Gene name: CYSLTR1
Protein name: Cysteinyl leukotriene receptor
List of molecules and drugs that interact with protein Q9Y271
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | Q9Y271_1PE | 1PE | n/a | 62551 | CHEMBL1229766 | PENTAETHYLENE GLYCOL | n/a | |
2 | Q9Y271_KNT | KNT | DB01411 | 4887 | CHEMBL21333 | pranlukast | antagonist | |
3 | Q9Y271_NA | NA | n/a | 923 | n/a | SODIUM ION | n/a | |
4 | Q9Y271_OLA | OLA | n/a | 445639 | CHEMBL8659 | OLEIC ACID | n/a | |
5 | Q9Y271_OLC | OLC | n/a | 11451146 | n/a | (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate | n/a | |
6 | Q9Y271_ZLK | ZLK | DB00549 | 5717 | CHEMBL603 | zafirlukast | antagonist | Ki(nM) = 0.26 IC50(nM) = 0.26 |
7 | Q9Y271_MTK | MTK | DB00471 | 5281040 | CHEMBL787 | Montelukast | antagonist | IC50(nM) = 0.43 EC50(nM) = 72.0 |
8 | Q9Y271_DB00587 | n/a | DB00587 | n/a | n/a | Cinalukast | antagonist | |
9 | Q9Y271_DB00716 | n/a | DB00716 | n/a | n/a | Nedocromil | antagonist | |
10 | Q9Y271_LTX | LTX | DB08855 | 5280493 | CHEMBL451509 | Leukotriene C4 | agonist | |
11 | Q9Y271_HQE | HQE | DB09526 | 785;152743433; | CHEMBL537 | Hydroquinone | activator | |
12 | Q9Y271_LTD | LTD | DB11858 | 5280878 | CHEMBL288943 | Leukotriene D4 | agonist |