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(17BETA)-17-HYDROXY-17-METHYLESTRA-4,9,11-TRIEN-3-ONE

P10275 — Androgen receptor

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Attributes

UniProt ID
P10275
Protein Name
Androgen receptor
Ligand Name
(17BETA)-17-HYDROXY-17-METHYLESTRA-4,9,11-TRIEN-3-ONE
DrugBank ID
DB02998
PDB Ligand Accession
R18
ChEMBL ID
CHEMBL166444
PubChem ID
261000
InChIKey
CCCIJQPRIXGQOE-XWSJACJDSA-N
SMILES
CC1(CCC2C1(C=CC3=C4CCC(=O)C=C4CCC23)C)O
Drug Action
activator
Affinity Metrics
ki:0.4 nM
ic50:0.302 nM
kd:0.52 nM
ec50:0.013 nM