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(14beta,17alpha)-17-ethynyl-17-hydroxyestr-4-en-3-one

P06401 — Progesterone receptor

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Attributes

UniProt ID
P06401
Protein Name
Progesterone receptor
Ligand Name
(14beta,17alpha)-17-ethynyl-17-hydroxyestr-4-en-3-one
DrugBank ID
DB00717
PDB Ligand Accession
NDR
ChEMBL ID
CHEMBL1162
PubChem ID
6230
InChIKey
VIKNJXKGJWUCNN-XGXHKTLJSA-N
SMILES
CC12CCC3C(C1CCC2(C#C)O)CCC4=CC(=O)CCC34
Drug Action
agonist
Affinity Metrics
ki:1.9 nM
ic50:3.2 nM
kd:0.4 nM
ec50:2.2 nM