Gene name: PDE10A
Protein name: cAMP and cAMP-inhibited
List of molecules and drugs that interact with protein Q9Y233
| # | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
|---|---|---|---|---|---|---|---|---|
| 1 | Q9Y233_0CV | 0CV | n/a | 46239840 | CHEMBL1939782 | 6-methoxy-3,8-dimethyl-4-(piperazin-1-yl)-1H-pyrazolo[3,4-b]quinoline | n/a | |
| 2 | Q9Y233_0JP | 0JP | n/a | 50903255 | CHEMBL2017087 | 8,9-dimethoxy-1-(1,3-thiazol-5-yl)-5,6-dihydroimidazo[5,1-a]isoquinoline | n/a | |
| 3 | Q9Y233_0JQ | 0JQ | n/a | 25196602 | CHEMBL1956250 | 2-{1-[5-(6,7-dimethoxycinnolin-4-yl)-3-methylpyridin-2-yl]piperidin-4-yl}propan-2-ol | n/a | |
| 4 | Q9Y233_0T6 | 0T6 | n/a | 60150358 | CHEMBL2069321 | 1-(2-chlorophenyl)-6,8-dimethoxy-3-methylimidazo[5,1-c][1,2,4]benzotriazine | n/a | |
| 5 | Q9Y233_0T7 | 0T7 | n/a | 57732460 | n/a | 3,4-dimethyl-1-propyl-7-(quinolin-2-ylmethoxy)imidazo[1,5-a]quinoxaline | n/a | |
| 6 | Q9Y233_15H | 15H | n/a | 70679303 | n/a | (1S)-1-(1-{3-[4-(1,3-benzothiazol-2-ylamino)phenoxy]pyrazin-2-yl}piperidin-4-yl)ethanol | n/a | |
| 7 | Q9Y233_15J | 15J | n/a | 70679302 | CHEMBL2206214 | (1-{3-[4-(1H-benzimidazol-2-ylamino)phenoxy]pyridin-2-yl}piperidin-4-yl)methanol | n/a | |
| 8 | Q9Y233_1IR | 1IR | n/a | n/a | CHEMBL3287906 | N-[cis-3-(2-methoxy-3H-imidazo[4,5-b]pyridin-3-yl)cyclobutyl]-1,3-benzothiazol-2-amine | n/a | |
| 9 | Q9Y233_1IS | 1IS | n/a | n/a | CHEMBL3287907 | N-[trans-3-(2-methoxy-3H-imidazo[4,5-b]pyridin-3-yl)cyclobutyl]-1,3-benzothiazol-2-amine | n/a | |
| 10 | Q9Y233_1XM | 1XM | n/a | 90253;1268262;135408756; | CHEMBL4436742 | 4-amino-1,7-dihydro-6H-pyrazolo[3,4-d]pyrimidine-6-thione | n/a | |
| 11 | Q9Y233_1XN | 1XN | n/a | 19935268 | CHEMBL4466464 | 2H-isoindole-1,3-diamine | n/a | |
| 12 | Q9Y233_2D0 | 2D0 | n/a | 29872 | CHEMBL1413383 | 4-chloro-1,3-benzothiazol-2-amine | n/a | |
| 13 | Q9Y233_2F4 | 2F4 | n/a | 24983496 | CHEMBL3086086 | 2-{4-[(6,7-difluoro-1H-benzimidazol-2-yl)amino]phenoxy}-N-methyl-3,4'-bipyridin-2'-amine | n/a | |
| 14 | Q9Y233_2F5 | 2F5 | n/a | 46207938 | CHEMBL3086091 | 1H-benzimidazol-2-yl(4-{[3-(morpholin-4-yl)pyrazin-2-yl]oxy}phenyl)methanone | n/a | |
| 15 | Q9Y233_2KR | 2KR | n/a | 76210621 | CHEMBL3287662 | N-[4-(2-methoxy-3H-imidazo[4,5-b]pyridin-3-yl)phenyl]-5-methylpyridin-2-amine | n/a | |
| 16 | Q9Y233_2W1 | 2W1 | n/a | 59326858 | CHEMBL3319208 | 1H-benzimidazol-2-yl(4-{[3-(tetrahydro-2H-pyran-4-yl)pyridin-2-yl]oxy}phenyl)methanone | n/a | |
| 17 | Q9Y233_2ZM | 2ZM | n/a | 7195;86262143; | CHEMBL164921 | 5-nitro-1H-benzimidazole | n/a | |
| 18 | Q9Y233_2ZQ | 2ZQ | n/a | 11830 | CHEMBL167727 | 8-nitroquinoline | n/a | |
| 19 | Q9Y233_2ZT | 2ZT | n/a | 73659152 | CHEMBL4583461 | 2-[(quinolin-7-yloxy)methyl]quinoline | n/a | |
| 20 | Q9Y233_2ZU | 2ZU | n/a | 73659153 | CHEMBL4453729 | 2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}quinoline | n/a | |
| 21 | Q9Y233_2ZV | 2ZV | n/a | 243166 | CHEMBL3981727 | 4-methyl-3-nitropyridin-2-amine | n/a | |
| 22 | Q9Y233_2ZX | 2ZX | n/a | 67432 | CHEMBL4517551 | 6-chloropyrimidine-2,4-diamine | n/a | |
| 23 | Q9Y233_35D | 35D | n/a | 58547814 | CHEMBL3356684 | 1-[4-(3-{[1-(quinolin-2-yl)azetidin-3-yl]oxy}quinoxalin-2-yl)piperidin-1-yl]ethanone | n/a | |
| 24 | Q9Y233_35E | 35E | n/a | 58547833 | CHEMBL2180767 | [1-(3-{[1-(quinolin-2-yl)azetidin-3-yl]oxy}pyrazin-2-yl)piperidin-4-yl]methanol | n/a | |
| 25 | Q9Y233_35G | 35G | DB02315 | 24316;5280386;135398570; | CHEMBL395336 | GUANOSINE-3',5'-MONOPHOSPHATE | n/a | |
| 26 | Q9Y233_3A6 | 3A6 | n/a | 70789261 | n/a | 3-AMINO-6-FLUORO-2-[4-(2-METHYLPYRIDIN-4-YL)PHENYL]-N-(METHYLSULFONYL)QUINOLINE-4-CARBOXAMIDE | n/a | |
| 27 | Q9Y233_3K9 | 3K9 | DB14774 | 46848915 | CHEMBL3989972 | 1-[2-fluoro-4-(1H-pyrazol-1-yl)phenyl]-5-methoxy-3-(1-phenyl-1H-pyrazol-5-yl)pyridazin-4(1H)-one | inhibitor | |
| 28 | Q9Y233_3KB | 3KB | n/a | 59436195 | n/a | 5-methoxy-3-(1-phenyl-1H-pyrazol-5-yl)-1-[3-(trifluoromethyl)phenyl]pyridazin-4(1H)-one | n/a | |
| 29 | Q9Y233_3KG | 3KG | n/a | 46219819 | n/a | 3-(1-phenyl-1H-pyrazol-5-yl)-1-[3-(trifluoromethyl)phenyl]pyridazin-4(1H)-one | n/a | |
| 30 | Q9Y233_3SJ | 3SJ | n/a | 66555959 | n/a | 1-methyl-5-(1-methyl-3-{[4-(quinolin-2-yl)phenoxy]methyl}-1H-pyrazol-4-yl)pyridin-2(1H)-one | n/a | |
| 31 | Q9Y233_490 | 490 | n/a | 66555104 | n/a | 1-methyl-5-(1-methyl-3-{[4-(1-methyl-1H-benzimidazol-4-yl)phenoxy]methyl}-1H-pyrazol-4-yl)pyridin-2(1H)-one | n/a | |
| 32 | Q9Y233_4F7 | 4F7 | n/a | 54755130 | CHEMBL2180006 | 2-[2-(4-phenyl-1H-imidazol-2-yl)ethyl]quinoxaline | n/a | |
| 33 | Q9Y233_4GK | 4GK | n/a | 57412063 | n/a | 2-[2-(5,8-dimethyl[1,2,4]triazolo[1,5-a]pyrazin-2-yl)ethyl]-3-methyl-3H-imidazo[4,5-f]quinoline | n/a | |
| 34 | Q9Y233_4HN | 4HN | n/a | 56587975 | CHEMBL1957361 | 2-(2'-ETHOXYBIPHENYL-4-YL)-4-HYDROXY-1,6-NAPHTHYRIDINE-3-CARBONITRILE | n/a | |
| 35 | Q9Y233_4LK | 4LK | n/a | 46848917 | CHEMBL3629540 | 3-[3-fluoranyl-4-[5-methoxy-4-oxidanylidene-3-(2-phenylpyrazol-3-yl)pyridazin-1-yl]phenyl]-1,3-oxazolidin-2-one | n/a | |
| 36 | Q9Y233_4LP | 4LP | n/a | 56651641 | CHEMBL3629735 | 1-(cyclopropylmethyl)-4-fluoranyl-5-[5-methoxy-4-oxidanylidene-3-(2-phenylpyrazol-3-yl)pyridazin-1-yl]-3,3-dimethyl-indol-2-one | n/a | |
| 37 | Q9Y233_4PX | 4PX | n/a | 91826676 | n/a | 3-(1-hydroxy-2-methylpropan-2-yl)-5-phenyl-3,5-dihydro-1H-imidazo[4,5-c][1,8]naphthyridine-2,4-dione | n/a | |
| 38 | Q9Y233_4Q0 | 4Q0 | n/a | 49821931 | CHEMBL3627841 | 2-{2-[3-(4-methoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl]ethyl}-4-(propan-2-yloxy)-1H-isoindole-1,3(2H)-dione | n/a | |
| 39 | Q9Y233_4XS | 4XS | n/a | 54595731 | CHEMBL3622905 | 4,6-dichloro-2-cyclopropyl-5-methylpyrimidine | n/a | |
| 40 | Q9Y233_4XU | 4XU | n/a | 56949451 | CHEMBL3622898 | 6-chloro-N-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]-5-methyl-2-[3-(quinolin-2-yl)propoxy]pyrimidin-4-amine | n/a | |
| 41 | Q9Y233_4XV | 4XV | n/a | 77230235 | CHEMBL3622906 | 6-chloro-2-cyclopropyl-5-methylpyrimidin-4-amine | n/a | |
| 42 | Q9Y233_4XY | 4XY | n/a | 80970780 | CHEMBL3621548 | 6-chloro-2-cyclopropyl-5-methyl-N-propylpyrimidin-4-amine | n/a | |
| 43 | Q9Y233_4Y1 | 4Y1 | n/a | 56949475 | CHEMBL3622894 | 6-chloro-N-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]-5-methyl-2-[2-(pyridin-2-yl)ethoxy]pyrimidin-4-amine | n/a | |
| 44 | Q9Y233_4Y2 | 4Y2 | n/a | 91885643 | CHEMBL3622879 | 6-chloro-2-cyclopropyl-N-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]-5-methylpyrimidin-4-amine | n/a | |
| 45 | Q9Y233_4ZE | 4ZE | n/a | 76081 | CHEMBL3092391 | 4-amino-2-methylphenol | n/a | |
| 46 | Q9Y233_540 | 540 | n/a | 42630191 | CHEMBL1916113 | 8-fluoro-6-methoxy-3,4-dimethyl-1-(3-methylpyridin-4-yl)imidazo[1,5-a]quinoxaline | n/a | |
| 47 | Q9Y233_546 | 546 | n/a | 42629702 | CHEMBL1916091 | 2-methoxy-6,7-dimethyl-9-(4-methylpyridin-3-yl)imidazo[1,5-a]pyrido[3,2-e]pyrazine | n/a | |
| 48 | Q9Y233_548 | 548 | n/a | 49821469 | CHEMBL1916132 | 6-chloro-3,4-dimethyl-1-(3-methylpyridin-4-yl)-8-(trifluoromethyl)imidazo[1,5-a]quinoxaline | n/a | |
| 49 | Q9Y233_5AV | 5AV | n/a | 127042560 | CHEMBL3747347 | 5-chloro-N-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine | n/a | |
| 50 | Q9Y233_5AY | 5AY | n/a | 76903477 | CHEMBL3695713 | N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-{[(1S,2S)-2-(pyridin-2-yl)cyclopropyl]methoxy}pyrazolo[1,5-a]pyrimidin-7-amine | n/a | |
| 51 | Q9Y233_5GP | 5GP | DB01972 | 6804;5280325;135398631; | CHEMBL283807 | GUANOSINE-5'-MONOPHOSPHATE | n/a | |
| 52 | Q9Y233_5M6 | 5M6 | n/a | 2393958 | n/a | 1-(4-chlorophenyl)-3-methyl-~{N}-[[(2~{R})-oxolan-2-yl]methyl]thieno[2,3-c]pyrazole-5-carboxamide | n/a | |
| 53 | Q9Y233_5M9 | 5M9 | n/a | 90033975 | CHEMBL3964469 | 6-chloranyl-5,8-dimethyl-2-[2-(2-methyl-5-pyrrolidin-1-yl-1,2,4-triazol-3-yl)ethyl]-[1,2,4]triazolo[1,5-a]pyridine | n/a | |
| 54 | Q9Y233_5MF | 5MF | n/a | 72705844 | CHEMBL3934495 | 8-ethyl-5-methyl-2-[2-(2-methyl-5-pyrrolidin-1-yl-1,2,4-triazol-3-yl)ethyl]-[1,2,4]triazolo[1,5-c]pyrimidine | n/a | |
| 55 | Q9Y233_5MG | 5MG | n/a | 135567090 | n/a | 3-(2-chloranyl-5-phenyl-1~{H}-imidazol-4-yl)-1-[3-(trifluoromethyloxy)phenyl]pyridazin-4-one | n/a | |
| 56 | Q9Y233_5NI | 5NI | DB04534 | 21501 | CHEMBL165372 | 5-NITROINDAZOLE | n/a | |
| 57 | Q9Y233_5ZE | 5ZE | n/a | 13021 | CHEMBL4546836 | 4,6-dimethylpyrimidin-2-amine | n/a | |
| 58 | Q9Y233_67A | 67A | n/a | 46219578 | CHEMBL2180789 | 3-(1-phenyl-1H-pyrazol-5-yl)-1-[3-(trifluoromethoxy)phenyl]pyridazin-4(1H)-one | n/a | |
| 59 | Q9Y233_6DT | 6DT | n/a | 52946084 | CHEMBL1253915 | N-(4-((5-methyl-5H-pyrrolo[3,2-d]pyrimidin-4-yl)oxy)phenyl)-1H-benzimidazol-2-amine | n/a | |
| 60 | Q9Y233_6DW | 6DW | n/a | 56654131 | CHEMBL3814662 | 1-(cyclopropylmethyl)-5-(2-(2,3-dihydro-1H-imidazo[1,2-a]benzimidazol-1-yl)ethoxy)-3-(1-phenyl-1H-pyrazol-5-yl)pyridazin-4(1H)-one | n/a | |
| 61 | Q9Y233_6RC | 6RC | n/a | 137348513 | n/a | 4-[5-[1-(2-methoxyethyl)pyrazol-4-yl]-2-(quinolin-2-yloxymethyl)imidazo[1,2-a]pyrazin-8-yl]morpholine | n/a | |
| 62 | Q9Y233_7ZE | 7ZE | n/a | 11829 | CHEMBL164449 | 5-nitroquinoline | n/a | |
| 63 | Q9Y233_8G3 | 8G3 | n/a | n/a | CHEMBL5273736 | 2-methyl-5-[2-([1,2,4]triazolo[1,5-a]pyrimidin-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-ol | n/a | |
| 64 | Q9Y233_8G6 | 8G6 | n/a | 735871 | CHEMBL4453824 | 7-(4-chlorophenyl)-2-methyl-pyrazolo[1,5-a]pyrimidine | n/a | |
| 65 | Q9Y233_8Q7 | 8Q7 | n/a | 126842986 | n/a | 9-[(1S)-2,2-difluorocyclopropane-1-carbonyl]-6-[(4-methoxyphenyl)methyl]-8,9,10,11-tetrahydropyrido[4',3':4,5]thieno[3,2-e][1,2,4]triazolo[1,5-c]pyrimidin-5(6H)-one | n/a | |
| 66 | Q9Y233_8ZE | 8ZE | n/a | 2776174 | CHEMBL4582404 | 2,3-dihydro-1,4-benzodioxin-6-ylmethanol | n/a | |
| 67 | Q9Y233_9G6 | 9G6 | n/a | 137332065 | CHEMBL4437555 | N-[2-(7-methoxy-4-morpholin-4-yl-quinazolin-6-yl)oxyethyl]-1,3-benzothiazol-2-amine | n/a | |
| 68 | Q9Y233_9ZE | 9ZE | n/a | 76143 | CHEMBL4557075 | 1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethanone | n/a | |
| 69 | Q9Y233_AEL | AEL | n/a | 137700779 | CHEMBL4558162 | 2-{2-[5-methyl-1-(pyridin-4-yl)-1H-benzimidazol-2-yl]ethyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione | n/a | |
| 70 | Q9Y233_AEO | AEO | n/a | 2884317 | CHEMBL4435239 | 2-[2-(4-phenyl-5-sulfanylidene-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-1H-benzo[de]isoquinoline-1,3(2H)-dione | n/a | |
| 71 | Q9Y233_AMP | AMP | DB00131 | 6083 | CHEMBL752 | ADENOSINE MONOPHOSPHATE | n/a | |
| 72 | Q9Y233_AXC | AXC | n/a | 50993785 | CHEMBL1641615 | 5-(1H-BENZIMIDAZOL-2-YLMETHYLSULFANYL)-2-METHYL-[1,2,4]TRIAZOLO[1,5-C]QUINAZOLINE | n/a | |
| 73 | Q9Y233_BR | BR | n/a | 259 | n/a | BROMIDE ION | n/a | |
| 74 | Q9Y233_C1L | C1L | n/a | 44243146 | CHEMBL1939914 | 6-methoxy-3,8-dimethyl-4-(morpholin-4-ylmethyl)-1H-pyrazolo[3,4-b]quinoline | n/a | |
| 75 | Q9Y233_CL | CL | n/a | 312 | n/a | CHLORIDE ION | n/a | |
| 76 | Q9Y233_CMP | CMP | DB02527 | 6076 | CHEMBL316966 | ADENOSINE-3',5'-CYCLIC-MONOPHOSPHATE | n/a | |
| 77 | Q9Y233_D6X | D6X | n/a | 138857395 | CHEMBL4446268 | N-[2-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)ethyl]quinolin-2-amine | n/a | |
| 78 | Q9Y233_D79 | D79 | n/a | n/a | CHEMBL4469155 | 4-[2-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)ethyl]-3,7,8,10-tetrazatricyclo[7.4.0.0^{2,7}]trideca-1,3,5,8,10,12-hexaen-6-ol | n/a | |
| 79 | Q9Y233_D7C | D7C | n/a | 138857397 | CHEMBL4559232 | 2-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-1-[(2S)-2-methyl-1,2-dihydroimidazo[1,2-a]benzimidazol-3-yl]ethanone | n/a | |
| 80 | Q9Y233_DKU | DKU | n/a | 146014934 | CHEMBL5280875 | 3-[2-(5-methyl-1-phenyl-benzimidazol-2-yl)ethyl]chromen-4-one | n/a | |
| 81 | Q9Y233_DL0 | DL0 | n/a | 146014935 | CHEMBL5274332 | 6-chloranyl-3-[2-(5-methyl-1-phenyl-benzimidazol-2-yl)ethyl]chromen-4-one | n/a | |
| 82 | Q9Y233_DZU | DZU | n/a | 154700483 | n/a | 8-[(E)-2-[5-methyl-1-[3-[3-(4-methylpiperazin-1-yl)propoxy]phenyl]benzimidazol-2-yl]ethenyl]quinoline | n/a | |
| 83 | Q9Y233_EDO | EDO | n/a | 174 | CHEMBL457299 | 1,2-ETHANEDIOL | n/a | |
| 84 | Q9Y233_EEI | EEI | n/a | 44548780 | CHEMBL3700112 | 5,7-dimethyl-2-[(1-methyl-4-phenyl-imidazol-2-yl)sulfanylmethyl]imidazo[1,2-a]pyrimidine | n/a | |
| 85 | Q9Y233_EFJ | EFJ | n/a | 1415219 | CHEMBL4164176 | 2-(1~{H}-benzimidazol-2-ylsulfanylmethyl)-3-bromanyl-5,7-dimethyl-imidazo[1,2-a]pyrimidine | n/a | |
| 86 | Q9Y233_EHI | EHI | n/a | 44547519 | CHEMBL3703517 | 8-methyl-2-[2-(1-methyl-4-phenyl-imidazol-2-yl)ethyl]-[1,2,4]triazolo[1,5-a]pyridine | n/a | |
| 87 | Q9Y233_EIH | EIH | n/a | 44549080 | CHEMBL3700126 | 2-[(1-methyl-4-phenyl-imidazol-2-yl)methylsulfanyl]-[1,2,4]triazolo[1,5-a]pyridine | n/a | |
| 88 | Q9Y233_EIK | EIK | n/a | 44537944 | CHEMBL2180414 | 5,8-dimethyl-2-[2-(1-methyl-4-phenyl-imidazol-2-yl)ethyl]-[1,2,4]triazolo[1,5-a]pyrazine | n/a | |
| 89 | Q9Y233_EV1 | EV1 | DB01113 | 4680 | CHEMBL19224 | 1-(3,4-DIMETHOXYBENZYL)-6,7-DIMETHOXYISOQUINOLINE | inhibitor | IC50(nM) = 17.0 |
| 90 | Q9Y233_F03 | F03 | n/a | 12603606;135566643; | CHEMBL6804 | N-(4-OXO-3H-QUINAZOLIN-2-YL)ACETAMIDE | n/a | |
| 91 | Q9Y233_F04 | F04 | n/a | 70789260 | n/a | 2-ETHYL-4-METHYL-PHTHALAZIN-1-ONE | n/a | |
| 92 | Q9Y233_F07 | F07 | n/a | 901686 | n/a | THIENO[3,2-C][1,6]NAPHTHYRIDINE | n/a | |
| 93 | Q9Y233_GIQ | GIQ | n/a | 53462 | CHEMBL1233049 | 3-METHYL-3H-IMIDAZO[4,5-F]QUINOLIN-2-AMINE | n/a | |
| 94 | Q9Y233_GOL | GOL | DB09462 | 753 | CHEMBL692 | GLYCEROL | n/a | |
| 95 | Q9Y233_I9Z | I9Z | n/a | 165368446 | n/a | 5-methyl-4-[2-(1-methyl-4-phenyl-1H-imidazol-2-yl)ethyl]-2-phenyl-1,3-oxazole | n/a | |
| 96 | Q9Y233_IAI | IAI | n/a | 53377588 | n/a | 1-methyl-N~4~-[(1,3-oxazol-4-yl)methyl]-N~5~-[(4R)-2-phenylimidazo[1,2-a]pyrimidin-7-yl]-1H-pyrazole-4,5-dicarboxamide | n/a | |
| 97 | Q9Y233_IAL | IAL | n/a | 165368447 | n/a | N~4~,N~4~,1-trimethyl-N~5~-(2-phenyl-1H-benzimidazol-5-yl)-1H-pyrazole-4,5-dicarboxamide | n/a | |
| 98 | Q9Y233_IAY | IAY | n/a | n/a | n/a | 4-(6-{2-[(4S)-1-methyl-4-phenyl-4,5-dihydro-1H-imidazol-2-yl]ethyl}pyridin-2-yl)morpholine | n/a | |
| 99 | Q9Y233_IB4 | IB4 | n/a | 123958596 | n/a | 6-cyclopropyl-N-[5-(dimethylcarbamoyl)-1-(2-methoxyethyl)-1H-pyrazol-4-yl]-3-[(pyrimidin-5-yl)amino]pyridine-2-carboxamide | n/a | |
| 100 | Q9Y233_IB7 | IB7 | n/a | 165368449 | n/a | 6-cyclopropyl-N-(3-{[(2S)-2,3-dihydroxypropyl](methyl)carbamoyl}-1-methyl-1H-pyrazol-4-yl)-3-[(pyrimidin-5-yl)amino]pyridine-2-carboxamide | n/a | |
| 101 | Q9Y233_IBJ | IBJ | n/a | 53328253 | CHEMBL3642183 | 6-cyclopropyl-N-[1-(2-hydroxyethyl)-3-(pyridin-2-yl)-1H-pyrazol-5-yl]-3-[(pyrimidin-5-yl)amino]pyridine-2-carboxamide | n/a | |
| 102 | Q9Y233_IBV | IBV | n/a | 58548370 | CHEMBL2180801 | 6-cyclopropyl-N-[3-(dimethylcarbamoyl)-1-methyl-1H-pyrazol-4-yl]-3-[(pyrimidin-5-yl)amino]pyridine-2-carboxamide | n/a | |
| 103 | Q9Y233_IBY | IBY | n/a | 70648564 | n/a | 2-[2-(1-methyl-4-phenyl-1H-imidazol-2-yl)ethyl]quinoline | n/a | |
| 104 | Q9Y233_ICK | ICK | n/a | 165368450 | n/a | 2-chloro-N-[(4S)-2-phenyl[1,2,4]triazolo[1,5-a]pyridin-7-yl]pyridine-4-carboxamide | n/a | |
| 105 | Q9Y233_ICW | ICW | n/a | 165368451 | n/a | (8S)-5-cyclopropyl-7-methyl-2-[2-(1-methyl-4-phenyl-1H-imidazol-2-yl)ethyl][1,2,4]triazolo[1,5-a]pyrimidine | n/a | |
| 106 | Q9Y233_ID9 | ID9 | n/a | 118278218 | n/a | (4R)-2,3-dimethyl-6-[(1-methyl-4-phenyl-1H-imidazol-2-yl)methoxy]imidazo[1,2-b]pyridazine | n/a | |
| 107 | Q9Y233_IE1 | IE1 | n/a | 165368452 | n/a | 4-(azetidine-1-carbonyl)-2-methyl-N-[2-(1-methyl-3-phenyl-1H-1,2,4-triazol-5-yl)ethyl]-2,5-dihydro-1H-pyrazole-3-carboxamide | n/a | |
| 108 | Q9Y233_IE7 | IE7 | n/a | 57378955 | n/a | 4-(azetidine-1-carbonyl)-1-methyl-N-[(4S)-2-phenyl[1,2,4]triazolo[1,5-a]pyridin-7-yl]-1H-pyrazole-5-carboxamide | n/a | |
| 109 | Q9Y233_IEB | IEB | n/a | 165368453 | n/a | 2,9-dimethyl-6-[(1-methyl-4-phenyl-1H-imidazol-2-yl)methoxy]-9H-purine | n/a | |
| 110 | Q9Y233_IEH | IEH | n/a | 54761299 | CHEMBL3685539 | 6-cyclopropyl-N-[1-methyl-5-(methylcarbamoyl)-1H-pyrazol-4-yl]-3-[(pyrimidin-5-yl)amino]pyrazine-2-carboxamide | n/a | |
| 111 | Q9Y233_IEN | IEN | n/a | 165368454 | n/a | 6-cyclopropyl-N-[1-(pyridin-2-yl)-1H-pyrazol-5-yl]-3-[(pyrimidin-5-yl)amino]pyridine-2-carboxamide | n/a | |
| 112 | Q9Y233_IEU | IEU | n/a | 165416121 | n/a | 6-chloro-2-{[(4S)-1-methyl-4-phenyl-4,5-dihydro-1H-imidazol-2-yl]methoxy}-4-(morpholin-4-yl)quinazoline | n/a | |
| 113 | Q9Y233_IEX | IEX | n/a | 165368456 | n/a | 2-[2-(1,4-diphenyl-1H-imidazol-2-yl)ethyl]-3-methylquinoxaline | n/a | |
| 114 | Q9Y233_IF2 | IF2 | n/a | 72704532 | CHEMBL3940291 | 2-methyl-3-{2-[1-methyl-3-(pyrrolidin-1-yl)-1H-1,2,4-triazol-5-yl]ethyl}quinoxaline | n/a | |
| 115 | Q9Y233_IF5 | IF5 | n/a | 165368457 | n/a | 6-cyclopropyl-N-(1-phenyl-1H-pyrazol-5-yl)-3-[(pyrimidin-5-yl)amino]pyridine-2-carboxamide | n/a | |
| 116 | Q9Y233_IFE | IFE | n/a | 123548203 | n/a | (4R)-6-chloro-2-{(E)-2-[1-methyl-3-(pyrrolidin-1-yl)-1H-1,2,4-triazol-5-yl]ethenyl}[1,2,4]triazolo[1,5-a]pyridine | n/a | |
| 117 | Q9Y233_IFI | IFI | n/a | 57377303 | n/a | 4-(azetidine-1-carbonyl)-1-methyl-N-[(4S)-2-(morpholin-4-yl)[1,2,4]triazolo[1,5-a]pyridin-7-yl]-1H-pyrazole-5-carboxamide | n/a | |
| 118 | Q9Y233_IFN | IFN | n/a | 165368458 | n/a | 5-[(5-bromo-1-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)amino]-N-(oxetan-3-yl)-2-phenyl-1H-benzimidazole-6-carboxamide | n/a | |
| 119 | Q9Y233_IFR | IFR | n/a | 72704900 | CHEMBL3975467 | (4R)-5,7,8-trimethyl-2-{2-[1-methyl-3-(pyrrolidin-1-yl)-1H-1,2,4-triazol-5-yl]ethyl}[1,2,4]triazolo[1,5-c]pyrimidine | n/a | |
| 120 | Q9Y233_IFV | IFV | n/a | 90026630 | CHEMBL3956406 | (4R)-6-chloro-2-{2-[1-methyl-3-(pyrrolidin-1-yl)-1H-1,2,4-triazol-5-yl]ethyl}[1,2,4]triazolo[1,5-a]pyridine | n/a | |
| 121 | Q9Y233_IFY | IFY | n/a | 165368459 | n/a | 2-methyl-3-[2-(1-methyl-4-phenyl-1H-imidazol-2-yl)ethyl]quinoxaline | n/a | |
| 122 | Q9Y233_IG1 | IG1 | n/a | 165368460 | n/a | 4-(azetidine-1-carbonyl)-1-methyl-N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]-1H-pyrazole-5-carboxamide | n/a | |
| 123 | Q9Y233_IG6 | IG6 | n/a | 118278237 | n/a | (4S)-3-methyl-6-[2-(1-methyl-4-phenyl-1H-imidazol-2-yl)ethyl]-2-(trifluoromethyl)imidazo[1,2-b]pyridazine | n/a | |
| 124 | Q9Y233_IG9 | IG9 | n/a | 165368461 | n/a | 4-(azetidine-1-carbonyl)-1-methyl-N-[1-(quinolin-2-yl)-1H-imidazol-4-yl]-1H-pyrazole-5-carboxamide | n/a | |
| 125 | Q9Y233_IGE | IGE | n/a | 22563291 | n/a | 2-[2-(4-methyl-2-phenyl-1H-imidazol-5-yl)ethyl]-1H-isoindole-1,3(2H)-dione | n/a | |
| 126 | Q9Y233_IGI | IGI | n/a | 165368462 | n/a | (4S)-2-[2-(4-cyclopentyl-1-methyl-1H-imidazol-2-yl)ethyl]-5,8-dimethyl[1,2,4]triazolo[1,5-a]pyrazine | n/a | |
| 127 | Q9Y233_IGO | IGO | n/a | 72704899 | CHEMBL3912952 | (4S)-5,6,8-trimethyl-2-{2-[1-methyl-3-(pyrrolidin-1-yl)-1H-1,2,4-triazol-5-yl]ethyl}[1,2,4]triazolo[1,5-a]pyrazine | n/a | |
| 128 | Q9Y233_IGW | IGW | n/a | 57377631 | n/a | N~4~-(2-fluoroethyl)-N~4~,1-dimethyl-N~5~-[(4S)-2-phenyl[1,2,4]triazolo[1,5-a]pyridin-7-yl]-1H-pyrazole-4,5-dicarboxamide | n/a | |
| 129 | Q9Y233_IGZ | IGZ | n/a | 165368463 | n/a | 4-(azetidine-1-carbonyl)-1-methyl-N-[(4R,7R)-2-phenyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-7-yl]-1H-pyrazole-5-carboxamide | n/a | |
| 130 | Q9Y233_IH8 | IH8 | n/a | 53328251 | CHEMBL3642181 | 6-cyclopropyl-N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]-3-[(pyrimidin-5-yl)amino]pyridine-2-carboxamide | n/a | |
| 131 | Q9Y233_IHL | IHL | n/a | 165368464 | n/a | (4R)-2-{2-[1-methyl-3-(pyrrolidin-1-yl)-1H-1,2,4-triazol-5-yl]ethyl}-6-(trifluoromethyl)[1,2,4]triazolo[1,5-a]pyridine | n/a | |
| 132 | Q9Y233_IHV | IHV | n/a | n/a | n/a | 2,3,5-trimethyl-6-{2-[(4S)-1-methyl-4-phenyl-4,5-dihydro-1H-imidazol-2-yl]ethyl}pyrazine | n/a | |
| 133 | Q9Y233_II5 | II5 | n/a | 54761643 | CHEMBL3685439 | 6-cyclopropyl-N-[1-(2-methoxyethyl)-5-(methylcarbamoyl)-1H-pyrazol-4-yl]-3-[(pyrimidin-5-yl)amino]pyridine-2-carboxamide | n/a | |
| 134 | Q9Y233_II9 | II9 | n/a | 165368466 | n/a | N-methyl-6-[(6-methylpyridine-2-carbonyl)amino]-2-phenyl-1H-benzimidazole-5-carboxamide | n/a | |
| 135 | Q9Y233_IIR | IIR | n/a | 118278240 | n/a | {(4S)-2-cyclopropyl-6-[(1-methyl-4-phenyl-1H-imidazol-2-yl)ethynyl]imidazo[1,2-b]pyridazin-3-yl}methanol | n/a | |
| 136 | Q9Y233_IIU | IIU | n/a | 165368467 | n/a | 2-chloro-6-ethyl-N-[(4S)-2-phenyl[1,2,4]triazolo[1,5-a]pyridin-7-yl]pyridine-4-carboxamide | n/a | |
| 137 | Q9Y233_IIX | IIX | n/a | 165368468 | n/a | 4-(azetidine-1-carbonyl)-1-methyl-N-[5-(pyridin-2-yl)-1H-pyrazol-3-yl]-1H-pyrazole-5-carboxamide | n/a | |
| 138 | Q9Y233_IJ0 | IJ0 | n/a | 118278206 | n/a | (4S)-2-(difluoromethyl)-3-methyl-6-[(1-methyl-4-phenyl-1H-imidazol-2-yl)ethynyl]imidazo[1,2-b]pyridazine | n/a | |
| 139 | Q9Y233_IJ7 | IJ7 | n/a | 165368469 | n/a | 6-cyclopropyl-N-(3-oxo-2,3-dihydro-1H-isoindol-5-yl)-3-[(pyrimidin-5-yl)amino]pyridine-2-carboxamide | n/a | |
| 140 | Q9Y233_IJA | IJA | n/a | 67388123 | n/a | 1-methyl-N~5~-[(4S)-2-phenylimidazo[1,2-a]pyrimidin-7-yl]-N~4~-[(1H-pyrazol-3-yl)methyl]-1H-pyrazole-4,5-dicarboxamide | n/a | |
| 141 | Q9Y233_IJD | IJD | n/a | 53328445 | CHEMBL3639410 | 6-cyclopropyl-N-{1-[2-(dimethylamino)ethyl]-3-(pyridin-2-yl)-1H-pyrazol-5-yl}-3-[(pyrimidin-5-yl)amino]pyridine-2-carboxamide | n/a | |
| 142 | Q9Y233_IJH | IJH | n/a | 118278153 | n/a | (4S)-2,3-dimethyl-6-[2-(1-methyl-4-phenyl-1H-imidazol-2-yl)ethyl]imidazo[1,2-b]pyridazine | n/a | |
| 143 | Q9Y233_IJK | IJK | n/a | 90154187 | n/a | (8S)-6,7-dimethyl-2-{2-[1-methyl-3-(pyrrolidin-1-yl)-1H-1,2,4-triazol-5-yl]ethyl}-N-(propan-2-yl)imidazo[2,1-f][1,2,4]triazin-4-amine | n/a | |
| 144 | Q9Y233_IJN | IJN | n/a | 165368470 | n/a | (10S)-1-(2-chlorophenyl)-8-methoxy-3,4-dimethylimidazo[1,5-a]quinazolin-5(4H)-one | n/a | |
| 145 | Q9Y233_IJQ | IJQ | n/a | 71288719 | CHEMBL3649576 | 4-(azetidine-1-carbonyl)-1-methyl-N-{2-[3-phenyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-pyrazole-5-carboxamide | n/a | |
| 146 | Q9Y233_IJT | IJT | n/a | n/a | n/a | 2-methyl-3-{[(4R)-1-methyl-4-phenyl-4,5-dihydro-1H-imidazol-2-yl]methoxy}quinoxaline | n/a | |
| 147 | Q9Y233_IJW | IJW | n/a | n/a | n/a | 6-cyclopropyl-3-{[(4S)-1-methyl-4-phenyl-4,5-dihydro-1H-imidazol-2-yl]methoxy}-N-[(3R)-oxolan-3-yl]pyrazine-2-carboxamide | n/a | |
| 148 | Q9Y233_IK0 | IK0 | n/a | 75201281 | n/a | (4S)-N,2,3-trimethyl-6-{2-[1-methyl-3-(pyrrolidin-1-yl)-1H-1,2,4-triazol-5-yl]ethyl}imidazo[1,2-b]pyridazine-8-carboxamide | n/a | |
| 149 | Q9Y233_IK6 | IK6 | n/a | n/a | n/a | 3-(azetidin-1-ylcarbonyl)-2-methyl-~{N}-(2-phenyl-2,3-dihydro-1~{H}-imidazo[1,2-a]pyrimidin-7-yl)-1,5-dihydropyrazole-4-carboxamide | n/a | |
| 150 | Q9Y233_IKB | IKB | n/a | 72705091 | CHEMBL3915989 | (4S)-5,8-dimethyl-2-{2-[1-methyl-3-(piperidin-1-yl)-1H-1,2,4-triazol-5-yl]ethyl}[1,2,4]triazolo[1,5-a]pyrazine | n/a | |
| 151 | Q9Y233_IKE | IKE | n/a | 68238816 | n/a | N~4~,1-dimethyl-N~5~-[(4R)-2-phenylimidazo[1,2-a]pyrimidin-7-yl]-1H-pyrazole-4,5-dicarboxamide | n/a | |
| 152 | Q9Y233_IKH | IKH | n/a | 91826747 | n/a | {(4S)-2-methyl-6-[(1-methyl-4-phenyl-1H-imidazol-2-yl)ethynyl]imidazo[1,2-b]pyridazin-3-yl}methanol | n/a | |
| 153 | Q9Y233_IKK | IKK | n/a | 165368474 | n/a | N-[(3R)-1-(5-chloropyridin-2-yl)pyrrolidin-3-yl]-6-cyclopropyl-3-[(pyrimidin-5-yl)amino]pyridine-2-carboxamide | n/a | |
| 154 | Q9Y233_IKO | IKO | n/a | 90016837 | CHEMBL3891571 | N-cyclopropyl-5-{2-[(4S)-5,8-dimethyl[1,2,4]triazolo[1,5-a]pyrazin-2-yl]ethyl}-N,1-dimethyl-1H-1,2,4-triazol-3-amine | n/a | |
| 155 | Q9Y233_IKU | IKU | n/a | 72705093 | CHEMBL3932717 | (4S)-5,8-dimethyl-2-(2-{1-methyl-3-[(2S)-2-methylpyrrolidin-1-yl]-1H-1,2,4-triazol-5-yl}ethyl)[1,2,4]triazolo[1,5-a]pyrazine | n/a | |
| 156 | Q9Y233_IKZ | IKZ | n/a | 53468844 | n/a | 1-methyl-N~5~-[(4R)-2-phenylimidazo[1,2-a]pyrimidin-7-yl]-N~4~-[(pyridin-2-yl)methyl]-1H-pyrazole-4,5-dicarboxamide | n/a | |
| 157 | Q9Y233_IL6 | IL6 | n/a | 165368475 | n/a | 6-cyclopropyl-3-[(pyrimidin-5-yl)amino]-N-[1-(2,2,2-trifluoroethyl)-1H-pyrazol-3-yl]pyridine-2-carboxamide | n/a | |
| 158 | Q9Y233_IL9 | IL9 | n/a | 54761297 | CHEMBL3685542 | 6-cyclopropyl-N-{5-[(2-hydroxy-2-methylpropyl)carbamoyl]-1-methyl-1H-pyrazol-4-yl}-3-[(pyrimidin-5-yl)amino]pyrazine-2-carboxamide | n/a | |
| 159 | Q9Y233_ILN | ILN | n/a | 165368476 | n/a | 1-methyl-4-(morpholine-4-carbonyl)-N-[(4S)-2-phenyl[1,2,4]triazolo[1,5-c]pyrimidin-7-yl]-1H-pyrazole-5-carboxamide | n/a | |
| 160 | Q9Y233_ILS | ILS | n/a | 71288499 | CHEMBL3649521 | 4-(azetidine-1-carbonyl)-1-methyl-N-[2-(1-methyl-1H-benzimidazol-2-yl)ethyl]-1H-pyrazole-5-carboxamide | n/a | |
| 161 | Q9Y233_ILZ | ILZ | n/a | n/a | n/a | 4-(azetidine-1-carbonyl)-2-methyl-N-{2-[(4S)-1-methyl-4-phenyl-4,5-dihydro-1H-imidazol-2-yl]ethyl}-2,5-dihydro-1H-pyrazole-3-carboxamide | n/a | |
| 162 | Q9Y233_IO4 | IO4 | n/a | 165368478 | n/a | (8S)-N-(2-chloropyridin-4-yl)-2-phenylpyrazolo[1,5-a]pyridine-6-carboxamide | n/a | |
| 163 | Q9Y233_IO7 | IO7 | n/a | 165368479 | n/a | 4-(azetidine-1-carbonyl)-N-[1-(2,2-difluoroethyl)-1H-pyrazol-3-yl]-1-methyl-1H-pyrazole-5-carboxamide | n/a | |
| 164 | Q9Y233_IOI | IOI | n/a | 87383148 | n/a | N~4~-ethyl-N~5~-{(4S)-2-[3-(2-fluoroethoxy)phenyl]imidazo[1,2-a]pyrimidin-7-yl}-N~4~,1-dimethyl-1H-pyrazole-4,5-dicarboxamide | n/a | |
| 165 | Q9Y233_IOU | IOU | n/a | 90016429 | n/a | (4S)-5,8-dimethyl-2-(2-{1-methyl-3-[(3S)-3-methylpyrrolidin-1-yl]-1H-1,2,4-triazol-5-yl}ethyl)[1,2,4]triazolo[1,5-a]pyrazine | n/a | |
| 166 | Q9Y233_IOZ | IOZ | n/a | 90018195 | CHEMBL3931252 | (4S)-5,8-dimethyl-2-{2-[1-methyl-5-(pyrrolidin-1-yl)-1H-1,2,4-triazol-3-yl]ethyl}[1,2,4]triazolo[1,5-a]pyrazine | n/a | |
| 167 | Q9Y233_IQ3 | IQ3 | n/a | 54760571 | CHEMBL3685449 | 6-cyclopropyl-3-[(pyrimidin-5-yl)amino]-N-[4-(pyrrolidine-1-carbonyl)pyridin-3-yl]pyridine-2-carboxamide | n/a | |
| 168 | Q9Y233_IQ9 | IQ9 | n/a | 165368480 | n/a | 4-(azetidine-1-carbonyl)-N-(1-cyclopentyl-1H-pyrazol-3-yl)-1-methyl-1H-pyrazole-5-carboxamide | n/a | |
| 169 | Q9Y233_IQF | IQF | n/a | 72705092 | CHEMBL3947336 | (4R)-5-ethyl-8-methyl-2-{2-[1-methyl-3-(pyrrolidin-1-yl)-1H-1,2,4-triazol-5-yl]ethyl}[1,2,4]triazolo[1,5-c]pyrimidine | n/a | |
| 170 | Q9Y233_IQJ | IQJ | n/a | 165368481 | n/a | N-(2-acetamido-1,3-benzothiazol-5-yl)-4-(azetidine-1-carbonyl)-1-methyl-1H-pyrazole-5-carboxamide | n/a | |
| 171 | Q9Y233_IQV | IQV | n/a | n/a | n/a | (4S)-5,8-dimethyl-2-{(E)-2-[1-methyl-3-(1H-pyrazol-4-yl)-1H-1,2,4-triazol-5-yl]ethenyl}[1,2,4]triazolo[1,5-a]pyrazine | n/a | |
| 172 | Q9Y233_IV0 | IV0 | n/a | 165368483 | n/a | N-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethyl]-N'-(1-phenyl-1H-pyrazol-5-yl)urea | n/a | |
| 173 | Q9Y233_IV4 | IV4 | n/a | 165368484 | n/a | 1-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethyl]-3-(1-phenyl-1H-pyrazol-5-yl)-1,3-dihydro-2H-imidazol-2-one | n/a | |
| 174 | Q9Y233_IV8 | IV8 | n/a | 90033536 | CHEMBL3955474 | (10R)-2-{2-[1-methyl-3-(pyrrolidin-1-yl)-1H-1,2,4-triazol-5-yl]ethyl}[1,2,4]triazolo[1,5-a]quinoline | n/a | |
| 175 | Q9Y233_IVE | IVE | n/a | 165368485 | n/a | (2S)-N'-[(4-bromo-3,5-dimethoxyphenyl)methyl]-2-ethoxy-2-[4-(morpholin-4-yl)phenyl]acetohydrazide | n/a | |
| 176 | Q9Y233_IVJ | IVJ | n/a | 165368486 | n/a | N~5~-[2-(3-chlorophenyl)-1H-benzimidazol-5-yl]-1-methyl-1H-pyrazole-4,5-dicarboxamide | n/a | |
| 177 | Q9Y233_IVP | IVP | n/a | 1454127;135429167; | n/a | N-[(4-methoxyphenyl)methyl]-N'-(4-methylphenyl)-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]urea | n/a | |
| 178 | Q9Y233_IVT | IVT | n/a | 72704531 | CHEMBL3981364 | (4S)-5,8-dimethyl-2-{2-[1-methyl-3-(pyrrolidin-1-yl)-1H-1,2,4-triazol-5-yl]ethyl}[1,2,4]triazolo[1,5-a]pyrazine | n/a | |
| 179 | Q9Y233_IVY | IVY | n/a | 46219816 | n/a | 3-[1-(2-fluorophenyl)-1H-pyrazol-5-yl]-1-[3-(trifluoromethyl)phenyl]pyridazin-4(1H)-one | n/a | |
| 180 | Q9Y233_IW9 | IW9 | n/a | 45094256 | n/a | 5-butoxy-4-ethoxypyrimidin-2-amine | n/a | |
| 181 | Q9Y233_IWC | IWC | n/a | 72706417 | n/a | 2-{(E)-2-[4-methyl-6-(pyrrolidin-1-yl)pyrimidin-2-yl]ethenyl}quinoline | n/a | |
| 182 | Q9Y233_IWG | IWG | n/a | 1476043 | n/a | 5-[(4-chloronaphthalen-1-yl)oxy]-1,2,3-thiadiazole | n/a | |
| 183 | Q9Y233_IWK | IWK | n/a | 165368487 | n/a | 4-(azetidine-1-carbonyl)-1-methyl-N-[(4S)-2-(morpholin-4-yl)[1,2,4]triazolo[1,5-c]pyrimidin-7-yl]-1H-pyrazole-5-carboxamide | n/a | |
| 184 | Q9Y233_IWN | IWN | n/a | 165368488 | n/a | 4-(methoxymethyl)-1-methyl-N-[(4S)-2-phenyl[1,2,4]triazolo[1,5-a]pyridin-7-yl]-1H-pyrazole-5-carboxamide | n/a | |
| 185 | Q9Y233_IWS | IWS | n/a | 19813289 | n/a | (4R,10aP)-imidazo[1,2-c]quinazolin-5(6H)-one | n/a | |
| 186 | Q9Y233_IWY | IWY | n/a | 165368489 | n/a | ethyl 1-methyl-5-(propylcarbamoyl)-1H-pyrazole-4-carboxylate | n/a | |
| 187 | Q9Y233_IX2 | IX2 | n/a | 165368490 | n/a | 2-{[(4-chloro-3,5-dimethylpyridin-2-yl)methyl]sulfanyl}-6,7-dihydro-1H-furo[2,3-f]benzimidazole | n/a | |
| 188 | Q9Y233_IX5 | IX5 | n/a | 165368491 | n/a | 1-methyl-6-[(1-methyl-4-phenyl-1H-imidazol-2-yl)methoxy]-4-(morpholin-4-yl)-1H-pyrazolo[3,4-d]pyrimidine | n/a | |
| 189 | Q9Y233_IX9 | IX9 | n/a | 165412413 | n/a | 6-(3-methylphenoxy)-2-[4-(pyridin-2-yl)piperazin-1-yl]-9H-purine | n/a | |
| 190 | Q9Y233_IXI | IXI | n/a | 165368492 | n/a | 5-[(3,6-dimethylpyridine-2-carbonyl)amino]-N-methyl-2-phenyl-1H-benzimidazole-6-carboxamide | n/a | |
| 191 | Q9Y233_IXL | IXL | n/a | 165368493 | n/a | 4-(azetidine-1-carbonyl)-1-methyl-N-[(4R,7R)-2-(2-methylphenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-7-yl]-1H-pyrazole-5-carboxamide | n/a | |
| 192 | Q9Y233_IXT | IXT | n/a | 165368494 | n/a | (2S)-N'-[(E)-(4-bromo-3,5-dimethoxyphenyl)methylidene]-2-ethoxy-2-[4-(1H-pyrazol-1-yl)phenyl]acetohydrazide | n/a | |
| 193 | Q9Y233_IY2 | IY2 | n/a | 51033483 | n/a | N~5~-[(4R)-2-(4-fluorophenyl)imidazo[1,2-a]pyridin-7-yl]-N~4~,N~4~,1-trimethyl-1H-pyrazole-4,5-dicarboxamide | n/a | |
| 194 | Q9Y233_IY6 | IY6 | n/a | 90135404 | n/a | (4S)-2,3-dimethyl-6-{2-[1-methyl-3-(pyrrolidin-1-yl)-1H-1,2,4-triazol-5-yl]ethyl}-7-(trifluoromethyl)imidazo[1,2-b]pyridazine | n/a | |
| 195 | Q9Y233_IYA | IYA | n/a | 11647802 | n/a | N-[3-(3-{[5-(4-fluorophenyl)thieno[2,3-d]pyrimidin-4-yl]oxy}propoxy)phenyl]acetamide | n/a | |
| 196 | Q9Y233_IYD | IYD | n/a | 51034483 | n/a | N~4~-(2-methoxyethyl)-N~4~,1-dimethyl-N~5~-[(4R)-2-phenylimidazo[1,2-a]pyridin-7-yl]-1H-pyrazole-4,5-dicarboxamide | n/a | |
| 197 | Q9Y233_IYK | IYK | n/a | 165368495 | n/a | 2-chloro-3-[(1-methyl-4-phenyl-1H-imidazol-2-yl)methoxy]quinoxaline | n/a | |
| 198 | Q9Y233_IYN | IYN | n/a | n/a | n/a | 2-methyl-3-{2-[(3S)-1-(pyridin-2-yl)pyrrolidin-3-yl]ethyl}quinoxaline | n/a | |
| 199 | Q9Y233_IYS | IYS | n/a | 1366773 | CHEMBL2180424 | 2-{2-[3-(4-methoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl]ethyl}-1H-isoindole-1,3(2H)-dione | n/a | |
| 200 | Q9Y233_IYW | IYW | n/a | 165368497 | n/a | 1-benzyl-3-(1-phenyl-1H-pyrazol-5-yl)pyridazin-4(1H)-one | n/a | |
| 201 | Q9Y233_IZ6 | IZ6 | n/a | 165368498 | n/a | 1-phenyl-3-(1-phenyl-1H-pyrazol-5-yl)-5,6-dihydropyridazin-4(1H)-one | n/a | |
| 202 | Q9Y233_IZH | IZH | n/a | 90017373 | n/a | (4S)-5,8-dimethyl-2-(2-{1-methyl-3-[(2R)-2-(trifluoromethyl)pyrrolidin-1-yl]-1H-1,2,4-triazol-5-yl}ethyl)[1,2,4]triazolo[1,5-c]pyrimidine | n/a | |
| 203 | Q9Y233_IZK | IZK | n/a | 67383693 | n/a | 4-chloro-1-(2-methylpropyl)-N-[(4R)-2-phenylimidazo[1,2-a]pyrimidin-7-yl]-1H-pyrazole-5-carboxamide | n/a | |
| 204 | Q9Y233_IZQ | IZQ | n/a | 110173677 | n/a | (10R)-9-(2-chlorophenyl)-2-methoxy-7-methylimidazo[1,5-a]pyrido[3,2-e]pyrazin-6(5H)-one | n/a | |
| 205 | Q9Y233_IZW | IZW | n/a | 165368499 | n/a | 8-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]quinoline | n/a | |
| 206 | Q9Y233_J0O | J0O | n/a | 165368500 | n/a | 4-(azetidine-1-carbonyl)-1-methyl-N-[2-(morpholin-4-yl)-1,3-benzothiazol-5-yl]-1H-pyrazole-5-carboxamide | n/a | |
| 207 | Q9Y233_J2L | J2L | n/a | 75201280 | n/a | (4S)-8-(methanesulfonyl)-2,3-dimethyl-6-{2-[1-methyl-3-(pyrrolidin-1-yl)-1H-1,2,4-triazol-5-yl]ethyl}imidazo[1,2-b]pyridazine | n/a | |
| 208 | Q9Y233_J4I | J4I | n/a | 165368501 | n/a | 6-{[(5-methoxy-3,4,6-trimethylpyridin-2-yl)methyl]sulfanyl}-2H,5H-[1,3]dioxolo[4,5-f]benzimidazole | n/a | |
| 209 | Q9Y233_J6I | J6I | n/a | 165368502 | n/a | 2-amino-4-{[(1S)-cyclohex-2-en-1-yl]oxy}quinoline-3-carbonitrile | n/a | |
| 210 | Q9Y233_J7M | J7M | n/a | 165368503 | n/a | 4-[2-(1-methyl-1H-benzimidazol-2-yl)ethyl]-3,4-dihydro-1,4-benzoxazepin-5(2H)-one | n/a | |
| 211 | Q9Y233_J8J | J8J | n/a | 165368504 | n/a | 5-[(5-cyclopropyl-2-oxo-1,2-dihydropyridine-3-carbonyl)amino]-N-(oxetan-3-yl)-2-phenyl-1H-benzimidazole-6-carboxamide | n/a | |
| 212 | Q9Y233_J9C | J9C | n/a | 165368505 | n/a | 6-methyl-N-(3-methyl-1-phenyl-1H-pyrazol-5-yl)-3-[(pyrimidin-5-yl)amino]pyridine-2-carboxamide | n/a | |
| 213 | Q9Y233_JAP | JAP | n/a | 90027123 | n/a | (4S)-2-(2-{3-[(3R)-3-fluoropyrrolidin-1-yl]-1-methyl-1H-1,2,4-triazol-5-yl}ethyl)-5,8-dimethyl[1,2,4]triazolo[1,5-a]pyrazine | n/a | |
| 214 | Q9Y233_JBV | JBV | n/a | 72703514 | CHEMBL3899676 | (4S)-2-(2-{3-[(3S)-3-(difluoromethyl)pyrrolidin-1-yl]-1-methyl-1H-1,2,4-triazol-5-yl}ethyl)-5,8-dimethyl[1,2,4]triazolo[1,5-a]pyrazine | n/a | |
| 215 | Q9Y233_JCJ | JCJ | n/a | 59453397 | n/a | 3-[1-(3-bromophenyl)-1H-pyrazol-5-yl]-1-(pyridin-4-yl)pyridazin-4(1H)-one | n/a | |
| 216 | Q9Y233_JCP | JCP | n/a | 54760757 | CHEMBL2180403 | 6-cyclopropyl-N-[4-(methylcarbamoyl)pyridin-3-yl]-3-[(pyrimidin-5-yl)amino]pyridine-2-carboxamide | n/a | |
| 217 | Q9Y233_JD6 | JD6 | n/a | 146053 | CHEMBL4548867 | 2,3-dimethylquinoxalin-6-amine | n/a | |
| 218 | Q9Y233_JDU | JDU | n/a | 165368507 | n/a | 1-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethyl]-2-oxo-N-(pyrimidin-5-yl)-1,2-dihydropyridine-3-carboxamide | n/a | |
| 219 | Q9Y233_JFG | JFG | n/a | 165368508 | n/a | 3,6-dimethyl-N-[(8R)-2-phenylpyrazolo[1,5-a]pyridin-6-yl]pyridine-2-carboxamide | n/a | |
| 220 | Q9Y233_JFO | JFO | n/a | 23624261 | n/a | (10R)-9-(2-chlorophenyl)-2-methoxy-7-methylimidazo[1,5-a]pyrido[3,2-e]pyrazin-6-amine | n/a | |
| 221 | Q9Y233_JFW | JFW | n/a | 165368509 | n/a | 7-{[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]sulfanyl}-8H-imidazo[4,5-g][1,3]benzothiazole | n/a | |
| 222 | Q9Y233_JG9 | JG9 | n/a | 165368510 | n/a | (4R)-2,3,5-trimethyl-6-[2-(1-methyl-4-phenyl-1H-imidazol-2-yl)ethyl]imidazo[1,2-a]pyridine | n/a | |
| 223 | Q9Y233_JGI | JGI | n/a | 165368511 | n/a | 4-(azetidine-1-carbonyl)-1-methyl-N-[3-(phenylcarbamoyl)phenyl]-1H-pyrazole-5-carboxamide | n/a | |
| 224 | Q9Y233_JH6 | JH6 | n/a | 16118696 | n/a | N-(6-methylpyridin-2-yl)-5-(pyridin-3-yl)-1,7-naphthyridin-8-amine | n/a | |
| 225 | Q9Y233_JHI | JHI | n/a | 135217363 | n/a | (4R)-6-chloro-2,3-dimethyl-8-(pyrrolidin-1-yl)imidazo[1,2-b]pyridazine | n/a | |
| 226 | Q9Y233_JHX | JHX | n/a | n/a | n/a | N-[(3R)-1-(5-chloropyridin-2-yl)pyrrolidin-3-yl]-6-cyclopropyl-3-methoxypyrazine-2-carboxamide | n/a | |
| 227 | Q9Y233_JI8 | JI8 | n/a | n/a | n/a | ~{N}4-(4,5-dihydro-1,3-oxazol-2-ylmethyl)-2-methyl-~{N}3-(2-phenyl-3~{H}-imidazo[1,2-a]pyrimidin-7-yl)-1,5-dihydropyrazole-3,4-dicarboxamide | n/a | |
| 228 | Q9Y233_JIC | JIC | n/a | 51034255 | n/a | N~4~-cyclopropyl-1-methyl-N~5~-[(4R)-2-phenylimidazo[1,2-a]pyridin-7-yl]-1H-pyrazole-4,5-dicarboxamide | n/a | |
| 229 | Q9Y233_JIG | JIG | n/a | 165368514 | n/a | 2-{[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]sulfanyl}-1H-imidazo[4,5-h]quinoline | n/a | |
| 230 | Q9Y233_JIJ | JIJ | n/a | 4428602 | CHEMBL4645765 | 4-(pyrrolidin-1-yl)-7H-pyrrolo[2,3-d]pyrimidine | n/a | |
| 231 | Q9Y233_JIP | JIP | n/a | 165412414 | n/a | N-{[(4R)-5,8-dimethyl[1,2,4]triazolo[1,5-a]pyrazin-2-yl]methyl}-N,1-dimethyl-3-phenyl-1H-1,2,4-triazol-5-amine | n/a | |
| 232 | Q9Y233_JIS | JIS | n/a | 5301054 | n/a | 3-[(naphthalen-1-yl)methyl]-7-(piperidin-1-yl)-3H-[1,2,3]triazolo[4,5-d]pyrimidine | n/a | |
| 233 | Q9Y233_JIV | JIV | n/a | 72705088 | CHEMBL3952690 | (4S)-8-chloro-5,7-dimethyl-2-{2-[1-methyl-3-(pyrrolidin-1-yl)-1H-1,2,4-triazol-5-yl]ethyl}[1,2,4]triazolo[1,5-c]pyrimidine | n/a | |
| 234 | Q9Y233_JIY | JIY | n/a | 165368515 | n/a | 2-{[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]sulfanyl}-1,5,6,7-tetrahydroimidazo[4,5-f]indole | n/a | |
| 235 | Q9Y233_JJ6 | JJ6 | n/a | 165368516 | n/a | [(4S)-2-phenyl[1,2,4]triazolo[1,5-a]pyridin-7-yl]methanol | n/a | |
| 236 | Q9Y233_JJF | JJF | n/a | 238490 | CHEMBL1450919 | 2-methyl-3-(pyrrolidin-1-yl)quinoxaline | n/a | |
| 237 | Q9Y233_JJR | JJR | n/a | 165368517 | n/a | {8-[(2-methyl-1,3-thiazol-4-yl)amino]-5-(pyridin-3-yl)-1,7-naphthyridin-2-yl}methanol | n/a | |
| 238 | Q9Y233_JK6 | JK6 | n/a | 46219698 | n/a | 3-[1-(3-ethynylphenyl)-1H-pyrazol-5-yl]-1-phenylpyridazin-4(1H)-one | n/a | |
| 239 | Q9Y233_JKD | JKD | n/a | 165368518 | n/a | (4R)-7-methyl-2,5-bis{2-[1-methyl-5-(pyrrolidin-1-yl)-1H-1,2,4-triazol-3-yl]ethyl}[1,2,4]triazolo[1,5-c]pyrimidine | n/a | |
| 240 | Q9Y233_JKO | JKO | n/a | 51034710 | CHEMBL2180796 | 1-methyl-4-(morpholine-4-carbonyl)-N-[(4R)-2-phenylimidazo[1,2-a]pyridin-7-yl]-1H-pyrazole-5-carboxamide | n/a | |
| 241 | Q9Y233_JKX | JKX | n/a | 1486289 | n/a | 1-(6-fluoropyridin-2-yl)piperidin-4-one | n/a | |
| 242 | Q9Y233_JL6 | JL6 | n/a | 165368519 | n/a | 6-cyclopropyl-N-[(3R)-1-(pyridin-2-yl)pyrrolidin-3-yl]-3-[(pyrimidin-5-yl)amino]pyridine-2-carboxamide | n/a | |
| 243 | Q9Y233_JLI | JLI | n/a | 67391850 | n/a | 1-methyl-5-{[(4R)-2-phenylimidazo[1,2-a]pyrimidin-7-yl]carbamoyl}-1H-pyrazole-4-carboxylic acid | n/a | |
| 244 | Q9Y233_JLR | JLR | n/a | 59369972 | n/a | 3-[1-(naphthalen-1-yl)-1H-pyrazol-5-yl]-1-[3-(trifluoromethoxy)phenyl]pyridazin-4(1H)-one | n/a | |
| 245 | Q9Y233_JM0 | JM0 | n/a | 23624262 | CHEMBL1085374 | N-[(10S)-2-methoxy-7-methyl-9-propylimidazo[1,5-a]pyrido[3,2-e]pyrazin-6-yl]methanesulfonamide | n/a | |
| 246 | Q9Y233_JME | JME | n/a | 51035025 | n/a | 4-(azetidine-1-carbonyl)-N-[(4R)-6-cyano-2-phenylimidazo[1,2-a]pyridin-7-yl]-1-methyl-1H-pyrazole-5-carboxamide | n/a | |
| 247 | Q9Y233_JML | JML | n/a | 165368520 | n/a | 2-benzyl-6,6-dimethyl-1H-imidazo[4,5-h]isoquinoline-7,9(6H,8H)-dione | n/a | |
| 248 | Q9Y233_JMU | JMU | n/a | 165368521 | n/a | N-[(4R)-6-cyano-2-phenylimidazo[1,2-a]pyridin-7-yl]-1-methyl-4-(morpholine-4-carbonyl)-1H-pyrazole-3-carboxamide | n/a | |
| 249 | Q9Y233_JN6 | JN6 | n/a | 53467162 | n/a | N~4~-(2-hydroxyethyl)-1-methyl-N~5~-[(4R)-2-phenylimidazo[1,2-a]pyrimidin-7-yl]-1H-pyrazole-4,5-dicarboxamide | n/a | |
| 250 | Q9Y233_JNL | JNL | n/a | 1072886 | CHEMBL1587056 | N-(2,3-dimethylquinoxalin-6-yl)-N'-(3-methoxyphenyl)urea | n/a | |
| 251 | Q9Y233_JNU | JNU | n/a | 75201355 | n/a | (4R)-3-methyl-6-{2-[1-methyl-3-(pyrrolidin-1-yl)-1H-1,2,4-triazol-5-yl]ethyl}-2-(trifluoromethyl)imidazo[1,2-b]pyridazine | n/a | |
| 252 | Q9Y233_JO6 | JO6 | n/a | 165368522 | n/a | (4S)-6,8-dichloro-2-[2-(5-chloro-1,3-benzothiazol-2-yl)ethyl]-5-methyl[1,2,4]triazolo[1,5-a]pyridine | n/a | |
| 253 | Q9Y233_JOF | JOF | n/a | 165368523 | n/a | 5-chloro-8-hydroxy-2-methyl-1,4-dihydropyrrolo[3,4-b]indol-3(2H)-one | n/a | |
| 254 | Q9Y233_JOO | JOO | n/a | 46218712 | n/a | 3-[1-(2,5-difluorophenyl)-1H-pyrazol-5-yl]-1-[3-(methanesulfonyl)phenyl]pyridazin-4(1H)-one | n/a | |
| 255 | Q9Y233_JP0 | JP0 | n/a | 1454116;135429163; | n/a | N-[(4-methoxyphenyl)methyl]-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-N'-phenylurea | n/a | |
| 256 | Q9Y233_JPF | JPF | n/a | 165368524 | n/a | 6-[(3-methylphenyl)sulfanyl]-2-[4-(pyridin-2-yl)piperazin-1-yl]-9H-purine | n/a | |
| 257 | Q9Y233_JPU | JPU | DB08811 | 5502 | CHEMBL404216 | (5R)-1-(3,4-dimethoxyphenyl)-5-ethyl-7,8-dimethoxy-4-methyl-5H-2,3-benzodiazepine | inhibitor | |
| 258 | Q9Y233_JPZ | JPZ | n/a | 63112;5320866;135408753; | CHEMBL266540 | quinazolin-4(1H)-one | n/a | |
| 259 | Q9Y233_JQ3 | JQ3 | n/a | 165368525 | n/a | 5-(cyclopentylmethoxy)pyrimidin-2-amine | n/a | |
| 260 | Q9Y233_JQC | JQC | n/a | 165368526 | n/a | 4-chloro-N-[2-(3,5-dimethylphenyl)-1H-benzimidazol-5-yl]-1-methyl-1H-pyrazole-5-carboxamide | n/a | |
| 261 | Q9Y233_JQL | JQL | n/a | n/a | n/a | 1-methyl-4-[(2R)-2-methylpyrrolidine-1-carbonyl]-N-[(4R)-2-phenylimidazo[1,2-a]pyridin-7-yl]-1H-pyrazole-5-carboxamide | n/a | |
| 262 | Q9Y233_JQU | JQU | n/a | 165368528 | n/a | N-[3-methyl-1-(pyridin-2-yl)-1H-thieno[2,3-c]pyrazol-5-yl]benzamide | n/a | |
| 263 | Q9Y233_JRC | JRC | n/a | 165368527 | n/a | 1-methyl-4-[(2R)-2-methylpyrrolidine-1-carbonyl]-N-[(4R)-2-phenylimidazo[1,2-a]pyridin-7-yl]-1H-pyrazole-5-carboxamide | n/a | |
| 264 | Q9Y233_JRL | JRL | n/a | 53467159 | n/a | 4-(azetidine-1-carbonyl)-1-methyl-N-[(4R)-2-phenylimidazo[1,2-a]pyrimidin-7-yl]-1H-pyrazole-5-carboxamide | n/a | |
| 265 | Q9Y233_JRX | JRX | n/a | 165368529 | n/a | 2-ethyl-3-[4-(4-methylbenzene-1-sulfonyl)piperazin-1-yl]quinoxaline | n/a | |
| 266 | Q9Y233_JSF | JSF | n/a | 53466711 | n/a | 3,6-dimethyl-N-[(4R)-2-phenylimidazo[1,2-a]pyrimidin-7-yl]pyridine-2-carboxamide | n/a | |
| 267 | Q9Y233_JSM | JSM | n/a | 51034254 | n/a | N~4~,1-dimethyl-N~4~-[2-(methylamino)ethyl]-N~5~-[(4R)-2-phenylimidazo[1,2-a]pyridin-7-yl]-1H-pyrazole-4,5-dicarboxamide | n/a | |
| 268 | Q9Y233_JSY | JSY | n/a | 6950411 | n/a | 6-methyl-N-(4-methylphenyl)pyrimidin-4-amine | n/a | |
| 269 | Q9Y233_JT9 | JT9 | n/a | 165368530 | n/a | 3-{2-[(4S)-6,8-dichloro-5-methyl[1,2,4]triazolo[1,5-a]pyridin-2-yl]ethyl}quinoxalin-2(1H)-one | n/a | |
| 270 | Q9Y233_JTL | JTL | n/a | 736232 | CHEMBL4580935 | N-[(thiophen-2-yl)methyl]quinoxaline-6-carboxamide | n/a | |
| 271 | Q9Y233_JTX | JTX | n/a | 165368531 | n/a | (4S)-5-methyl-2-{2-[1-methyl-3-(pyrrolidin-1-yl)-1H-1,2,4-triazol-5-yl]ethyl}-8-(trifluoromethyl)[1,2,4]triazolo[1,5-c]pyrimidine | n/a | |
| 272 | Q9Y233_JU6 | JU6 | n/a | 76026103 | n/a | (8S)-5-[(3S)-3-fluoropyrrolidin-1-yl]-2-(3-methylquinoxalin-2-yl)-N-(oxan-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine | n/a | |
| 273 | Q9Y233_JUC | JUC | n/a | 77745997 | CHEMBL5315514 | (8R)-5-[(3R)-3-fluoropyrrolidin-1-yl]-N-methyl-2-(3-methylquinoxalin-2-yl)-N-(oxan-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine | n/a | |
| 274 | Q9Y233_JWC | JWC | n/a | 165368532 | n/a | 6-cyclopropyl-3-methoxy-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyrazine-2-carboxamide | n/a | |
| 275 | Q9Y233_JWJ | JWJ | n/a | 165368533 | n/a | 7-[(3,5-dimethyl-4-propan-2-yloxy-pyridin-2-yl)methyl-oxidanyl-$l^{3}-sulfanyl]-8~{H}-imidazo[4,5-g][1,3]benzothiazole | n/a | |
| 276 | Q9Y233_JWR | JWR | n/a | 165368534 | n/a | 2,3-dichloro-N-[(4S)-2-phenyl[1,2,4]triazolo[1,5-a]pyridin-7-yl]pyridine-4-carboxamide | n/a | |
| 277 | Q9Y233_JX0 | JX0 | n/a | 2004610 | n/a | [1-(4-chlorophenyl)-3-methyl-1H-thieno[2,3-c]pyrazol-5-yl](piperidin-1-yl)methanone | n/a | |
| 278 | Q9Y233_JX9 | JX9 | n/a | 2155057 | CHEMBL4928131 | N-cyclohexyl-N-methyl-7H-purin-6-amine | n/a | |
| 279 | Q9Y233_JXI | JXI | n/a | n/a | n/a | 1-methyl-6-{2-[(4R)-1-methyl-4-phenyl-4,5-dihydro-1H-imidazol-2-yl]ethyl}-1,2,3,5-tetrahydro-4H-pyrazolo[3,4-d]pyrimidin-4-one | n/a | |
| 280 | Q9Y233_JXO | JXO | n/a | 13532735 | n/a | 6-chloroquinoxalin-2-amine | n/a | |
| 281 | Q9Y233_JXX | JXX | n/a | 2338466 | n/a | 2-chloro-4-(morpholin-4-yl)quinazoline | n/a | |
| 282 | Q9Y233_JY3 | JY3 | n/a | 165368536 | n/a | 7-[({5-methyl-4-[(propan-2-yl)oxy]pyridin-2-yl}methyl)sulfanyl]-8H-imidazo[4,5-g][1,3]benzothiazole | n/a | |
| 283 | Q9Y233_JY4 | JY4 | n/a | 3814427;6413369; | CHEMBL4534373 | 7,8-dimethoxy-1-methyl-2H-pyrazolo[3,4-c]cinnoline | n/a | |
| 284 | Q9Y233_JY7 | JY7 | n/a | 73387743 | CHEMBL4456157 | 8-fluoro-6-methoxy-3-methyl-1-(3-methylpyridin-4-yl)-3H-pyrazolo[3,4-c]cinnoline | n/a | |
| 285 | Q9Y233_JYA | JYA | n/a | 24805199 | CHEMBL1086265 | (10S)-2-methoxy-7-methyl-9-propylimidazo[1,5-a]pyrido[3,2-e]pyrazine-6-carbonitrile | n/a | |
| 286 | Q9Y233_JYL | JYL | n/a | 165368537 | n/a | (4S)-N-[2-(1-methyl-4-phenyl-1H-imidazol-2-yl)ethyl]-3-(propan-2-yl)[1,2,4]triazolo[4,3-a]pyridine-8-carboxamide | n/a | |
| 287 | Q9Y233_JYU | JYU | n/a | 165368538 | n/a | N-(1-tert-butyl-3-methyl-1H-pyrazol-5-yl)-1-phenyl-3-{[(pyridin-2-yl)oxy]methyl}-1H-thieno[2,3-c]pyrazole-5-carboxamide | n/a | |
| 288 | Q9Y233_K | K | n/a | 813 | CHEMBL1233793 | POTASSIUM ION | n/a | |
| 289 | Q9Y233_K0C | K0C | n/a | 165368539 | n/a | 2-{[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]sulfanyl}-1H-imidazo[4,5-f]quinoline | n/a | |
| 290 | Q9Y233_K0R | K0R | n/a | 67384369 | n/a | 4-chloro-1,3-dimethyl-N-[(4R)-2-phenylimidazo[1,2-a]pyrimidin-7-yl]-1H-pyrazole-5-carboxamide | n/a | |
| 291 | Q9Y233_K18 | K18 | n/a | 165368540 | n/a | N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N'-(1-phenyl-1H-pyrazol-5-yl)urea | n/a | |
| 292 | Q9Y233_K1I | K1I | n/a | 59370144 | n/a | 3-[1-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-1H-pyrazol-5-yl]-1-[3-(methanesulfonyl)phenyl]pyridazin-4(1H)-one | n/a | |
| 293 | Q9Y233_K1X | K1X | n/a | 59370001 | n/a | 3-[1-(quinolin-4-yl)-1H-pyrazol-5-yl]-1-[3-(trifluoromethoxy)phenyl]pyridazin-4(1H)-one | n/a | |
| 294 | Q9Y233_K2L | K2L | n/a | 118111828 | n/a | 1-(2-{2-[(4S)-5,8-dimethyl[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl}-1-methyl-1H-imidazol-4-yl)pyrrolidin-2-one | n/a | |
| 295 | Q9Y233_K3F | K3F | n/a | 3147227 | CHEMBL1779658 | 4-chloro-1-methyl-N-(2-phenyl-1H-benzimidazol-5-yl)-1H-pyrazole-5-carboxamide | n/a | |
| 296 | Q9Y233_K3O | K3O | n/a | 165368541 | n/a | N~4~-ethyl-5-[3-(trifluoromethyl)phenyl]-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine | n/a | |
| 297 | Q9Y233_K40 | K40 | n/a | 665194 | CHEMBL1345945 | 5,8-dichloro-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-one | n/a | |
| 298 | Q9Y233_K49 | K49 | n/a | 70098086 | CHEMBL3685495 | 6-cyclopropyl-N-{4-[(2-hydroxy-2-methylpropyl)carbamoyl]pyridin-3-yl}-3-[(pyrimidin-5-yl)amino]pyridine-2-carboxamide | n/a | |
| 299 | Q9Y233_K4L | K4L | n/a | n/a | n/a | (5S)-5-(2-phenylethyl)[3,4'-bipyridin]-6(5H)-one | n/a | |
| 300 | Q9Y233_K4U | K4U | n/a | n/a | n/a | 6-cyclopropyl-N-{(4S)-4-[(piperidin-1-yl)methyl]-4,5-dihydro-1,3-thiazol-2-yl}-3-[(pyrimidin-5-yl)amino]pyrazine-2-carboxamide | n/a | |
| 301 | Q9Y233_K5F | K5F | n/a | 51033482 | CHEMBL2180795 | N~4~,N~4~,1-trimethyl-N~5~-[(4R)-2-phenylimidazo[1,2-a]pyridin-7-yl]-1H-pyrazole-4,5-dicarboxamide | n/a | |
| 302 | Q9Y233_K5R | K5R | n/a | 54760756 | CHEMBL3685450 | 6-cyclopropyl-N-[4-(dimethylcarbamoyl)pyridin-3-yl]-3-[(pyrimidin-5-yl)amino]pyridine-2-carboxamide | n/a | |
| 303 | Q9Y233_K63 | K63 | n/a | 11698194 | CHEMBL248380 | N-[3-cyano-2-(2'-ethoxy[1,1'-biphenyl]-4-yl)-6-fluoroquinolin-4-yl]-D-alanine | n/a | |
| 304 | Q9Y233_K6F | K6F | n/a | 236280 | CHEMBL1707141 | 6-chloro-2,3-dimethylquinoxaline | n/a | |
| 305 | Q9Y233_K6O | K6O | n/a | 165368544 | n/a | ethyl [(4-{[4-(azetidine-1-carbonyl)-1-methyl-1H-pyrazole-5-carbonyl]amino}-6-methylpyridin-2-yl)carbamothioyl]carbamate | n/a | |
| 306 | Q9Y233_K79 | K79 | n/a | 59370140 | n/a | 3-[1-(2,4-difluorophenyl)-1H-pyrazol-5-yl]-1-[3-(trifluoromethoxy)phenyl]pyridazin-4(1H)-one | n/a | |
| 307 | Q9Y233_K7O | K7O | n/a | 165368545 | n/a | (4R)-6,8-dichloro-2-[2-(6,7-dimethyl-1H-benzimidazol-2-yl)ethyl]-5-methyl[1,2,4]triazolo[1,5-a]pyridine | n/a | |
| 308 | Q9Y233_K9F | K9F | n/a | 165368547 | n/a | 5-[2-(1-methyl-4-phenyl-1H-imidazol-2-yl)ethyl]quinoxaline | n/a | |
| 309 | Q9Y233_K9O | K9O | n/a | 165368548 | n/a | 4-chloro-1-(2-methylpropyl)-N-(2-phenyl-1H-benzimidazol-6-yl)-1H-pyrazole-5-carboxamide | n/a | |
| 310 | Q9Y233_K9X | K9X | n/a | 67388402 | n/a | 4-bromo-1,3-dimethyl-N-[(4R)-2-phenylimidazo[1,2-a]pyrimidin-7-yl]-1H-pyrazole-5-carboxamide | n/a | |
| 311 | Q9Y233_KA6 | KA6 | n/a | 57378288 | n/a | 1-methyl-4-(morpholine-4-carbonyl)-N-[(4S)-2-(pyrrolidin-1-yl)[1,2,4]triazolo[1,5-a]pyridin-7-yl]-1H-pyrazole-5-carboxamide | n/a | |
| 312 | Q9Y233_KAU | KAU | n/a | 165368549 | n/a | N-[(3R)-1-(5-chloropyridin-2-yl)pyrrolidin-3-yl]-1-methyl-4-(pyridin-4-yl)-1H-pyrazole-3-carboxamide | n/a | |
| 313 | Q9Y233_KB6 | KB6 | n/a | 165368550 | n/a | 3-{2-[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]ethoxy}isoquinoline | n/a | |
| 314 | Q9Y233_KBL | KBL | n/a | 165368551 | n/a | 6-methyl-3-(1-phenyl-1H-pyrazol-5-yl)-1-[3-(trifluoromethoxy)phenyl]pyridazin-4(1H)-one | n/a | |
| 315 | Q9Y233_KC9 | KC9 | n/a | 165368552 | n/a | 4-(azetidine-1-carbonyl)-N-[3-(1,3-benzoxazol-2-yl)phenyl]-1-methyl-1H-pyrazole-5-carboxamide | n/a | |
| 316 | Q9Y233_KCF | KCF | n/a | 67775541 | n/a | 4-bromanyl-~{N},~{N}-dimethyl-1$l^{4},7,9-triazabicyclo[4.3.0]nona-1,3,5-trien-8-amine | n/a | |
| 317 | Q9Y233_KCU | KCU | n/a | 165368553 | n/a | 4-chloro-N-(2-phenyl-1H-benzimidazol-5-yl)-1-propyl-1H-pyrazole-5-carboxamide | n/a | |
| 318 | Q9Y233_KD4 | KD4 | n/a | 89428907 | n/a | 2-chloro-5-methoxy-3-methylquinoxaline | n/a | |
| 319 | Q9Y233_KDC | KDC | n/a | 165368554 | n/a | 7-{[(4-ethoxy-5-methylpyridin-2-yl)methyl]sulfanyl}-8H-imidazo[4,5-g][1,3]benzothiazole | n/a | |
| 320 | Q9Y233_KDX | KDX | n/a | 944145;135448689; | CHEMBL1592850 | 9-methoxy-3,5-dihydro-4H-pyrimido[5,4-b]indol-4-one | n/a | |
| 321 | Q9Y233_KE6 | KE6 | n/a | 165368555 | n/a | 6-methyl-N-[1-(propan-2-yl)-1H-pyrazol-3-yl]-3-[(pyrimidin-5-yl)amino]pyridine-2-carboxamide | n/a | |
| 322 | Q9Y233_KER | KER | n/a | 59369999 | n/a | 3-[1-(2,5-difluorophenyl)-1H-pyrazol-5-yl]-1-[3-(trifluoromethoxy)phenyl]pyridazin-4(1H)-one | n/a | |
| 323 | Q9Y233_KF3 | KF3 | n/a | 165368557 | n/a | 2-tert-butyl-5-[(pyrimidin-5-yl)amino]-N-[3-(trifluoromethoxy)phenyl]pyrimidine-4-carboxamide | n/a | |
| 324 | Q9Y233_KF9 | KF9 | n/a | 59370047 | n/a | 3-{5-[1-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-4-oxo-1,4-dihydropyridazin-3-yl]-1H-pyrazol-1-yl}benzonitrile | n/a | |
| 325 | Q9Y233_KFI | KFI | n/a | 165368559 | n/a | 2-chloro-6-(cyclopropylamino)-N-[(4S)-2-phenyl[1,2,4]triazolo[1,5-a]pyridin-7-yl]pyridine-4-carboxamide | n/a | |
| 326 | Q9Y233_KFO | KFO | n/a | 59370137 | n/a | 3-[1-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-[3-(trifluoromethoxy)phenyl]pyridazin-4(1H)-one | n/a | |
| 327 | Q9Y233_KFX | KFX | n/a | 165368560 | n/a | N-{[(4R)-5,8-dimethyl[1,2,4]triazolo[1,5-a]pyrazin-2-yl]methyl}-1-methyl-3-phenyl-1H-1,2,4-triazol-5-amine | n/a | |
| 328 | Q9Y233_KG3 | KG3 | n/a | 165368561 | n/a | 6-cyclopropyl-N-{2-[2-(methylamino)-2-oxoethyl]phenyl}-3-[(pyrimidin-5-yl)amino]pyridine-2-carboxamide | n/a | |
| 329 | Q9Y233_KGO | KGO | n/a | 54761122 | CHEMBL3685578 | N-[1-methyl-5-(methylcarbamoyl)-1H-pyrazol-4-yl]-6-[(3S)-oxolan-3-yl]-3-[(pyrimidin-5-yl)amino]pyrazine-2-carboxamide | n/a | |
| 330 | Q9Y233_KH6 | KH6 | n/a | 51034818 | n/a | N-[(4R)-6-cyano-2-phenylimidazo[1,2-a]pyridin-7-yl]-1-methyl-4-(morpholine-4-carbonyl)-1H-pyrazole-5-carboxamide | n/a | |
| 331 | Q9Y233_KHI | KHI | n/a | n/a | n/a | 6-chloro-N,N-dimethyl-2-{2-[(3S)-1-(pyridin-2-yl)pyrrolidin-3-yl]ethyl}quinazolin-4-amine | n/a | |
| 332 | Q9Y233_KHU | KHU | n/a | 46218709 | n/a | N-(3-{3-[1-(2-fluorophenyl)-1H-pyrazol-5-yl]-4-oxopyridazin-1(4H)-yl}phenyl)acetamide | n/a | |
| 333 | Q9Y233_KI4 | KI4 | n/a | 165368563 | n/a | N-{3-[(4R)-imidazo[1,2-a]pyridin-2-yl]phenyl}-1-methyl-3-[(pyrimidin-5-yl)amino]-1H-pyrazole-4-carboxamide | n/a | |
| 334 | Q9Y233_KI8 | KI8 | n/a | 2030782 | n/a | [4-(2-methoxyphenyl)piperazin-1-yl](3-methyl-1-phenyl-1H-thieno[2,3-c]pyrazol-5-yl)methanone | n/a | |
| 335 | Q9Y233_KIE | KIE | n/a | 165368564 | n/a | N-ethyl-6-[(4-fluorophenyl)sulfanyl]-N-methyl-7H-purin-2-amine | n/a | |
| 336 | Q9Y233_KII | KII | n/a | 165368565 | n/a | 1-methyl-N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]-4-(pyridin-4-yl)-1H-pyrazole-3-carboxamide | n/a | |
| 337 | Q9Y233_KIS | KIS | n/a | 165368566 | n/a | diethyl 1,1'-[oxydi(3,1-phenylene)]bis(5-methyl-1H-imidazole-4-carboxylate) | n/a | |
| 338 | Q9Y233_KIY | KIY | n/a | 18452840 | n/a | 7-(cyclopropylmethoxy)-2-methyl-4-(pyrrolidin-1-yl)quinazoline | n/a | |
| 339 | Q9Y233_KJ3 | KJ3 | n/a | 165368567 | n/a | (2S)-3-(4-{2-[2-(2-ethoxy-4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]ethoxy}naphthalen-1-yl)-2-methoxypropanoic acid | n/a | |
| 340 | Q9Y233_KJC | KJC | n/a | 58548230 | CHEMBL3685469 | 6-cyclopropyl-N-{3-[(2-hydroxy-2-methylpropyl)carbamoyl]-1-methyl-1H-pyrazol-4-yl}-3-[(pyrimidin-5-yl)amino]pyridine-2-carboxamide | n/a | |
| 341 | Q9Y233_LKF | LKF | n/a | 67458671 | CHEMBL3262043 | 4-[3-[1-[(2S)-2-methoxypropyl]pyrazol-4-yl]-2-methyl-imidazo[1,2-a]pyrazin-8-yl]morpholine | n/a | |
| 342 | Q9Y233_MEW | MEW | n/a | 15674;135400457; | CHEMBL395092 | 2-methylquinazolin-4(3H)-one | n/a | |
| 343 | Q9Y233_MG | MG | n/a | 888 | n/a | MAGNESIUM ION | n/a | |
| 344 | Q9Y233_MRW | MRW | n/a | 66593 | CHEMBL1409793 | 7-chloroquinolin-4-ol | n/a | |
| 345 | Q9Y233_NI | NI | n/a | 934 | n/a | NICKEL (II) ION | n/a | |
| 346 | Q9Y233_P98 | P98 | n/a | 72193890 | CHEMBL3091492 | 2-({[1-phenyl-2-(propan-2-yl)-1H-benzimidazol-6-yl]oxy}methyl)quinoline | n/a | |
| 347 | Q9Y233_PF9 | PF9 | DB08387 | 11581936 | CHEMBL562318 | 2-{[4-(1-methyl-4-pyridin-4-yl-1H-pyrazol-3-yl)phenoxy]methyl}quinoline | inhibitor | IC50(nM) = 0.18 |
| 348 | Q9Y233_PG4 | PG4 | n/a | 8200 | CHEMBL1235254 | TETRAETHYLENE GLYCOL | n/a | |
| 349 | Q9Y233_PO4 | PO4 | DB14523 | 1061 | n/a | PHOSPHATE ION | n/a | |
| 350 | Q9Y233_PR | PR | n/a | 185491 | n/a | PRASEODYMIUM ION | n/a | |
| 351 | Q9Y233_S9I | S9I | DB19153 | 71271414 | CHEMBL5314924 | 2-methyl-6-{[(1S,2S)-2-(5-methylpyridin-2-yl)cyclopropyl]methoxy}-N-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]pyrimidin-4-amine | n/a | |
| 352 | Q9Y233_SO4 | SO4 | DB14546 | 1117 | n/a | SULFATE ION | n/a | |
| 353 | Q9Y233_WP3 | WP3 | n/a | 67387846 | n/a | N~5~-[(2P,4S)-2-(3-fluorophenyl)imidazo[1,2-a]pyrimidin-7-yl]-N~4~,N~4~,1-trimethyl-1H-pyrazole-4,5-dicarboxamide | n/a | |
| 354 | Q9Y233_X4C | X4C | n/a | 74049853 | CHEMBL3288410 | 8-methyl-6-[2-(5-methyl-1-phenyl-1H-benzimidazol-2-yl)ethyl]imidazo[1,5-a]pyrimidine | n/a | |
| 355 | Q9Y233_X4D | X4D | n/a | 74049854 | CHEMBL3288411 | 7-[2-(5-methyl-1-phenyl-1H-benzimidazol-2-yl)ethyl]imidazo[1,5-b]pyridazine | n/a | |
| 356 | Q9Y233_Z73 | Z73 | n/a | 24802717 | CHEMBL1086110 | 2-methoxy-6,7-dimethyl-9-propylimidazo[1,5-a]pyrido[3,2-e]pyrazine | n/a | |
| 357 | Q9Y233_ZN | ZN | n/a | 32051 | CHEMBL1236970 | ZINC ION | n/a | |
| 358 | Q9Y233_H9F | H9F | DB00975 | 3108 | CHEMBL932 | Dipyridamole | inhibitor | Ki(nM) = 1000.0 |
| 359 | Q9Y233_PF4 | PF4 | DB08383 | 1122713 | CHEMBL1235237 | 4,5-bis(4-methoxyphenyl)-2-thiophen-2-yl-1H-imidazole | n/a | IC50(nM) = 35.0 |
| 360 | Q9Y233_PF6 | PF6 | DB08384 | 44141871 | CHEMBL562317 | 2-({4-[4-(pyridin-4-ylmethyl)-1H-pyrazol-3-yl]phenoxy}methyl)quinoline | n/a | |
| 361 | Q9Y233_PF8 | PF8 | DB08386 | 11610553 | CHEMBL560377 | 2-{[4-(4-pyridin-4-yl-1H-pyrazol-3-yl)phenoxy]methyl}quinoline | n/a | |
| 362 | Q9Y233_PFH | PFH | DB08389 | 15991588 | CHEMBL410834 | 6,7-DIMETHOXY-4-[(3R)-3-(2-NAPHTHYLOXY)PYRROLIDIN-1-YL]QUINAZOLINE | n/a | Ki(nM) = 12.0 |
| 363 | Q9Y233_PFJ | PFJ | DB08391 | 11955614 | CHEMBL219445 | PQ-10 | n/a | Ki(nM) = 4.0 IC50(nM) = 6.0 |
| 364 | Q9Y233_DB08814 | n/a | DB08814 | n/a | n/a | Triflusal | antagonist |