetic acid | n/a | |
5 | Q9UBS5_2BY | 2BY | n/a | 6603957 | CHEMBL1435984 | phaclofen | n/a | |
6 | Q9UBS5_2C0 | 2C0 | DB08891 | 44602;6918881; | CHEMBL301742 | baclofen | agonist | |
7 | Q9UBS5_381 | 381 | n/a | 130022 | CHEMBL112362 | (S)-(3-aminopropyl)(cyclohexylmethyl)phosphinic acid | n/a | |
8 | Q9UBS5_ABU | ABU | DB02530 | 119;6992099; | CHEMBL96 | GAMMA-AMINO-BUTANOIC ACID | inhibitor | IC50(nM) = 25.0 EC50(nM) = 530.0 |
9 | Q9UBS5_CA | CA | n/a | 271 | n/a | CALCIUM ION | n/a | |
10 | Q9UBS5_CLR | CLR | DB04540 | 5997 | CHEMBL112570 | CHOLESTEROL | n/a | |
11 | Q9UBS5_FN0 | FN0 | n/a | 7023848 | CHEMBL3600959 | (3S)-5,7-ditert-butyl-3-oxidanyl-3-(trifluoromethyl)-1-benzofuran-2-one | n/a | |
12 | Q9UBS5_L9Q | L9Q | n/a | 23727970 | n/a | (1S)-2-{[(S)-(2-aminoethoxy)(hydroxy)phosphoryl]oxy}-1-[(octadecanoyloxy)methyl]ethyl (9Z)-octadec-9-enoate | n/a | |
13 | Q9UBS5_MG | MG | n/a | 888 | n/a | MAGNESIUM ION | n/a | |
14 | Q9UBS5_NAG | NAG | DB00141 | 24139 | CHEMBL447878 | 2-acetamido-2-deoxy-beta-D-glucopyranose | n/a | |
15 | Q9UBS5_QD7 | QD7 | n/a | 5230;28559746; | CHEMBL112710 | (R)-(3-aminopropyl)methylphosphinic acid | n/a | |
16 | Q9UBS5_QDA | QDA | n/a | 6604928 | CHEMBL392394 | N~4~,N~6~-dicyclopentyl-2-(methylsulfanyl)-5-nitropyrimidine-4,6-diamine | n/a | |
17 | Q9UBS5_SGG | SGG | n/a | 5311042 | CHEMBL455185 | [(2~{S})-3-[[(1~{S})-1-(3,4-dichlorophenyl)ethyl]amino]-2-oxidanyl-propyl]-(phenylmethyl)phosphinic acid | n/a | |
18 | Q9UBS5_U3G | U3G | n/a | 52924645 | n/a | (2R)-3-{[(S)-(2-aminoethoxy)(hydroxy)phosphoryl]oxy}-2-{[(9Z)-octadec-9-enoyl]oxy}propyl (5Z,8Z,11Z,14Z)-icosa-5,8,11,14-tetraenoate | n/a | |
19 | Q9UBS5_UNL | UNL | n/a | |||||
20 | Q9UBS5_DB00181 | n/a | DB00181 | n/a | n/a | Baclofen | agonist | Ki(nM) = 6000.0 IC50(nM) = 35.0 EC50(nM) = 1700.0 |
21 | Q9UBS5_DB00659 | n/a | DB00659 | n/a | n/a | Acamprosate | inhibitor | |
22 | Q9UBS5_DB00837 | n/a | DB00837 | n/a | n/a | Progabide | agonist | |
23 | Q9UBS5_TAU | TAU | DB01956 | 1123;4068592; | CHEMBL239243 | Taurine | agonist | |
24 | Q9UBS5_DB05010 | n/a | DB05010 | n/a | n/a | SGS-742 | modulator | |
25 | Q9UBS5_DB06354 | n/a | DB06354 | n/a | n/a | Tezampanel | n/a | |
26 | Q9UBS5_DB08892 | n/a | DB08892 | n/a | n/a | Arbaclofen Placarbil | agonist | |
27 | Q9UBS5_DB12098 | n/a | DB12098 | n/a | n/a | L-Baclofen | agonist |