Gene name: HRH3
Protein name: Histamine H3 receptor
List of molecules and drugs that interact with protein Q9Y5N1
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | Q9Y5N1_1IB | 1IB | DB12201 | n/a | CHEMBL2151197 | N-ethyl-3-fluoranyl-3-[3-fluoranyl-4-(pyrrolidin-1-ylmethyl)phenyl]cyclobutane-1-carboxamide | n/a | |
2 | Q9Y5N1_CLR | CLR | DB04540 | 5997 | CHEMBL112570 | CHOLESTEROL | n/a | |
3 | Q9Y5N1_DB00768 | n/a | DB00768 | n/a | n/a | Olopatadine | antagonist | |
4 | Q9Y5N1_9SC | 9SC | DB01238 | 60795 | CHEMBL1112 | Aripiprazole | ligand | Ki(nM) = 2361.0 |
5 | Q9Y5N1_HSM | HSM | DB05381 | 774 | CHEMBL90 | Histamine | agonist | |
6 | Q9Y5N1_DB06698 | n/a | DB06698 | n/a | n/a | Betahistine | antagonist | |
7 | Q9Y5N1_DB11642 | n/a | DB11642 | n/a | n/a | Pitolisant | antagonist |